BDBM50406795 Cozaar LOSARTAN POTASSIUM
BDBM50422638 Losartan 5-(Nitrooxy)Pentanoate CHEMBL360220
Losartan CAS_114798-26-4 NSC_3961 BDBM82258
BDBM50422637 Losartan 3-[(Nitrooxy)Methyl]Benzoate CHEMBL186572
US9527857, M BDBM253921 US9464092, M
BDBM204122 US9539260, M US9763952, Example M
BDBM256611 US9790174, Example 85(m) US10435361, Example 85(m) US9481648, 85(m)
US11267820, Compound m US10689395, Compound m BDBM448086
1,3-xylene 1,3-Dimethylbenzol m-methyltoluene BDBM50008556 m-xylene CHEMBL286727 m-Xylol 3-xylene meta-xylene m-dimethylbenzene
- Segarra, V; Crespo, MI; Pujol, F; Beleta, J; Doménech, T; Miralpeix, M; Palacios, JM; Castro, A; Martinez, A Phosphodiesterase inhibitory properties of losartan. Design and synthesis of new lead compounds. Bioorg Med Chem Lett 8: 505-10 (1998)
- Ono, K; Ueda, H; Yoshizawa, Y; Akazawa, D; Tanimura, R; Shimada, I; Takahashi, H Structural basis for platelet antiaggregation by angiotensin II type 1 receptor antagonist losartan (DuP-753) via glycoprotein VI. J Med Chem 53: 2087-93 (2010)
- Kim, TW; Yoo, BW; Lee, JK; Kim, JH; Lee, KT; Chi, YH; Lee, JY Synthesis and antihypertensive activity of pyrimidin-4(3H)-one derivatives as losartan analogue for new angiotensin II receptor type 1 (AT1) antagonists. Bioorg Med Chem Lett 22: 1649-54 (2012)
- Armani, E; Rizzi, A; Capaldi, C; De Fanti, R; Delcanale, M; Villetti, G; Marchini, G; Pisano, AR; Pitozzi, V; Pittelli, MG; Trevisani, M; Salvadori, M; Cenacchi, V; Puccini, P; Amadei, F; Pappani, A; Civelli, M; Patacchini, R; Baker-Glenn, CAG; Van de Poël, H; Blackaby, WP; Nash, K; Amari, G Discovery of M J Med Chem 64: 9100-9119 (2021)
- Poslusney, MS; Salovich, JM; Wood, MR; Melancon, BJ; Bollinger, KA; Luscombe, VB; Rodriguez, AL; Engers, DW; Bridges, TM; Niswender, CM; Conn, PJ; Lindsley, CW Novel M Bioorg Med Chem Lett 29: 362-366 (2019)
- Melancon, BJ; Wood, MR; Noetzel, MJ; Nance, KD; Engelberg, EM; Han, C; Lamsal, A; Chang, S; Cho, HP; Byers, FW; Bubser, M; Jones, CK; Niswender, CM; Wood, MW; Engers, DW; Wu, D; Brandon, NJ; Duggan, ME; Conn, PJ; Bridges, TM; Lindsley, CW Optimization of M Bioorg Med Chem Lett 27: 2296-2301 (2017)
- A M Subbaiah, M; Mandlekar, S; Desikan, S; Ramar, T; Subramani, L; Annadurai, M; Desai, SD; Sinha, S; Jenkins, SM; Krystal, MR; Subramanian, M; Sridhar, S; Padmanabhan, S; Bhutani, P; Arla, R; Singh, S; Sinha, J; Thakur, M; Kadow, JF; Meanwell, NA J Med Chem 62: 3553-3574 (2019)
- Hedner, E; Sjögren, M; Frändberg, PA; Johansson, T; Göransson, U; Dahlström, M; Jonsson, P; Nyberg, F; Bohlin, L J Nat Prod 69: 1421-4 (2006)
- Karlberg, T; Markova, N; Johansson, I; Hammarström, M; Schütz, P; Weigelt, J; Schüler, H J Med Chem 53: 5352-5 (2010)
- Delouvrié, B; Al-Kadhimi, K; Arnould, JC; Barry, ST; Cross, DA; Didelot, M; Gavine, PR; Germain, H; Harris, CS; Hughes, AM; Jude, DA; Kendrew, J; Lambert-van der Brempt, C; Lohmann, JJ; Ménard, M; Mortlock, AA; Pass, M; Rooney, C; Vautier, M; Vincent, JL; Warin, N Bioorg Med Chem Lett 22: 4111-6 (2012)
- Dannhardt, G; Plutizki, S; Kramb, J; Müller, A; Möhler, M US Patent US9364459 (2016)
- Vasbinder, MM; Aquila, B; Augustin, M; Chen, H; Cheung, T; Cook, D; Drew, L; Fauber, BP; Glossop, S; Grondine, M; Hennessy, E; Johannes, J; Lee, S; Lyne, P; Mörtl, M; Omer, C; Palakurthi, S; Pontz, T; Read, J; Sha, L; Shen, M; Steinbacher, S; Wang, H; Wu, A; Ye, M J Med Chem 56: 1996-2015 (2013)
- Scott, WJ; Petrov, O; Möwes, M; Liu, N; Bömer, U US Patent US9675616 (2017)
- Traxler, P; Trinks, U; Buchdunger, E; Mett, H; Meyer, T; Müller, M; Regenass, U; Rösel, J; Lydon, N J Med Chem 38: 2441-8 (1995)
- Brauers, G; Edrada, RA; Ebel, R; Proksch, P; Wray, V; Berg, A; Gräfe, U; Schächtele, C; Totzke, F; Finkenzeller, G; Marme, D; Kraus, J; Münchbach, M; Michel, M; Bringmann, G; Schaumann, K J Nat Prod 63: 739-45 (2000)
- Volgraf, M; Lumb, JP; Brastianos, HC; Carr, G; Chung, MK; Münzel, M; Mauk, AG; Andersen, RJ; Trauner, D Nat Chem Biol 4: 535-7 (2008)
- Ahlström, MM; Ridderström, M; Zamora, I J Med Chem 50: 5382-91 (2007)
- Swahn, BM; Holenz, J; Kihlström, J; Kolmodin, K; Lindström, J; Plobeck, N; Rotticci, D; Sehgelmeble, F; Sundström, M; Berg, Sv; Fälting, J; Georgievska, B; Gustavsson, S; Neelissen, J; Ek, M; Olsson, LL; Berg, S Bioorg Med Chem Lett 22: 1854-9 (2012)
- Jin, J; An, M; Sapienza, A; Aiyar, N; Naselsky, D; Sarau, HM; Foley, JJ; Salyers, KL; Knight, SD; Keenan, RM; Rivero, RA; Dhanak, D; Douglas, SA Bioorg Med Chem Lett 18: 3950-4 (2008)
- Hidaka, K; Kimura, T; Sankaranarayanan, R; Wang, J; McDaniel, KF; Kempf, DJ; Kameoka, M; Adachi, M; Kuroki, R; Nguyen, JT; Hayashi, Y; Kiso, Y J Med Chem 61: 5138-5153 (2018)
- Helal, CJ; Sanner, MA; Cooper, CB; Gant, T; Adam, M; Lucas, JC; Kang, Z; Kupchinsky, S; Ahlijanian, MK; Tate, B; Menniti, FS; Kelly, K; Peterson, M Bioorg Med Chem Lett 14: 5521-5 (2004)
- Hughes, TV; Xu, G; Wetter, SK; Connolly, PJ; Emanuel, SL; Karnachi, P; Pollack, SR; Pandey, N; Adams, M; Moreno-Mazza, S; Middleton, SA; Greenberger, LM Bioorg Med Chem Lett 18: 4896-9 (2008)
- Kochanny, MJ; Adler, M; Ewing, J; Griedel, BD; Ho, E; Karanjawala, R; Lee, W; Lentz, D; Liang, AM; Morrissey, MM; Phillips, GB; Post, J; Sacchi, KL; Sakata, ST; Subramanyam, B; Vergona, R; Walters, J; White, KA; Whitlow, M; Ye, B; Zhao, Z; Shaw, KJ Bioorg Med Chem 15: 2127-46 (2007)
- Adonias, M; Anayaba, J; Cámara, J; Canet, E; Gateau-Olesker, A; Gero, SD; Grande, M; Hernando, JI Bioorg Med Chem Lett 3: 2547-2552 (1993)
- Campestre, C; Tortorella, P; Agamennone, M; Preziuso, S; Biasone, A; Nuti, E; Rossello, A; Gallina, C Eur J Med Chem 43: 1008-14 (2008)
- Hen, N; Bialer, M; Yagen, B; Maresca, A; Aggarwal, M; Robbins, AH; McKenna, R; Scozzafava, A; Supuran, CT J Med Chem 54: 3977-81 (2011)
- Louvel, J; Guo, D; Agliardi, M; Mocking, TA; Kars, R; Pham, TP; Xia, L; de Vries, H; Brussee, J; Heitman, LH; Ijzerman, AP J Med Chem 57: 3213-22 (2014)
- Bargota, RS; Akhtar, M; Biggadike, K; Gani, D; Allemann, RK Bioorg Med Chem Lett 13: 1623-6 (2003)
- Yamaguchi, M; Kamei, K; Koga, T; Akima, M; Maruyama, A; Kuroki, T; Ohi, N J Med Chem 36: 4061-8 (1994)
- Muralidharan, VP; Alagumuthu, M; Iyer, SK Bioorg Med Chem Lett 27: 2510-2514 (2017)
- Chen, P; Cheng, PT; Alam, M; Beyer, BD; Bisacchi, GS; Dejneka, T; Evans, AJ; Greytok, JA; Hermsmeier, MA; Humphreys, WG; Jacobs, GA; Kocy, O; Lin, PF; Lis, KA; Marella, MA; Ryono, DE; Sheaffer, AK; Spergel, SH; Sun, CQ; Tino, JA; Vite, G; Colonno, RJ; Zahler, R; Barrish, JC J Med Chem 39: 1991-2007 (1996)
- Lawson, M; Rodrigo, J; Baratte, B; Robert, T; Delehouzé, C; Lozach, O; Ruchaud, S; Bach, S; Brion, JD; Alami, M; Hamze, A Eur J Med Chem 123: 105-114 (2016)
- Tanis, VM; Venkatesan, H; Cummings, MD; Albers, M; Kent Barbay, J; Herman, K; Kummer, DA; Milligan, C; Nelen, MI; Nishimura, R; Schlueter, T; Scott, B; Spurlino, J; Wolin, R; Woods, C; Xue, X; Edwards, JP; Fourie, AM; Leonard, K Bioorg Med Chem Lett 29: 1463-1470 (2019)
- Hansen, JD; Correa, M; Nagy, MA; Alexander, M; Plantevin, V; Grant, V; Whitefield, B; Huang, D; Kercher, T; Harris, R; Narla, RK; Leisten, J; Tang, Y; Moghaddam, M; Ebinger, K; Piccotti, J; Havens, CG; Cathers, B; Carmichael, J; Daniel, T; Vessey, R; Hamann, LG; Leftheris, K; Mendy, D; Baculi, F; LeBrun, LA; Khambatta, G; Lopez-Girona, A J Med Chem 63: 6648-6676 (2020)
- Taha, M; Ismail, NH; Imran, S; Selvaraj, M; Rahim, A; Ali, M; Siddiqui, S; Rahim, F; Khan, KM Bioorg Med Chem 23: 7394-404 (2015)
- Grimster, NP; Anderson, E; Alimzhanov, M; Bebernitz, G; Bell, K; Chuaqui, C; Deegan, T; Ferguson, AD; Gero, T; Harsch, A; Huszar, D; Kawatkar, A; Kettle, JG; Lyne, P; Read, JA; Rivard Costa, C; Ruston, L; Schroeder, P; Shi, J; Su, Q; Throner, S; Toader, D; Vasbinder, M; Woessner, R; Wang, H; Wu, A; Ye, M; Zheng, W; Zinda, M J Med Chem 61: 5235-5244 (2018)
- Allan, M; Manku, S; Therrien, E; Nguyen, N; Styhler, S; Robert, MF; Goulet, AC; Petschner, AJ; Rahil, G; Robert Macleod, A; Déziel, R; Besterman, JM; Nguyen, H; Wahhab, A Bioorg Med Chem Lett 19: 1218-23 (2009)
- Morera, E; Di Marzo, V; Monti, L; Allarŕ, M; Schiano Moriello, A; Nalli, M; Ortar, G; De Petrocellis, L Bioorg Med Chem Lett 26: 1401-5 (2016)
- Giannotti, D; Perrotta, E; Di Bugno, C; Nannicini, R; Harmat, NJ; Giolitti, A; Patacchini, R; Renzetti, AR; Rotondaro, L; Giuliani, S; Altamura, M; Maggi, CA J Med Chem 43: 4041-4 (2000)
- Mahalingam, AK; Wan, Y; Murugaiah, AM; Wallinder, C; Wu, X; Plouffe, B; Botros, M; Nyberg, F; Hallberg, A; Gallo-Payet, N; Alterman, M Bioorg Med Chem 18: 4570-90 (2010)
- Sadeghzadeh, M; Sheibani, S; Ghandi, M; Daha, FJ; Amanlou, M; Arjmand, M; Hasani Bozcheloie, A Eur J Med Chem 64: 488-97 (2013)
- Iio, K; Saitoh, T; Ohshita, R; Hino, T; Amezawa, M; Takayama, Y; Nagumo, Y; Yamamoto, N; Kutsumura, N; Irukayama-Tomobe, Y; Ishikawa, Y; Tanimura, R; Yanagisawa, M; Nagase, H Bioorg Med Chem Lett 60: (2022)
- Hansen, JD; Correa, M; Alexander, M; Nagy, M; Huang, D; Sapienza, J; Lu, G; LeBrun, LA; Cathers, BE; Zhang, W; Tang, Y; Ammirante, M; Narla, RK; Piccotti, JR; Pourdehnad, M; Lopez-Girona, A J Med Chem 64: 1835-1843 (2021)
- Rahm, F; Viklund, J; Trésaugues, L; Ellermann, M; Giese, A; Ericsson, U; Forsblom, R; Ginman, T; Günther, J; Hallberg, K; Lindström, J; Persson, LB; Silvander, C; Talagas, A; Díaz-Sáez, L; Fedorov, O; Huber, KVM; Panagakou, I; Siejka, P; Gorjánácz, M; Bauser, M; Andersson, M J Med Chem 61: 2533-2551 (2018)
- Nepovimova, E; Korabecny, J; Dolezal, R; Babkova, K; Ondrejicek, A; Jun, D; Sepsova, V; Horova, A; Hrabinova, M; Soukup, O; Bukum, N; Jost, P; Muckova, L; Kassa, J; Malinak, D; Andrs, M; Kuca, K J Med Chem 58: 8985-9003 (2015)
- Salimbeni, A; Paleari, F; Canevotti, R; Criscuoli, M; Criscuoli, M; Lippi, A; Angiolini, M; Belvisi, L; Scolastico, C; Colombo, L Bioorg Med Chem Lett 7: 2205-2210 (1997)
- Mollica, L; Theret, I; Antoine, M; Perron-Sierra, F; Charton, Y; Fourquez, JM; Wierzbicki, M; Boutin, JA; Ferry, G; Decherchi, S; Bottegoni, G; Ducrot, P; Cavalli, A J Med Chem 59: 7167-76 (2016)
- Cappelli, A; Manini, M; Paolino, M; Gallelli, A; Anzini, M; Mennuni, L; Del Cadia, M; De Rienzo, F; Menziani, MC; Vomero, S ACS Med Chem Lett 2: 571-576 (2011)
- Miyazaki, M; Naito, H; Sugimoto, Y; Kawato, H; Okayama, T; Shimizu, H; Miyazaki, M; Kitagawa, M; Seki, T; Fukutake, S; Aonuma, M; Soga, T Bioorg Med Chem Lett 23: 728-32 (2013)
- Yonezawa, S; Fujiwara, K; Yamamoto, T; Hattori, K; Yamakawa, H; Muto, C; Hosono, M; Tanaka, Y; Nakano, T; Takemoto, H; Arisawa, M; Shuto, S Bioorg Med Chem 21: 6506-22 (2013)
- Sadeghzadeh, M; Sheibani, S; Ghandi, M; Daha, FJ; Amanlou, M; Arjmand, M; Hasani Bozcheloie, A Eur J Med Chem 64: 488-97 (2013)
- Liessi, N; Cichero, E; Pesce, E; Arkel, M; Salis, A; Tomati, V; Paccagnella, M; Damonte, G; Tasso, B; Galietta, LJV; Pedemonte, N; Fossa, P; Millo, E Eur J Med Chem 144: 179-200 (2018)
- Huryn, DM; Wipf, P; LaPorte, MG; Colombo, R; Kovaliov, M; Lim, C; Alverez, CN; Yue, Z; Samankumara, LP; Chatterley, AJ; Yan, Y; Liang, M; Green, NJ; Baldwin, ET; Moore, WJ; Arkin, M; Neitz, RJ; Ang, K; Bryant, C; Bulfer, S US Patent US11247985 (2022)
- Fidan, I; Salmas, RE; Arslan, M; Sentürk, M; Durdagi, S; Ekinci, D; Sentürk, E; Cosgun, S; Supuran, CT Bioorg Med Chem 23: 7353-8 (2015)
- Asada, M; Obitsu, T; Kinoshita, A; Nagase, T; Yoshida, T; Yamaura, Y; Takizawa, H; Yoshikawa, K; Sato, K; Narita, M; Nakai, H; Toda, M; Tobe, Y Bioorg Med Chem 18: 3212-23 (2010)
- Montanari, R; Saccoccia, F; Scotti, E; Crestani, M; Godio, C; Gilardi, F; Loiodice, F; Fracchiolla, G; Laghezza, A; Tortorella, P; Lavecchia, A; Novellino, E; Mazza, F; Aschi, M; Pochetti, G J Med Chem 51: 7768-76 (2008)
- Di Maro, S; Di Leva, FS; Trotta, AM; Brancaccio, D; Portella, L; Aurilio, M; Tomassi, S; Messere, A; Sementa, D; Lastoria, S; Carotenuto, A; Novellino, E; Scala, S; Marinelli, L J Med Chem 60: 9641-9652 (2017)
- Velcicky, J; Mathison, CJN; Nikulin, V; Pflieger, D; Epple, R; Azimioara, M; Cow, C; Michellys, PY; Rigollier, P; Beisner, DR; Bodendorf, U; Guerini, D; Liu, B; Wen, B; Zaharevitz, S; Brandl, T ACS Med Chem Lett 10: 887-892 (2019)
- Babler, M; Gerritsen, ME US Patent US9572811 (2017)
- Banerjee, A; Narayana, L; Raje, FA; Pisal, DV; Kadam, PA; Gullapalli, S; Kumar, H; More, SV; Bajpai, M; Sangana, RR; Jadhav, S; Gudi, GS; Khairatkar-Joshi, N; Merugu, RR; Voleti, SR; Gharat, LA Bioorg Med Chem Lett 23: 6747-54 (2013)
- Bansal, S; Bala, M; Suthar, SK; Choudhary, S; Bhattacharya, S; Bhardwaj, V; Singla, S; Joseph, A Eur J Med Chem 80: 167-74 (2014)
- Serrán-Aguilera, L; Mariotto, E; Rubbini, G; Castro Navas, FF; Marco, C; Carrasco-Jiménez, MP; Ballarotto, M; Macchiarulo, A; Hurtado-Guerrero, R; Viola, G; Lopez-Cara, LC Eur J Med Chem 207: (2020)
- Czudor, Z; Balogh, M; Bánhegyi, P; Boros, S; Breza, N; Dobos, J; Fábián, M; Horváth, Z; Illyés, E; Markó, P; Sipos, A; Szántai-Kis, C; Szokol, B; ?rfi, L Bioorg Med Chem Lett 28: 769-773 (2018)
- Doe, C; Bentley, R; Behm, DJ; Lafferty, R; Stavenger, R; Jung, D; Bamford, M; Panchal, T; Grygielko, E; Wright, LL; Smith, GK; Chen, Z; Webb, C; Khandekar, S; Yi, T; Kirkpatrick, R; Dul, E; Jolivette, L; Marino, JP; Willette, R; Lee, D; Hu, E J Pharmacol Exp Ther 320: 89-98 (2006)
- Banerjee, M; Middya, S; Shrivastava, R; Raina, S; Surya, A; Yadav, DB; Yadav, VK; Kapoor, KK; Venkatesan, A; Smith, RA; Thompson, SK US Patent US10294212 (2019)
- van der Stelt, M; van Kuik, JA; Bari, M; van Zadelhoff, G; Leeflang, BR; Veldink, GA; Finazzi-Agrò, A; Vliegenthart, JF; Maccarrone, M J Med Chem 45: 3709-20 (2002)
- Carosati, E; Mannhold, R; Wahl, P; Hansen, JB; Fremming, T; Zamora, I; Cianchetta, G; Baroni, M J Med Chem 50: 2117-26 (2007)
- D'Agostino, LA; Sjin, RT; Niu, D; McDonald, JJ; Zhu, Z; Liu, H; Mazdiyasni, H; Petter, RC; Singh, J; Barrague, M; Gross, A; Munson, M US Patent US9695132 (2017)
- Hille, UE; Hu, Q; Vock, C; Negri, M; Bartels, M; Müller-Vieira, U; Lauterbach, T; Hartmann, RW Eur J Med Chem 44: 2765-75 (2009)
- Camps, P; Formosa, X; Galdeano, C; Gómez, T; Muñoz-Torrero, D; Scarpellini, M; Viayna, E; Badia, A; Clos, MV; Camins, A; Pallàs, M; Bartolini, M; Mancini, F; Andrisano, V; Estelrich, J; Lizondo, M; Bidon-Chanal, A; Luque, FJ J Med Chem 51: 3588-98 (2008)
- De Simone, A; Bartolini, M; Baschieri, A; Apperley, KYP; Chen, HH; Guardigni, M; Montanari, S; Kobrlova, T; Soukup, O; Valgimigli, L; Andrisano, V; Keillor, JW; Basso, M; Milelli, A Eur J Med Chem 139: 378-389 (2017)
- Nar, H; Bauer, M; Schmid, A; Stassen, JM; Wienen, W; Priepke, HW; Kauffmann, IK; Ries, UJ; Hauel, NH Structure 9: 29-37 (2001)
- Rahm, F; Viklund, J; Trésaugues, L; Ellermann, M; Giese, A; Ericsson, U; Forsblom, R; Ginman, T; Günther, J; Hallberg, K; Lindström, J; Persson, LB; Silvander, C; Talagas, A; Díaz-Sáez, L; Fedorov, O; Huber, KVM; Panagakou, I; Siejka, P; Gorjánácz, M; Bauser, M; Andersson, M J Med Chem 61: 2533-2551 (2018)
- Grob, NM; Häussinger, D; Deupi, X; Schibli, R; Behe, M; Mindt, TL J Med Chem 63: 4484-4495 (2020)
- Stefanowicz, J; S?owi?ski, T; Wróbel, MZ; Herold, F; Gomó?ka, AE; Weso?owska, A; Jastrz?bska-Wi?sek, M; Partyka, A; Andres-Mach, M; Czuczwar, SJ; ?uszczki, JJ; Zagaja, M; Siwek, A; Nowak, G; ?o?nierek, M; B?czek, T; Ulenberg, S; Belka, M; Tur?o, J Bioorg Med Chem 24: 3994-4007 (2016)
- Gallant, M; Belley, M; Carrière, MC; Chateauneuf, A; Denis, D; Lachance, N; Lamontagne, S; Metters, KM; Sawyer, N; Slipetz, D; Truchon, JF; Labelle, M Bioorg Med Chem Lett 13: 3813-6 (2003)
- Blake, JF; Burkard, M; Chan, J; Chen, H; Chou, KJ; Diaz, D; Dudley, DA; Gaudino, JJ; Gould, SE; Grina, J; Hunsaker, T; Liu, L; Martinson, M; Moreno, D; Mueller, L; Orr, C; Pacheco, P; Qin, A; Rasor, K; Ren, L; Robarge, K; Shahidi-Latham, S; Stults, J; Sullivan, F; Wang, W; Yin, J; Zhou, A; Belvin, M; Merchant, M; Moffat, J; Schwarz, JB J Med Chem 59: 5650-60 (2016)
- Swahn, BM; Sandell, J; Pyring, D; Bergh, M; Jeppsson, F; Juréus, A; Neelissen, J; Johnström, P; Schou, M; Svensson, S Bioorg Med Chem Lett 22: 4332-7 (2012)
- Zeng, Q; Rosenblum, SB; Yang, Z; Jiang, Y; McCormick, KD; Aslanian, RG; Duguma, L; Kozlowski, JA; Shih, NY; Hey, JA; West, RE; Korfmacher, WA; Berlin, M; Boyce, CW Bioorg Med Chem Lett 23: 6001-3 (2013)
- Schaller, D; Hagenow, S; Alpert, G; Naß, A; Schulz, R; Bermudez, M; Stark, H; Wolber, G ACS Med Chem Lett 8: 648-653 (2017)
- Saupe, SM; Leubner, S; Betz, M; Klebe, G; Steinmetzer, T J Med Chem 56: 820-31 (2013)
- Skerlj, R; Bridger, G; Zhou, Y; Bourque, E; McEachern, E; Langille, J; Harwig, C; Veale, D; Yang, W; Li, T; Zhu, Y; Bey, M; Baird, I; Sartori, M; Metz, M; Mosi, R; Nelson, K; Bodart, V; Wong, R; Fricker, S; Mac Farland, R; Huskens, D; Schols, D Bioorg Med Chem Lett 21: 6950-4 (2011)
- Dawson, MI; Xia, Z; Jiang, T; Ye, M; Fontana, JA; Farhana, L; Patel, B; Xue, LP; Bhuiyan, M; Pellicciari, R; Macchiarulo, A; Nuti, R; Zhang, XK; Han, YH; Tautz, L; Hobbs, PD; Jong, L; Waleh, N; Chao, WR; Feng, GS; Pang, Y; Su, Y J Med Chem 51: 5650-62 (2008)
- Hen, N; Bialer, M; Yagen, B; Maresca, A; Aggarwal, M; Robbins, AH; McKenna, R; Scozzafava, A; Supuran, CT J Med Chem 54: 3977-81 (2011)
- Battilocchio, C; Poce, G; Alfonso, S; Porretta, GC; Consalvi, S; Sautebin, L; Pace, S; Rossi, A; Ghelardini, C; Di Cesare Mannelli, L; Schenone, S; Giordani, A; Di Francesco, L; Patrignani, P; Biava, M Bioorg Med Chem 21: 3695-701 (2013)
- Mahy, W; Willis, NJ; Zhao, Y; Woodward, HL; Svensson, F; Sipthorp, J; Vecchia, L; Ruza, RR; Hillier, J; Kjćr, S; Frew, S; Monaghan, A; Bictash, M; Salinas, PC; Whiting, P; Vincent, JP; Jones, EY; Fish, PV J Med Chem 63: 12942-12956 (2020)
- Rossi, C; Porcelloni, M; D'Andrea, P; Fincham, CI; Ettorre, A; Mauro, S; Squarcia, A; Bigioni, M; Parlani, M; Nardelli, F; Binaschi, M; Maggi, CA; Fattori, D Bioorg Med Chem Lett 21: 2305-8 (2011)
- Axford, LC; Agarwal, PK; Anderson, KH; Andrau, LN; Atherall, J; Barker, S; Bennett, JM; Blair, M; Collins, I; Czaplewski, LG; Davies, DT; Gannon, CT; Kumar, D; Lancett, P; Logan, A; Lunniss, CJ; Mitchell, DR; Offermann, DA; Palmer, JT; Palmer, N; Pitt, GR; Pommier, S; Price, D; Narasinga Rao, B; Saxena, R; Shukla, T; Singh, AK; Singh, M; Srivastava, A; Steele, C; Stokes, NR; Thomaides-Brears, HB; Tyndall, EM; Watson, D; Haydon, DJ Bioorg Med Chem Lett 23: 6598-603 (2013)
- Arora, J; Bordeleau, M; Dube, L; Jarvie, K; Mazzocco, L; Peragine, J; Tehim, A; Egle, I Bioorg Med Chem Lett 15: 5253-6 (2005)
- Marzaro, G; Guiotto, A; Borgatti, M; Finotti, A; Gambari, R; Breveglieri, G; Chilin, A J Med Chem 56: 1830-42 (2013)
- Rosenström, U; Sköld, C; Lindeberg, G; Botros, M; Nyberg, F; Karlén, A; Hallberg, A J Med Chem 49: 6133-7 (2006)
- Manetti, F; Brullo, C; Magnani, M; Mosci, F; Chelli, B; Crespan, E; Schenone, S; Naldini, A; Bruno, O; Trincavelli, ML; Maga, G; Carraro, F; Martini, C; Bondavalli, F; Botta, M J Med Chem 51: 1252-9 (2008)
- Doll, F; Dolci, L; Valette, H; Hinnen, F; Vaufrey, F; Guenther, I; Fuseau, C; Coulon, C; Bottlaender, M; Crouzel, C J Med Chem 42: 2251-9 (1999)
- Bouaboula, M; Brollo, M; Certal, V; El-Ahmad, Y; Filoche-Romme, B; Halley, F; McCort, G; Schio, L; Tabart, M; Terrier, C; Thompson, F US Patent US9714221 (2017)
- Giraud, F; Bourhis, M; Ebrahimi, E; Herfindal, L; Choudhury, RR; Bjřrnstad, R; Dřskeland, SO; Anizon, F; Moreau, P Bioorg Med Chem 23: 7313-23 (2015)
- Knoepfel, T; Nimsgern, P; Jacquier, S; Bourrel, M; Vangrevelinghe, E; Glatthar, R; Behnke, D; Alper, PB; Michellys, PY; Deane, J; Junt, T; Zipfel, G; Limonta, S; Hawtin, S; Andre, C; Boulay, T; Loetscher, P; Faller, M; Blank, J; Feifel, R; Betschart, C J Med Chem 63: 8276-8295 (2020)
- Siu, T; Kozina, ES; Jung, J; Rosenstein, C; Mathur, A; Altman, MD; Chan, G; Xu, L; Bachman, E; Mo, JR; Bouthillette, M; Rush, T; Dinsmore, CJ; Marshall, CG; Young, JR Bioorg Med Chem Lett 20: 7421-5 (2010)
- Corręa, MF; Balico-Silva, AL; Kiss, DJ; Fernandes, GAB; Maraschin, JC; Parreiras-E-Silva, LT; Varela, MT; Simőes, SC; Bouvier, M; Keser?, GM; Costa-Neto, CM; Fernandes, JPS Bioorg Med Chem 30: (2021)
- Bozdag, M; Alafeefy, AM; Altamimi, AM; Carta, F; Supuran, CT; Vullo, D Bioorg Med Chem 25: 2782-2788 (2017)
- Baxter, EW; Conway, KA; Kennis, L; Bischoff, F; Mercken, MH; Winter, HL; Reynolds, CH; Tounge, BA; Luo, C; Scott, MK; Huang, Y; Braeken, M; Pieters, SM; Berthelot, DJ; Masure, S; Bruinzeel, WD; Jordan, AD; Parker, MH; Boyd, RE; Qu, J; Alexander, RS; Brenneman, DE; Reitz, AB J Med Chem 50: 4261-4 (2007)
- Holt, DA; Yamashita, DS; Konialian-Beck, AL; Luengo, JI; Abell, AD; Bergsma, DJ; Brandt, M; Levy, MA J Med Chem 38: 13-5 (1995)
- Butini, S; Brindisi, M; Cosconati, S; Marinelli, L; Borrelli, G; Coccone, SS; Ramunno, A; Campiani, G; Novellino, E; Zanoli, S; Samuele, A; Giorgi, G; Bergamini, A; Mattia, MD; Lalli, S; Galletti, B; Gemma, S; Maga, G J Med Chem 52: 1224-8 (2009)
- Vaz, RJ; Gao, Z; Pribish, J; Chen, X; Levell, J; Davis, L; Albert, E; Brollo, M; Ugolini, A; Cramer, DM; Cairns, J; Sides, K; Liu, F; Kwong, J; Kang, J; Rebello, S; Elliot, M; Lim, H; Chellaraj, V; Singleton, RW; Li, Y Bioorg Med Chem Lett 14: 6053-6 (2004)
- Bruncko, M; Tahir, SK; Song, X; Chen, J; Ding, H; Huth, JR; Jin, S; Judge, RA; Madar, DJ; Park, CH; Park, CM; Petros, AM; Tse, C; Rosenberg, SH; Elmore, SW Bioorg Med Chem Lett 20: 7503-6 (2010)
- Yeh, VS; Patel, JR; Yong, H; Kurukulasuriya, R; Fung, S; Monzon, K; Chiou, W; Wang, J; Stolarik, D; Imade, H; Beno, D; Brune, M; Jacobson, P; Sham, H; Link, JT Bioorg Med Chem Lett 16: 5414-9 (2006)
- Spicer, JA; Lena, G; Lyons, DM; Huttunen, KM; Miller, CK; O'Connor, PD; Bull, M; Helsby, N; Jamieson, SM; Denny, WA; Ciccone, A; Browne, KA; Lopez, JA; Rudd-Schmidt, J; Voskoboinik, I; Trapani, JA J Med Chem 56: 9542-55 (2014)
- Urbani, P; Cavallo, P; Cascio, MG; Buonerba, M; De Martino, G; Di Marzo, V; Saturnino, C Bioorg Med Chem Lett 16: 138-41 (2005)
- Volgraf, M; Chan, L; Huestis, MP; Purkey, HE; Burkard, M; Geck Do, M; Harris, J; Hunt, KW; Liu, X; Lyssikatos, JP; Rana, S; Thomas, AA; Vigers, GP; Siu, M Bioorg Med Chem Lett 24: 2477-80 (2014)
- Kinzel, O; Steeneck, C; Schlüter, T; Schulz, A; Gege, C; Hahn, U; Hambruch, E; Hornberger, M; Spalwisz, A; Frick, K; Perovic-Ottstadt, S; Deuschle, U; Burnet, M; Kremoser, C Bioorg Med Chem Lett 26: 3746-53 (2016)
- Mallinger, A; Schiemann, K; Rink, C; Stieber, F; Calderini, M; Crumpler, S; Stubbs, M; Adeniji-Popoola, O; Poeschke, O; Busch, M; Czodrowski, P; Musil, D; Schwarz, D; Ortiz-Ruiz, MJ; Schneider, R; Thai, C; Valenti, M; de Haven Brandon, A; Burke, R; Workman, P; Dale, T; Wienke, D; Clarke, PA; Esdar, C; Raynaud, FI; Eccles, SA; Rohdich, F; Blagg, J J Med Chem 59: 1078-101 (2016)
- Zhou, Y; Mowlazadeh Haghighi, S; Zoi, I; Sawyer, JR; Hruby, VJ; Cai, M J Med Chem 60: 9320-9329 (2017)
- Caldarelli, M; Habermann, J; Ley, SV Bioorg Med Chem Lett 9: 2049-52 (1999)
- Wucherer-Plietker, M; Merkul, E; Müller, TJ; Esdar, C; Knöchel, T; Heinrich, T; Buchstaller, HP; Greiner, H; Dorsch, D; Finsinger, D; Calderini, M; Bruge, D; Grädler, U Bioorg Med Chem Lett 26: 3073-80 (2016)
- Caligiuri, M; Molz, L; Liu, Q; Kaplan, F; Xu, JP; Majeti, JZ; Ramos-Kelsey, R; Murthi, K; Lievens, S; Tavernier, J; Kley, N Chem Biol 13: 711-22 (2006)
- Porter, J; Lumb, S; Franklin, RJ; Gascon-Simorte, JM; Calmiano, M; Riche, KL; Lallemand, B; Keyaerts, J; Edwards, H; Maloney, A; Delgado, J; King, L; Foley, A; Lecomte, F; Reuberson, J; Meier, C; Batchelor, M Bioorg Med Chem Lett 19: 2780-4 (2009)
- Richard, DJ; Lena, R; Bannister, T; Blake, N; Pierceall, WE; Carlson, NE; Keller, CE; Koenig, M; He, Y; Minond, D; Mishra, J; Cameron, M; Spicer, T; Hodder, P; Cardone, MH Bioorg Med Chem 21: 6642-9 (2013)
- Zhang, H; Ding, CZ; Lai, Z; Chen, SS; Devasthale, P; Herpin, T; Morton, G; Qu, F; Ryono, D; Smirk, R; Wang, W; Wu, S; Ye, XX; Li, YX; Apedo, A; Farrelly, D; Wang, T; Gu, L; Morgan, N; Flynn, N; Chu, C; Kunselman, L; Lippy, J; Locke, K; O'Malley, K; Harrity, T; Cap, M; Zhang, L; Hosagrahara, V; Kadiyala, P; Xu, C; Doweyko, AM; Zahler, R; Hariharan, N; Cheng, PT Bioorg Med Chem Lett 25: 1196-205 (2015)
- Costantino, L; Rastelli, G; Vescovini, K; Cignarella, G; Vianello, P; Del Corso, A; Cappiello, M; Mura, U; Barlocco, D J Med Chem 39: 4396-405 (1996)
- Sechi, M; Innocenti, A; Pala, N; Rogolino, D; Carcelli, M; Scozzafava, A; Supuran, CT Bioorg Med Chem Lett 22: 5801-6 (2012)
- Castillo, M; Forns, P; Erra, M; Mir, M; López, M; Maldonado, M; Orellana, A; Carreño, C; Ramis, I; Miralpeix, M; Vidal, B Bioorg Med Chem Lett 22: 5419-23 (2012)
- Pisani, L; Catto, M; Nicolotti, O; Grossi, G; Di Braccio, M; Soto-Otero, R; Mendez-Alvarez, E; Stefanachi, A; Gadaleta, D; Carotti, A Eur J Med Chem 70: 723-39 (2013)
- Abdel-Aziz, AA; El-Azab, AS; Ceruso, M; Supuran, CT Bioorg Med Chem Lett 24: 5185-9 (2014)
- Ceruti, M; Rocco, F; Viola, F; Balliano, G; Milla, P; Arpicco, S; Cattel, L J Med Chem 41: 540-54 (1998)
- Jacobson, KA; Ohno, M; Duong, HT; Kim, SK; Tchilibon, S; Cesnek, M; Holý, A; Gao, ZG Chem Biol 12: 237-47 (2005)
- Chao, H; Turdi, H; Herpin, TF; Roberge, JY; Liu, Y; Schnur, DM; Poss, MA; Rehfuss, R; Hua, J; Wu, Q; Price, LA; Abell, LM; Schumacher, WA; Bostwick, JS; Steinbacher, TE; Stewart, AB; Ogletree, ML; Huang, CS; Chang, M; Cacace, AM; Arcuri, MJ; Celani, D; Wexler, RR; Lawrence, RM J Med Chem 56: 1704-14 (2013)
- Rewcastle, GW; Gamage, SA; Flanagan, JU; Kendall, JD; Denny, WA; Baguley, BC; Buchanan, CM; Chao, M; Kestell, P; Kolekar, S; Lee, WJ; Lill, CL; Malik, A; Singh, R; Jamieson, SM; Shepherd, PR Eur J Med Chem 64: 137-47 (2013)
- Liedtke, AJ; Adeniji, AO; Chen, M; Byrns, MC; Jin, Y; Christianson, DW; Marnett, LJ; Penning, TM J Med Chem 56: 2429-46 (2013)
- Xing, G; Pan, L; Yi, C; Li, X; Ge, X; Zhao, Y; Liu, Y; Li, J; Woo, A; Lin, B; Zhang, Y; Cheng, M Bioorg Med Chem 27: 2306-2314 (2019)
- Matthews, TP; McHardy, T; Klair, S; Boxall, K; Fisher, M; Cherry, M; Allen, CE; Addison, GJ; Ellard, J; Aherne, GW; Westwood, IM; van Montfort, R; Garrett, MD; Reader, JC; Collins, I Bioorg Med Chem Lett 20: 4045-9 (2010)
- Cheung, M; Tangirala, RS US Patent US9796729 (2017)
- Rueeger, H; Rigollier, P; Yamaguchi, Y; Schmidlin, T; Schilling, W; Criscione, L; Whitebread, S; Chiesi, M; Walker, MW; Dhanoa, D; Islam, I; Zhang, J; Gluchowski, C Bioorg Med Chem Lett 10: 1175-9 (2000)
- Seabrook, GR; Sutton, KG; Jarolimek, W; Hollingworth, GJ; Teague, S; Webb, J; Clark, N; Boyce, S; Kerby, J; Ali, Z; Chou, M; Middleton, R; Kaczorowski, G; Jones, AB J Pharmacol Exp Ther 303: 1052-60 (2002)
- Chu, M; Mierzwa, R; He, L; King, A; Patel, M; Pichardo, J; Hart, A; Butkiewicz, N; Puar, MS Bioorg Med Chem Lett 9: 1949-52 (1999)
- Flavin, MT; Rizzo, JD; Khilevich, A; Kucherenko, A; Sheinkman, AK; Vilaychack, V; Lin, L; Chen, W; Greenwood, EM; Pengsuparp, T; Pezzuto, JM; Hughes, SH; Flavin, TM; Cibulski, M; Boulanger, WA; Shone, RL; Xu, ZQ J Med Chem 39: 1303-13 (1996)
- Kaller, MR; Harried, SS; Albrecht, B; Amarante, P; Babu-Khan, S; Bartberger, MD; Brown, J; Brown, R; Chen, K; Cheng, Y; Citron, M; Croghan, MD; Graceffa, R; Hickman, D; Judd, T; Kriemen, C; La, D; Li, V; Lopez, P; Luo, Y; Masse, C; Monenschein, H; Nguyen, T; Pennington, LD; Miguel, TS; Sickmier, EA; Wahl, RC; Weiss, MM; Wen, PH; Williamson, T; Wood, S; Xue, M; Yang, B; Zhang, J; Patel, V; Zhong, W; Hitchcock, S ACS Med Chem Lett 3: 886-891 (2012)
- Armani, E; Amari, G; Rizzi, A; De Fanti, R; Ghidini, E; Capaldi, C; Carzaniga, L; Caruso, P; Guala, M; Peretto, I; La Porta, E; Bolzoni, PT; Facchinetti, F; Carnini, C; Moretto, N; Patacchini, R; Bassani, F; Cenacchi, V; Volta, R; Amadei, F; Capacchi, S; Delcanale, M; Puccini, P; Catinella, S; Civelli, M; Villetti, G J Med Chem 57: 793-816 (2014)
- Neidhart, W; Breu, V; Burri, K; Clozel, M; Hirth, G; Klinkhammer, U; Giller, T; Ramuz, H Bioorg Med Chem Lett 7: 2223-2228 (1997)
- McCoull, W; Boyd, S; Brown, MR; Coen, M; Collingwood, O; Davies, NL; Doherty, A; Fairley, G; Goldberg, K; Hardaker, E; He, G; Hennessy, EJ; Hopcroft, P; Hodgson, G; Jackson, A; Jiang, X; Karmokar, A; Lainé, AL; Lindsay, N; Mao, Y; Markandu, R; McMurray, L; McLean, N; Mooney, L; Musgrove, H; Nissink, JWM; Pflug, A; Reddy, VP; Rawlins, PB; Rivers, E; Schimpl, M; Smith, GF; Tentarelli, S; Travers, J; Troup, RI; Walton, J; Wang, C; Wilkinson, S; Williamson, B; Winter-Holt, J; Yang, D; Zheng, Y; Zhu, Q; Smith, PD J Med Chem 64: 13524-13539 (2021)
- Stahlecker, J; Klett, T; Schwer, M; Jaag, S; Dammann, M; Ernst, LN; Braun, MB; Zimmermann, MO; Kramer, M; Lämmerhofer, M; Stehle, T; Coles, M; Boeckler, FM RSC Med Chem 13: 1575-1586 (2022)
- Collin, M; Brohm, D; Héroult, M; Lobell, M; Hübsch, W; Lustig, K; Grünewald, S; Bömer, U; Vöhringer, V; Lindner, N US Patent US9598416 (2017)
- Wang, Y; Yu, M; Zhu, J; Zhang, JK; Kayser, F; Medina, JC; Siegler, K; Conn, M; Shan, B; Grillo, MP; Liu, JJ; Coward, P Bioorg Med Chem Lett 24: 1133-7 (2014)
- Njoroge, FG; Taveras, AG; Kelly, J; Remiszewski, S; Mallams, AK; Wolin, R; Afonso, A; Cooper, AB; Rane, DF; Liu, YT; Wong, J; Vibulbhan, B; Pinto, P; Deskus, J; Alvarez, CS; del Rosario, J; Connolly, M; Wang, J; Desai, J; Rossman, RR; Bishop, WR; Patton, R; Wang, L; Kirschmeier, P; Ganguly, AK J Med Chem 41: 4890-902 (1998)
- Berardi, F; Ferorelli, S; Abate, C; Pedone, MP; Colabufo, NA; Contino, M; Perrone, R J Med Chem 48: 8237-44 (2005)
- Elhalem, E; Bellomo, A; Cooke, M; Scravaglieri, A; Pearce, LV; Peach, ML; Gandolfi Donadío, L; Kazanietz, MG; Comin, MJ J Med Chem 64: 11418-11431 (2021)
- Andrés, JI; Alonso, JM; Díaz, A; Fernández, J; Iturrino, L; Martínez, P; Matesanz, E; Freyne, EJ; Deroose, F; Boeckx, G; Petit, D; Diels, G; Megens, A; Somers, M; Van Wauwe, J; Stoppie, P; Cools, M; De Clerck, F; Peeters, D; de Chaffoy, D Bioorg Med Chem Lett 12: 653-8 (2002)
- Verhoest, PR; Proulx-Lafrance, C; Corman, M; Chenard, L; Helal, CJ; Hou, X; Kleiman, R; Liu, S; Marr, E; Menniti, FS; Schmidt, CJ; Vanase-Frawley, M; Schmidt, AW; Williams, RD; Nelson, FR; Fonseca, KR; Liras, S J Med Chem 52: 7946-9 (2009)
- Hansen, JD; Correa, M; Nagy, MA; Alexander, M; Plantevin, V; Grant, V; Whitefield, B; Huang, D; Kercher, T; Harris, R; Narla, RK; Leisten, J; Tang, Y; Moghaddam, M; Ebinger, K; Piccotti, J; Havens, CG; Cathers, B; Carmichael, J; Daniel, T; Vessey, R; Hamann, LG; Leftheris, K; Mendy, D; Baculi, F; LeBrun, LA; Khambatta, G; Lopez-Girona, A J Med Chem 63: 6648-6676 (2020)
- Micheli, F; Cavanni, P; Andreotti, D; Arban, R; Benedetti, R; Bertani, B; Bettati, M; Bettelini, L; Bonanomi, G; Braggio, S; Carletti, R; Checchia, A; Corsi, M; Fazzolari, E; Fontana, S; Marchioro, C; Merlo-Pich, E; Negri, M; Oliosi, B; Ratti, E; Read, KD; Roscic, M; Sartori, I; Spada, S; Tedesco, G; Tarsi, L; Terreni, S; Visentini, F; Zocchi, A; Zonzini, L; Di Fabio, R J Med Chem 53: 4989-5001 (2010)
- Varnes, JG; Gardner, DS; Santella, JB; Duncia, JV; Estrella, M; Watson, PS; Clark, CM; Ko, SS; Welch, P; Covington, M; Stowell, N; Wadman, E; Davies, P; Solomon, K; Newton, RC; Trainor, GL; Decicco, CP; Wacker, DA Bioorg Med Chem Lett 14: 1645-9 (2004)
- Albaugh, PA; Marshall, L; Gregory, J; White, G; Hutchison, A; Ross, PC; Gallagher, DW; Tallman, JF; Crago, M; Cassella, JV J Med Chem 45: 5043-51 (2002)
- Huang, D; Poon, SF; Chapman, DF; Chung, J; Cramer, M; Reger, TS; Roppe, JR; Tehrani, L; Cosford, ND; Smith, ND Bioorg Med Chem Lett 14: 5473-6 (2004)
- Blum, CA; Caldwell, T; Zheng, X; Bakthavatchalam, R; Capitosti, S; Brielmann, H; De Lombaert, S; Kershaw, MT; Matson, D; Krause, JE; Cortright, D; Crandall, M; Martin, WJ; Murphy, BA; Boyce, S; Jones, AB; Mason, G; Rycroft, W; Perrett, H; Conley, R; Burnaby-Davies, N; Chenard, BL; Hodgetts, KJ J Med Chem 53: 3330-48 (2010)
- Pochetti, G; Godio, C; Mitro, N; Caruso, D; Galmozzi, A; Scurati, S; Loiodice, F; Fracchiolla, G; Tortorella, P; Laghezza, A; Lavecchia, A; Novellino, E; Mazza, F; Crestani, M J Biol Chem 282: 17314-24 (2007)
- Salimbeni, A; Paleari, F; Canevotti, R; Criscuoli, M; Criscuoli, M; Lippi, A; Angiolini, M; Belvisi, L; Scolastico, C; Colombo, L Bioorg Med Chem Lett 7: 2205-2210 (1997)
- Talukdar, A; Morgunova, E; Duan, J; Meining, W; Foloppe, N; Nilsson, L; Bacher, A; Illarionov, B; Fischer, M; Ladenstein, R; Cushman, M Bioorg Med Chem 18: 3518-34 (2010)
- Klein, SI; Molino, BF; Czekaj, M; Dener, JS; Leadley, RJ; Sabatino, R; Dunwiddie, CT; Chu, V Bioorg Med Chem Lett 6: 1403-1408 (1996)
- Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296-315 (2010)
- Cioffi, G; D'Auria, M; Braca, A; Mendez, J; Castillo, A; Morelli, I; De Simone, F; De Tommasi, N J Nat Prod 65: 1526-9 (2002)
- Shi, J; Gu, Z; Jurica, EA; Wu, X; Haque, LE; Williams, KN; Hernandez, AS; Hong, Z; Gao, Q; Dabros, M; Davulcu, AH; Mathur, A; Rampulla, RA; Gupta, AK; Jayaram, R; Apedo, A; Moore, DB; Liu, H; Kunselman, LK; Brady, EJ; Wilkes, JJ; Zinker, BA; Cai, H; Shu, YZ; Sun, Q; Dierks, EA; Foster, KA; Xu, C; Wang, T; Panemangalore, R; Cvijic, ME; Xie, C; Cao, GG; Zhou, M; Krupinski, J; Whaley, JM; Robl, JA; Ewing, WR; Ellsworth, BA J Med Chem 61: 681-694 (2018)
- Hamilton, NM; Dawson, M; Fairweather, EE; Hamilton, NS; Hitchin, JR; James, DI; Jones, SD; Jordan, AM; Lyons, AJ; Small, HF; Thomson, GJ; Waddell, ID; Ogilvie, DJ J Med Chem 55: 4431-45 (2012)
- Hemmerling, M; Edman, K; Lepistö, M; Eriksson, A; Ivanova, S; Dahmén, J; Rehwinkel, H; Berger, M; Hendrickx, R; Dearman, M; Jensen, TJ; Wissler, L; Hansson, T Bioorg Med Chem Lett 26: 5741-5748 (2016)
- Brak, K; Kerr, ID; Barrett, KT; Fuchi, N; Debnath, M; Ang, K; Engel, JC; McKerrow, JH; Doyle, PS; Brinen, LS; Ellman, JA J Med Chem 53: 1763-73 (2010)
- Dechantsreiter, M; Grob, JE; Macsweeney, A; Miltz, W; Randl, SA; Sedrani, R; Sellner, H; Sirockin, F; Valeur, E US Patent US9452990 (2016)
- Hoefgen, B; Decker, M; Mohr, P; Schramm, AM; Rostom, SA; El-Subbagh, H; Schweikert, PM; Rudolf, DR; Kassack, MU; Lehmann, J J Med Chem 49: 760-9 (2006)
- Zeinyeh, W; Esvan, YJ; Josselin, B; Defois, M; Baratte, B; Knapp, S; Chaikuad, A; Anizon, F; Giraud, F; Ruchaud, S; Moreau, P Eur J Med Chem 236: (2022)
- Mejdrová, I; Chalupská, D; Placková, P; Müller, C; ?ála, M; Klíma, M; Baumlová, A; Hrebabecký, H; Procházková, E; Dejmek, M; Strunin, D; Weber, J; Lee, G; Matou?ová, M; Mertlíková-Kaiserová, H; Ziebuhr, J; Birkus, G; Boura, E; Nencka, R J Med Chem 60: 100-118 (2017)
- Armani, E; Amari, G; Rizzi, A; De Fanti, R; Ghidini, E; Capaldi, C; Carzaniga, L; Caruso, P; Guala, M; Peretto, I; La Porta, E; Bolzoni, PT; Facchinetti, F; Carnini, C; Moretto, N; Patacchini, R; Bassani, F; Cenacchi, V; Volta, R; Amadei, F; Capacchi, S; Delcanale, M; Puccini, P; Catinella, S; Civelli, M; Villetti, G J Med Chem 57: 793-816 (2014)
- Shishodia, S; Demetriades, M; Zhang, D; Tam, NY; Maheswaran, P; Clunie-O'Connor, C; Tumber, A; Leung, IKH; Ng, YM; Leissing, TM; El-Sagheer, AH; Salah, E; Brown, T; Aik, WS; McDonough, MA; Schofield, CJ J Med Chem 64: 16609-16625 (2021)
- Tian, C; Yang, C; Wu, T; Lu, M; Chen, Y; Yang, Y; Liu, X; Ling, Y; Deng, M; Jia, Y; Zhou, Y Bioorg Med Chem Lett 48: (2021)
- Poel, TJ; Thomas, RC; Adams, WJ; Aristoff, PA; Barbachyn, MR; Boyer, FE; Brieland, J; Brideau, R; Brodfuehrer, J; Brown, AP; Choy, AL; Dermyer, M; Dority, M; Ford, CW; Gadwood, RC; Hanna, D; Hongliang, C; Huband, MD; Huber, C; Kelly, R; Kim, JY; Martin, JP; Pagano, PJ; Ross, D; Skerlos, L; Sulavik, MC; Zhu, T; Zurenko, GE; Prasad, JV J Med Chem 50: 5886-9 (2007)
- Wiles, JA; Phadke, AS; Deshpande, M; Agarwal, A; Chen, D; Gadhachanda, VR; Hashimoto, A; Pais, G; Wang, Q; Wang, X; Greenlee, W US Patent US11407738 (2022)
- Desjardins, M; Desgagnes, J; Lacoste, L; Yang, F; Morin, M; Lapointe, J; Chenevert, R Bioorg Med Chem Lett 7: 2363-2366 (1997)
- Kozlova, A; Thabault, L; Dauguet, N; Deskeuvre, M; Stroobant, V; Pilotte, L; Liberelle, M; Van den Eynde, B; Frédérick, R Eur J Med Chem 227: (2022)
- Xiao, Y; Karra, S; Goutopoulos, A; Morse, NT; Zhang, S; Dhanabal, M; Tian, H; Seenisamy, J; Jayadevan, J; Caldwell, R; Potnick, J; Bleich, M; Chekler, E; Sherer, B; Sriraman, V Bioorg Med Chem Lett 29: 1660-1664 (2019)
- Colabufo, NA; Berardi, F; Perrone, R; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A J Med Chem 51: 1415-22 (2008)
- Singh, A; Dirain, M; Witek, R; Rocca, JR; Edison, AS; Haskell-Luevano, C J Med Chem 56: 2747-63 (2013)
- Sinha, S; Doble, M; Manju, SL Bioorg Med Chem 27: 3745-3759 (2019)
- Wu, WL; Burnett, DA; Domalski, M; Greenlee, WJ; Li, C; Bertorelli, R; Fredduzzi, S; Lozza, G; Veltri, A; Reggiani, A J Med Chem 50: 5550-3 (2007)
- Parcella, K; Eastman, K; Yeung, KS; Grant-Young, KA; Zhu, J; Wang, T; Zhang, Z; Yin, Z; Parker, D; Mosure, K; Fang, H; Wang, YK; Lemm, J; Zhuo, X; Hanumegowda, U; Liu, M; Rigat, K; Donoso, M; Tuttle, M; Zvyaga, T; Haarhoff, Z; Meanwell, NA; Soars, MG; Roberts, SB; Kadow, JF ACS Med Chem Lett 8: 771-774 (2017)
- Poel, TJ; Thomas, RC; Adams, WJ; Aristoff, PA; Barbachyn, MR; Boyer, FE; Brieland, J; Brideau, R; Brodfuehrer, J; Brown, AP; Choy, AL; Dermyer, M; Dority, M; Ford, CW; Gadwood, RC; Hanna, D; Hongliang, C; Huband, MD; Huber, C; Kelly, R; Kim, JY; Martin, JP; Pagano, PJ; Ross, D; Skerlos, L; Sulavik, MC; Zhu, T; Zurenko, GE; Prasad, JV J Med Chem 50: 5886-9 (2007)
- Michaelis, S; Marais, A; Schrey, AK; Graebner, OY; Schaudt, C; Sefkow, M; Kroll, F; Dreger, M; Glinski, M; Koester, H; Metternich, R; Fischer, JJ J Med Chem 55: 3934-44 (2012)
- Ji, Q; Zhang, X; Du, Z; Gong, L; Wang, L; Gao, C; Du, M US Patent US11584726 (2023)
- Okolotowicz, KJ; Dwyer, M; Ryan, D; Cheng, J; Cashman, EA; Moore, S; Mercola, M; Cashman, JR Bioorg Med Chem 26: 4441-4451 (2018)
- Gray, NS; De Clercq, D; Jang, J; Janne, P; To, C; Eck, M; Park, E; Heppner, D US Patent US11584746 (2023)
- Eckhardt, M; Frattini, S; Langkopf, E; Wagner, H US Patent US9597310 (2017)
- Smith, CJ; Ali, A; Balkovec, JM; Graham, DW; Hammond, ML; Patel, GF; Rouen, GP; Smith, SK; Tata, JR; Einstein, M; Ge, L; Harris, GS; Kelly, TM; Mazur, P; Thompson, CM; Wang, CF; Williamson, JM; Miller, DK; Pandit, S; Santoro, JC; Sitlani, A; Yamin, TT; O'Neill, EA; Zaller, DM; Carballo-Jane, E; Forrest, MJ; Luell, S Bioorg Med Chem Lett 15: 2926-31 (2005)
- Ojima, I; Deutsch, D; Kaczocha, M; Hu, K; Tong, S; Elmes, M; Yan, S US Patent US10968163 (2021)
- Caraballo, R; Larsson, M; Nilsson, SK; Ericsson, M; Qian, W; Nguyen Tran, NP; Kindahl, T; Svensson, R; Saar, V; Artursson, P; Olivecrona, G; Enquist, PA; Elofsson, M Eur J Med Chem 103: 191-209 (2015)
- Cee, VJ; Albrecht, BK; Geuns-Meyer, S; Hughes, P; Bellon, S; Bready, J; Caenepeel, S; Chaffee, SC; Coxon, A; Emery, M; Fretland, J; Gallant, P; Gu, Y; Hodous, BL; Hoffman, D; Johnson, RE; Kendall, R; Kim, JL; Long, AM; McGowan, D; Morrison, M; Olivieri, PR; Patel, VF; Polverino, A; Powers, D; Rose, P; Wang, L; Zhao, H J Med Chem 50: 627-40 (2007)
- Bestgen, B; Kufareva, I; Seetoh, W; Abell, C; Hartmann, RW; Abagyan, R; Le Borgne, M; Filhol, O; Cochet, C; Lomberget, T; Engel, M J Med Chem 62: 1817-1836 (2019)
- Castillo, M; Forns, P; Erra, M; Mir, M; López, M; Maldonado, M; Orellana, A; Carreño, C; Ramis, I; Miralpeix, M; Vidal, B Bioorg Med Chem Lett 22: 5419-23 (2012)
- Gogate, PN; Ethirajan, M; Kurenova, EV; Magis, AT; Pandey, RK; Cance, WG Eur J Med Chem 80: 154-66 (2014)
- Furber, M; Alcaraz, L; Bent, JE; Beyerbach, A; Bowers, K; Braddock, M; Caffrey, MV; Cladingboel, D; Collington, J; Donald, DK; Fagura, M; Ince, F; Kinchin, EC; Laurent, C; Lawson, M; Luker, TJ; Mortimore, MM; Pimm, AD; Riley, RJ; Roberts, N; Robertson, M; Theaker, J; Thorne, PV; Weaver, R; Webborn, P; Willis, P J Med Chem 50: 5882-5 (2007)
- Manca, I; Mastinu, A; Olimpieri, F; Falzoi, M; Sani, M; Ruiu, S; Loriga, G; Volonterio, A; Tambaro, S; Bottazzi, ME; Zanda, M; Pinna, GA; Lazzari, P Eur J Med Chem 62: 256-69 (2013)
- Maccallini, C; Arias, F; Gallorini, M; Amoia, P; Ammazzalorso, A; De Filippis, B; Fantacuzzi, M; Giampietro, L; Cataldi, A; Camacho, ME; Amoroso, R ACS Med Chem Lett 11: 1470-1475 (2020)
- Fantini, M; Rivara, M; Zuliani, V; Kalmar, CL; Vacondio, F; Silva, C; Baheti, AR; Singh, N; Merrick, EC; Katari, RS; Cocconcelli, G; Ghiron, C; Patel, MK Bioorg Med Chem 17: 3642-8 (2009)
- Fardis, M; Jin, H; Jabri, S; Cai, RZ; Mish, M; Tsiang, M; Kim, CU Bioorg Med Chem Lett 16: 4031-5 (2006)
- Laufer, R; Forrest, B; Li, SW; Liu, Y; Sampson, P; Edwards, L; Lang, Y; Awrey, DE; Mao, G; Plotnikova, O; Leung, G; Hodgson, R; Beletskaya, I; Mason, JM; Luo, X; Wei, X; Yao, Y; Feher, M; Ban, F; Kiarash, R; Green, E; Mak, TW; Pan, G; Pauls, HW J Med Chem 56: 6069-87 (2013)
- Feledziak, M; Michaux, C; Urbach, A; Labar, G; Muccioli, GG; Lambert, DM; Marchand-Brynaert, J J Med Chem 52: 7054-68 (2009)
- Zhang, S; Chen, X; Wu, C; Xu, H; Xie, X; Feng, M; Hu, S; Bai, H; Gao, F; Tong, L; Ding, J; Liu, H; Xie, Z; Wang, J J Med Chem 65: 7697-7716 (2022)
- Zampieri, D; Laurini, E; Vio, L; Fermeglia, M; Pricl, S; Wünsch, B; Schepmann, D; Mamolo, MG Eur J Med Chem 90: 797-808 (2015)
- Narjes, F; Crescenzi, B; Ferrara, M; Habermann, J; Colarusso, S; Ferreira, Mdel R; Stansfield, I; Mackay, AC; Conte, I; Ercolani, C; Zaramella, S; Palumbi, MC; Meuleman, P; Leroux-Roels, G; Giuliano, C; Fiore, F; Di Marco, S; Baiocco, P; Koch, U; Migliaccio, G; Altamura, S; Laufer, R; De Francesco, R; Rowley, M J Med Chem 54: 289-301 (2011)
- Nocentini, A; Ferraroni, M; Carta, F; Ceruso, M; Gratteri, P; Lanzi, C; Masini, E; Supuran, CT J Med Chem 59: 10692-10704 (2016)
- Haworth, KE; Harrison, T; Kulagowski, JJ; Leeson, PD; Owens, AP; Ridgill, MP; Teall, MR; Fielding, M; Chapman, K; Emms, F; Marwood, R; Patel, S; Moss, KL Bioorg Med Chem Lett 7: 2211-2216 (1997)
- Chakraborty, S; DiBerto, JF; Faouzi, A; Bernhard, SM; Gutridge, AM; Ramsey, S; Zhou, Y; Provasi, D; Nuthikattu, N; Jilakara, R; Nelson, MNF; Asher, WB; Eans, SO; Wilson, LL; Chintala, SM; Filizola, M; van Rijn, RM; Margolis, EB; Roth, BL; McLaughlin, JP; Che, T; Sames, D; Javitch, JA; Majumdar, S J Med Chem 64: 13873-13892 (2021)
- Bornot, A; Bauer, U; Brown, A; Firth, M; Hellawell, C; Engkvist, O J Med Chem 56: 1197-210 (2013)
- Zahid, H; Buchholz, CR; Singh, M; Ciccone, MF; Chan, A; Nithianantham, S; Shi, K; Aihara, H; Fischer, M; Schönbrunn, E; Dos Santos, CO; Landry, JW; Pomerantz, WCK J Med Chem 64: 13902-13917 (2021)
- Matthews, TP; McHardy, T; Klair, S; Boxall, K; Fisher, M; Cherry, M; Allen, CE; Addison, GJ; Ellard, J; Aherne, GW; Westwood, IM; van Montfort, R; Garrett, MD; Reader, JC; Collins, I Bioorg Med Chem Lett 20: 4045-9 (2010)
- Xiang, Y; Hirth, B; Asmussen, G; Biemann, HP; Bishop, KA; Good, A; Fitzgerald, M; Gladysheva, T; Jain, A; Jancsics, K; Liu, J; Metz, M; Papoulis, A; Skerlj, R; Stepp, JD; Wei, RR Bioorg Med Chem Lett 21: 3050-6 (2011)
- Fleck, M; Heine, N; Nosse, B; Roth, GJ; Heimann, A US Patent US9169205 (2015)
- Hughes, AD; Byun, D; Chen, Y; Fleury, M; Jacobsen, JR; Stangeland, EL; Wilson, RD; Yen, R US Patent US9572802 (2017)
- Pedreira, JGB; Nahidino, P; Kudolo, M; Pantsar, T; Berger, BT; Forster, M; Knapp, S; Laufer, S; Barreiro, EJ J Med Chem 63: 7347-7354 (2020)
- Merlino, F; Daniele, S; La Pietra, V; Di Maro, S; Di Leva, FS; Brancaccio, D; Tomassi, S; Giuntini, S; Cerofolini, L; Fragai, M; Luchinat, C; Reichart, F; Cavallini, C; Costa, B; Piccarducci, R; Taliani, S; Da Settimo, F; Martini, C; Kessler, H; Novellino, E; Marinelli, L J Med Chem 61: 4791-4809 (2018)
- Desage-El Murr, M; Cano, C; Golding, BT; Hardcastle, IR; Hummersome, M; Frigerio, M; Curtin, NJ; Menear, K; Richardson, C; Smith, GC; Griffin, RJ Bioorg Med Chem Lett 18: 4885-90 (2008)
- Frizler, M; Lohr, F; Furtmann, N; Kläs, J; Gütschow, M J Med Chem 54: 396-400 (2011)
- Sapkota, GP; Cummings, L; Newell, FS; Armstrong, C; Bain, J; Frodin, M; Grauert, M; Hoffmann, M; Schnapp, G; Steegmaier, M; Cohen, P; Alessi, DR Biochem J 401: 29-38 (2007)
- Hartmann, R; Frotscher, M; Oberwinkler, S; Ziegler, E; Messinger, J; Thole, H US Patent US8546392 (2013)
- Li, Z; Pan, M; Su, X; Dai, Y; Fu, M; Cai, X; Shi, W; Huang, W; Qian, H Bioorg Med Chem 24: 1981-7 (2016)
- Gilbert, J; Fuentes, M; Ojasoo, T; Doré, JC; Pons, M J Med Chem 40: 1104-11 (1997)
- Shiryaev, SA; Remacle, AG; Ratnikov, BI; Nelson, NA; Savinov, AY; Wei, G; Bottini, M; Rega, MF; Parent, A; Desjardins, R; Fugere, M; Day, R; Sabet, M; Pellecchia, M; Liddington, RC; Smith, JW; Mustelin, T; Guiney, DG; Lebl, M; Strongin, AY J Biol Chem 282: 20847-53 (2007)
- Kiyama, R; Honma, T; Hayashi, K; Ogawa, M; Hara, M; Fujimoto, M; Fujishita, T J Med Chem 38: 2728-41 (1995)
- Fukunaga, K; Uehara, F; Aritomo, K; Shoda, A; Hiki, S; Okuyama, M; Usui, Y; Watanabe, K; Yamakoshi, K; Kohara, T; Hanano, T; Tanaka, H; Tsuchiya, S; Sunada, S; Saito, K; Eguchi, J; Yuki, S; Asano, S; Tanaka, S; Mori, A; Yamagami, K; Baba, H; Horikawa, T; Fujimura, M Bioorg Med Chem Lett 23: 6933-7 (2013)
- Kumata, K; Yui, J; Hatori, A; Fujinaga, M; Yanamoto, K; Yamasaki, T; Kawamura, K; Wakizaka, H; Nengaki, N; Yoshida, Y; Ogawa, M; Fukumura, T; Zhang, MR J Med Chem 54: 6040-9 (2011)
- Pike, VW; Rash, KS; Chen, Z; Pedregal, C; Statnick, MA; Kimura, Y; Hong, J; Zoghbi, SS; Fujita, M; Toledo, MA; Diaz, N; Gackenheimer, SL; Tauscher, JT; Barth, VN; Innis, RB J Med Chem 54: 2687-700 (2011)
- Fukuda, M; Sasaki, T; Hashimoto, T; Miyachi, H; Waki, M; Asai, A; Takikawa, O; Ohno, O; Matsuno, K Bioorg Med Chem Lett 28: 2846-2849 (2018)
- Ueda, T; Ito, T; Tomita, K; Togame, H; Fumoto, M; Asakura, K; Oshima, T; Nishimura, S; Hanasaki, K Bioorg Med Chem Lett 20: 4631-4 (2010)
- Czudor, Z; Balogh, M; Bánhegyi, P; Boros, S; Breza, N; Dobos, J; Fábián, M; Horváth, Z; Illyés, E; Markó, P; Sipos, A; Szántai-Kis, C; Szokol, B; ?rfi, L Bioorg Med Chem Lett 28: 769-773 (2018)
- Banville, J; Rémillard, R; Ruediger, EH; Deon, DH; Gagnon, M; Dubé, L; Guy, J; Priestley, ES; Posy, SL; Maxwell, BD; Wong, PC; Lawrence, RM; Miller, MM US Patent US9688695 (2017)
- Su, S; Clarke, A; Han, Y; Chao, HJ; Bostwick, J; Schumacher, W; Wang, T; Yan, M; Hsu, MY; Simmons, E; Luk, C; Xu, C; Dabros, M; Galella, M; Onorato, J; Gordon, D; Wexler, R; Gargalovic, PS; Lawrence, RM J Med Chem 62: 10456-10465 (2019)
- Meziane-Cherif, D; Lambert, T; Dupêchez, M; Courvalin, P; Galimand, M Antimicrob Agents Chemother 52: 1264-8 (2008)
- Macdonald, D; Mastracchio, A; Perrier, H; Dubé, D; Gallant, M; Lacombe, P; Deschênes, D; Roy, B; Scheigetz, J; Bateman, K; Li, C; Trimble, LA; Day, S; Chauret, N; Nicoll-Griffith, DA; Silva, JM; Huang, Z; Laliberté, F; Liu, S; Ethier, D; Pon, D; Muise, E; Boulet, L; Chan, CC; Styhler, A; Charleson, S; Mancini, J; Masson, P; Claveau, D; Nicholson, D; Turner, M; Young, RN; Girard, Y Bioorg Med Chem Lett 15: 5241-6 (2005)
- Maccallini, C; Arias, F; Gallorini, M; Amoia, P; Ammazzalorso, A; De Filippis, B; Fantacuzzi, M; Giampietro, L; Cataldi, A; Camacho, ME; Amoroso, R ACS Med Chem Lett 11: 1470-1475 (2020)
- Mahasenan, KV; Ding, D; Gao, M; Nguyen, TT; Suckow, MA; Schroeder, VA; Wolter, WR; Chang, M; Mobashery, S ACS Med Chem Lett 9: 708-713 (2018)
- Moss, N; Beaulieu, P; Duceppe, JS; Ferland, JM; Garneau, M; Gauthier, J; Ghiro, E; Goulet, S; Guse, I; Jaramillo, J; Llinas-Brunet, M; Malenfant, E; Plante, R; Poirier, M; Soucy, F; Wernic, D; Yoakim, C; Déziel, R J Med Chem 39: 4173-80 (1996)
- Gazvoda, M; Beranic, N; Turk, S; Burja, B; Kocevar, M; Rižner, TL; Gobec, S; Polanc, S Eur J Med Chem 62: 89-97 (2013)
- ?apkauskait?, E; Zak?auskas, A; Ruibys, V; Linkuvien?, V; Paketuryt?, V; Gedgaudas, M; Kairys, V; Matulis, D Bioorg Med Chem 26: 675-687 (2018)
- Tao, Z; Barker, J; Shi, SD; Gehring, M; Sun, S Biochemistry 49: 8488-98 (2010)
- Geitmann, M; Retra, K; de Kloe, GE; Homan, E; Smit, AB; de Esch, IJ; Danielson, UH Biochemistry 49: 8143-54 (2010)
- Ding, P; Gelman, M; Kinsella, T; Singh, R; Bhamidipati, S; Velaparthi, U; Borzilleri, RM; Rahaman, H; Warrier, JS US Patent US9981944 (2018)
- Zhang, A; Ding, J; Xie, H; Song, Z; Xue, Y; Tong, L; Geng, M US Patent US10829491 (2020)
- Gerasimov, M; Marona-Lewicka, D; Kurrasch-Orbaugh, DM; Qandil, AM; Nichols, DE J Med Chem 42: 4257-63 (1999)
- Defaux, J; Antoine, M; Logé, C; Le Borgne, M; Schuster, T; Seipelt, I; Aicher, B; Teifel, M; Günther, E; Gerlach, M; Marchand, P Bioorg Med Chem Lett 24: 3748-52 (2014)
- Sadeghzadeh, M; Sheibani, S; Ghandi, M; Daha, FJ; Amanlou, M; Arjmand, M; Hasani Bozcheloie, A Eur J Med Chem 64: 488-97 (2013)
- Li, L; Chenna, BC; Yang, KS; Cole, TR; Goodall, ZT; Giardini, M; Moghadamchargari, Z; Hernandez, EA; Gomez, J; Calvet, CM; Bernatchez, JA; Mellott, DM; Zhu, J; Rademacher, A; Thomas, D; Blankenship, LR; Drelich, A; Laganowsky, A; Tseng, CK; Liu, WR; Wand, AJ; Cruz-Reyes, J; Siqueira-Neto, JL; Meek, TD J Med Chem 64: 11267-11287 (2021)
- Burns, CJ; Harte, MF; Bu, X; Fantino, E; Giarrusso, M; Joffe, M; Kurek, M; Legge, FS; Razzino, P; Su, S; Treutlein, H; Wan, SS; Zeng, J; Wilks, AF Bioorg Med Chem Lett 19: 1206-9 (2009)
- Köse, M; Ritter, K; Thiemke, K; Gillard, M; Kostenis, E; Müller, CE ACS Med Chem Lett 5: 326-30 (2014)
- Bharathan, IT; Blackburn, C; Ciavarri, JP; Chouitar, J; Cullis, CA; D Amore, N; Fleming, PE; Gigstad, KM; Gipson, KE; Girard, M; Hu, Y; Lee, J; Li, G; Rezaei, M; Sintchak, MD; Soucy, F; Stroud, SG; Vos, TJ; Xu, H; Ye, Y US Patent US10202373 (2019)
- Cooper, AG; MacDonald, C; Glass, M; Hook, S; Tyndall, JDA; Vernall, AJ Eur J Med Chem 145: 770-789 (2018)
- Michaelis, S; Marais, A; Schrey, AK; Graebner, OY; Schaudt, C; Sefkow, M; Kroll, F; Dreger, M; Glinski, M; Koester, H; Metternich, R; Fischer, JJ J Med Chem 55: 3934-44 (2012)
- Rahm, F; Viklund, J; Trésaugues, L; Ellermann, M; Giese, A; Ericsson, U; Forsblom, R; Ginman, T; Günther, J; Hallberg, K; Lindström, J; Persson, LB; Silvander, C; Talagas, A; Díaz-Sáez, L; Fedorov, O; Huber, KVM; Panagakou, I; Siejka, P; Gorjánácz, M; Bauser, M; Andersson, M J Med Chem 61: 2533-2551 (2018)
- Schwink, L; Stengelin, S; Gossel, M; Wirth, K US Patent US8552199 (2013)
- Huynh, T; Chen, Z; Pang, S; Geng, J; Bandiera, T; Bindi, S; Vianello, P; Roletto, F; Thieffine, S; Galvani, A; Vaccaro, W; Poss, MA; Trainor, GL; Lorenzi, MV; Gottardis, M; Jayaraman, L; Purandare, AV Bioorg Med Chem Lett 19: 2924-7 (2009)
- Adonias, M; Anayaba, J; Cámara, J; Canet, E; Gateau-Olesker, A; Gero, SD; Grande, M; Hernando, JI Bioorg Med Chem Lett 3: 2547-2552 (1993)
- Sapkota, GP; Cummings, L; Newell, FS; Armstrong, C; Bain, J; Frodin, M; Grauert, M; Hoffmann, M; Schnapp, G; Steegmaier, M; Cohen, P; Alessi, DR Biochem J 401: 29-38 (2007)
- Aktoudianakis, E; Cho, A; Du, Z; Graupe, M; Lad, LT; Machicao Tello, PA; Medley, JW; Metobo, SE; Mukherjee, PK; Naduthambi, D; Parkhill, EQ; Phillips, BW; Simonovich, SP; Squires, NH; Wang, P; Watkins, WJ; Xu, J; Yang, KS; Ziebenhaus, CA US Patent US10899735 (2021)
- Smith, ND; Poon, SF; Huang, D; Green, M; King, C; Tehrani, L; Roppe, JR; Chung, J; Chapman, DP; Cramer, M; Cosford, ND Bioorg Med Chem Lett 14: 5481-4 (2004)
- Zhou, H; Topiol, SW; Grenon, M; Jimenez, HN; Uberti, MA; Smith, DG; Brodbeck, RM; Chandrasena, G; Pedersen, H; Madsen, JC; Doller, D; Li, G Bioorg Med Chem Lett 23: 1398-406 (2013)
- Franchetti, P; Messini, L; Cappellacci, L; Grifantini, M; Lucacchini, A; Martini, C; Senatore, G J Med Chem 37: 2970-5 (1994)
- Liu, J; Li, AR; Wang, Y; Johnson, MG; Su, Y; Shen, W; Wang, X; Lively, S; Brown, M; Lai, S; Gonzalez Lopez De Turiso, F; Xu, Q; Van Lengerich, B; Schmitt, M; Fu, Z; Sun, Y; Lawlis, S; Seitz, L; Danao, J; Wait, J; Ye, Q; Tang, HL; Grillo, M; Collins, TL; Sullivan, TJ; Medina, JC ACS Med Chem Lett 2: 326-330 (2011)
- Jarvis, MF; Honore, P; Shieh, CC; Chapman, M; Joshi, S; Zhang, XF; Kort, M; Carroll, W; Marron, B; Atkinson, R; Thomas, J; Liu, D; Krambis, M; Liu, Y; McGaraughty, S; Chu, K; Roeloffs, R; Zhong, C; Mikusa, JP; Hernandez, G; Gauvin, D; Wade, C; Zhu, C; Pai, M; Scanio, M; Shi, L; Drizin, I; Gregg, R; Matulenko, M; Hakeem, A; Gross, M; Johnson, M; Marsh, K; Wagoner, PK; Sullivan, JP; Faltynek, CR; Krafte, DS Proc Natl Acad Sci U S A 104: 8520-5 (2007)
- Anderskewitz, R; Binder, F; Grauert, M; Grundl, M; Haebel, PW; Oost, T; Pautsch, A; Peters, S; Vintonyak, V US Patent US9713606 (2017)
- Hangeland, JJ; Friends, TJ; Doweyko, AM; Mellström, K; Sandberg, J; Grynfarb, M; Ryono, DE Bioorg Med Chem Lett 15: 4579-84 (2005)
- Redwan, IN; Dyrager, C; Solano, C; Fernández de Trocóniz, G; Voisin, L; Bliman, D; Meloche, S; Grřtli, M Eur J Med Chem 85: 127-38 (2014)
- Ceccarelli, SM; Chomienne, O; Gubler, M; Arduini, A J Med Chem 54: 3109-52 (2011)
- Guerrero, M; Urbano, M; Schaeffer, MT; Brown, S; Rosen, H; Roberts, E Bioorg Med Chem Lett 23: 614-9 (2013)
- Liu, J; He, S; Jian, T; Dobbelaar, PH; Sebhat, IK; Lin, LS; Goodman, A; Guo, C; Guzzo, PR; Hadden, M; Henderson, AJ; Pattamana, K; Ruenz, M; Sargent, BJ; Swenson, B; Yet, L; Tamvakopoulos, C; Peng, Q; Pan, J; Kan, Y; Palyha, O; Kelly, TM; Guan, XM; Howard, AD; Marsh, DJ; Metzger, JM; Reitman, ML; Wyvratt, MJ; Nargund, RP Bioorg Med Chem Lett 20: 2074-7 (2010)
- Yoshimoto, N; Sakamaki, Y; Haeta, M; Kato, A; Inaba, Y; Itoh, T; Nakabayashi, M; Ito, N; Yamamoto, K J Med Chem 55: 4373-81 (2012)
- Ogawa, T; Miyamae, T; Murayama, K; Okuyama, K; Okayama, T; Hagiwara, M; Sakurada, S; Morikawa, T J Med Chem 45: 5081-9 (2002)
- Hahn, M; Rogers, D J Med Chem 38: 2091-102 (1995)
- Endo, J; Hikawa, H; Hamada, M; Ishibuchi, S; Fujie, N; Sugiyama, N; Tanaka, M; Kobayashi, H; Sugahara, K; Oshita, K; Iwata, K; Ooike, S; Murata, M; Sumichika, H; Chiba, K; Adachi, K Bioorg Med Chem Lett 26: 1365-70 (2016)
- Rueda, DC; Schöffmann, A; De Mieri, M; Raith, M; Jähne, EA; Hering, S; Hamburger, M Bioorg Med Chem 22: 1276-84 (2014)
- Sisay, MT; Steinmetzer, T; Stirnberg, M; Maurer, E; Hammami, M; Bajorath, J; Gütschow, M J Med Chem 53: 5523-35 (2010)
- Hanaki, M; Murakami, K; Akagi, K; Irie, K Bioorg Med Chem 24: 304-13 (2016)
- Ashraf, A; Ejaz, SA; Rahman, SU; Siddiqui, WA; Arshad, MN; Lecka, J; Sévigny, J; Zayed, MEM; Asiri, AM; Iqbal, J; Hartinger, CG; Hanif, M Eur J Med Chem 159: 282-291 (2018)
- Kiyama, R; Honma, T; Hayashi, K; Ogawa, M; Hara, M; Fujimoto, M; Fujishita, T J Med Chem 38: 2728-41 (1995)
- Shiraishi, T; Kadono, S; Haramura, M; Kodama, H; Ono, Y; Iikura, H; Esaki, T; Koga, T; Hattori, K; Watanabe, Y; Sakamoto, A; Yoshihashi, K; Kitazawa, T; Esaki, K; Ohta, M; Sato, H; Kozono, T Bioorg Med Chem Lett 18: 4533-7 (2008)
- Ono, M; Yoshida, N; Ishibashi, K; Haratake, M; Arano, Y; Mori, H; Nakayama, M J Med Chem 48: 7253-60 (2005)
- Halim, R; Harding, M; Hufton, R; Morton, CJ; Jahangiri, S; Pool, BR; Jeynes, TP; Draffan, AG; Frey, B; Lilly, MJ US Patent US8546389 (2013)
- Wu, S; Fluxe, A; Sheffer, J; Janusz, JM; Blass, BE; White, R; Jackson, C; Hedges, R; Murawsky, M; Fang, B; Fadayel, GM; Hare, M; Djandjighian, L Bioorg Med Chem Lett 16: 6213-8 (2006)
- Jiao, X; Kopecky, DJ; Fisher, B; Piper, DE; Labelle, M; McKendry, S; Harrison, M; Jones, S; Jaen, J; Shiau, AK; Escaron, P; Danao, J; Chai, A; Coward, P; Kayser, F Bioorg Med Chem Lett 22: 5966-70 (2012)
- Vanjare, BD; Choi, NG; Mahajan, PG; Raza, H; Hassan, M; Han, Y; Yu, SM; Kim, SJ; Seo, SY; Lee, KH Bioorg Med Chem 41: (2021)
- Kawahata, N; Yang, MG; Luke, GP; Shakespeare, WC; Sundaramoorthi, R; Wang, Y; Johnson, D; Merry, T; Violette, S; Guan, W; Bartlett, C; Smith, J; Hatada, M; Lu, X; Dalgarno, DC; Eyermann, CJ; Bohacek, RS; Sawyer, TK Bioorg Med Chem Lett 11: 2319-23 (2001)
- Pettersson, I; Ebdrup, S; Havranek, M; Pihera, P; Korínek, M; Mogensen, JP; Jeppesen, CB; Johansson, E; Sauerberg, P Bioorg Med Chem Lett 17: 4625-9 (2007)
- Hayakawa, M; Kawaguchi, K; Kaizawa, H; Koizumi, T; Ohishi, T; Yamano, M; Okada, M; Ohta, M; Tsukamoto, S; Raynaud, FI; Parker, P; Workman, P; Waterfield, MD Bioorg Med Chem 15: 5837-44 (2007)
- Zhang, M; Jiang, L; Tao, J; Pan, Z; He, M; Su, D; He, G; Jiang, Q Bioorg Med Chem 27: 2268-2279 (2019)
- Wermuth, CG; Bourguignon, JJ; Schlewer, G; Gies, JP; Schoenfelder, A; Melikian, A; Bouchet, MJ; Chantreux, D; Molimard, JC; Heaulme, M J Med Chem 30: 239-49 (1987)
- Fensome, A; Ambler, CM; Arnold, E; Banker, ME; Brown, MF; Chrencik, J; Clark, JD; Dowty, ME; Efremov, IV; Flick, A; Gerstenberger, BS; Gopalsamy, A; Hayward, MM; Hegen, M; Hollingshead, BD; Jussif, J; Knafels, JD; Limburg, DC; Lin, D; Lin, TH; Pierce, BS; Saiah, E; Sharma, R; Symanowicz, PT; Telliez, JB; Trujillo, JI; Vajdos, FF; Vincent, F; Wan, ZK; Xing, L; Yang, X; Yang, X; Zhang, L J Med Chem 61: 8597-8612 (2018)
- Williamson, DS; Smith, GP; Mikkelsen, GK; Jensen, T; Acheson-Dossang, P; Badolo, L; Bedford, ST; Chell, V; Chen, IJ; Dokurno, P; Hentzer, M; Newland, S; Ray, SC; Shaw, T; Surgenor, AE; Terry, L; Wang, Y; Christensen, KV J Med Chem 64: 10312-10332 (2021)
- Humphries, PS; Bailey, S; Almaden, JV; Barnum, SJ; Carlson, TJ; Christie, LC; Do, QQ; Fraser, JD; Hess, M; Kellum, J; Kim, YH; McClellan, GA; Ogilvie, KM; Simmons, BH; Skalitzky, D; Sun, S; Wilhite, D; Zehnder, LR Bioorg Med Chem Lett 16: 6120-3 (2006)
- Matyskiela, ME; Zhang, W; Man, HW; Muller, G; Khambatta, G; Baculi, F; Hickman, M; LeBrun, L; Pagarigan, B; Carmel, G; Lu, CC; Lu, G; Riley, M; Satoh, Y; Schafer, P; Daniel, TO; Carmichael, J; Cathers, BE; Chamberlain, PP J Med Chem 61: 535-542 (2017)
- Flesch, D; Ness, J; Lamers, C; Dehm, F; Popella, S; Steri, R; Ogorek, I; Hieke, M; Dannhardt, G; Werz, O; Weggen, S; Schubert-Zsilavecz, M Bioorg Med Chem Lett 25: 841-6 (2015)
- Lacivita, E; De Giorgio, P; Lee, IT; Rodeheaver, SI; Weiss, BA; Fracasso, C; Caccia, S; Berardi, F; Perrone, R; Zhang, MR; Maeda, J; Higuchi, M; Suhara, T; Schetz, JA; Leopoldo, M J Med Chem 53: 7344-55 (2010)
- Sakamoto, T; Koga, Y; Hikota, M; Matsuki, K; Murakami, M; Kikkawa, K; Fujishige, K; Kotera, J; Omori, K; Morimoto, H; Yamada, K Bioorg Med Chem Lett 24: 5175-80 (2014)
- Ma, B; Metrick, CM; Gu, C; Hoemberger, M; Bajrami, B; Bame, E; Huang, J; Mingueneau, M; Murugan, P; Santoro, JC; Tang, H; Wang, T; Hopkins, BT Bioorg Med Chem Lett 60: (2022)
- Sapkota, GP; Cummings, L; Newell, FS; Armstrong, C; Bain, J; Frodin, M; Grauert, M; Hoffmann, M; Schnapp, G; Steegmaier, M; Cohen, P; Alessi, DR Biochem J 401: 29-38 (2007)
- Levin, JI; Chen, J; Du, M; Hogan, M; Kincaid, S; Nelson, FC; Venkatesan, AM; Wehr, T; Zask, A; DiJoseph, J; Killar, LM; Skala, S; Sung, A; Sharr, M; Roth, C; Jin, G; Cowling, R; Mohler, KM; Black, RA; March, CJ; Skotnicki, JS Bioorg Med Chem Lett 11: 2189-92 (2001)
- Nomura, S; Sakamaki, S; Hongu, M; Kawanishi, E; Koga, Y; Sakamoto, T; Yamamoto, Y; Ueta, K; Kimata, H; Nakayama, K; Tsuda-Tsukimoto, M J Med Chem 53: 6355-60 (2010)
- Pinkerton, AB; Sessions, EH; Hershberger, P; Maloney, PR; Peddibhotla, S; Hopf, M; Sergienko, E; Ma, CT; Smith, LH; Jackson, MR; Tanaka, J; Tsuji, T; Akiu, M; Cohen, SE; Nakamura, T; Gardell, SJ Bioorg Med Chem Lett 41: (2021)
- Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A ACS Med Chem Lett 4: 1163-8 (2013)
- Qiu, Z; Lin, X; Zhou, M; Liu, Y; Zhu, W; Chen, W; Zhang, W; Guo, L; Liu, H; Wu, G; Huang, M; Jiang, M; Xu, Z; Zhou, Z; Qin, N; Ren, S; Qiu, H; Zhong, S; Zhang, Y; Zhang, Y; Wu, X; Shi, L; Shen, F; Mao, Y; Zhou, X; Yang, W; Wu, JZ; Yang, G; Mayweg, AV; Shen, HC; Tang, G J Med Chem 59: 7651-66 (2016)
- Desage-El Murr, M; Cano, C; Golding, BT; Hardcastle, IR; Hummersome, M; Frigerio, M; Curtin, NJ; Menear, K; Richardson, C; Smith, GC; Griffin, RJ Bioorg Med Chem Lett 18: 4885-90 (2008)
- Novellino, E; Abignente, E; Cosimelli, B; Greco, G; Iadanza, M; Laneri, S; Lavecchia, A; Rimoli, MG; Settimo, FD; Primofiore, G; Tuscano, D; Trincavelli, L; Martini, C J Med Chem 45: 5030-6 (2002)
- Ichikawa, M; Ohtsuka, M; Ohki, H; Haginoya, N; Itoh, M; Sugita, K; Usui, H; Suzuki, M; Terayama, K; Kanda, A Bioorg Med Chem 20: 3072-93 (2012)
- Devillers, I; Pevet, I; Jacobelli, H; Durand, C; Fasquelle, V; Puaud, J; Gaudillière, B; Idrissi, M; Moreau, F; Wrigglesworth, R Bioorg Med Chem Lett 14: 3303-6 (2004)
- Zhang, X; Raghavan, S; Ihnat, M; Hamel, E; Zammiello, C; Bastian, A; Mooberry, SL; Gangjee, A Bioorg Med Chem 23: 2408-23 (2015)
- Kitagawa, H; Ozawa, T; Takahata, S; Iida, M Bioorg Med Chem Lett 17: 4982-6 (2007)
- Ilic, M; Ilaš, J; Dunkel, P; Mátyus, P; Bohác, A; Liekens, S; Kikelj, D Eur J Med Chem 58: 160-70 (2012)
- Kalaba, P; Aher, NY; Ili?, M; Draga?evi?, V; Wieder, M; Miklosi, AG; Zehl, M; Wackerlig, J; Roller, A; Beryozkina, T; Radoman, B; Saroja, SR; Lindner, W; Gonzalez, EP; Bakulev, V; Leban, JJ; Sitte, HH; Urban, E; Langer, T; Lubec, G J Med Chem 60: 9330-9348 (2017)
- Fujimoto, J; Okamoto, R; Noguchi, N; Hara, R; Masada, S; Kawamoto, T; Nagase, H; Tamura, YO; Imanishi, M; Takagahara, S; Kubo, K; Tohyama, K; Iida, K; Andou, T; Miyahisa, I; Matsui, J; Hayashi, R; Maekawa, T; Matsunaga, N J Med Chem 60: 8963-8981 (2017)
- Babine, RE; Bleckman, TM; Littlefield, ES; Parge, HE; Pelletier, LA; Lewis, CT; French, JV; Imbacuan, M; Katoh, S; Tatlock, JH; Showalter, RE; Villafranca, JE Bioorg Med Chem Lett 6: 385-390 (1996)
- Nagata, T; Inoue, M; Ashida, Y; Noguchi, K; Ono, M US Patent US8609710 (2013)
- Bhamidipati, S; Shaw, S; Darwish, I; Yu, J; Kolluri, R; Taylor, V; Masuda, E; Irving, M US Patent US11667643 (2023)
- Nishiyama, Y; Mori, S; Makishima, M; Fujii, S; Kagechika, H; Hashimoto, Y; Ishikawa, M ACS Med Chem Lett 9: 641-645 (2018)
- Roaten, JB; Kazanietz, MG; Sweatman, TW; Lothstein, L; Israel, M; Parrill, AL J Med Chem 44: 1028-34 (2001)
- Ito, M; Tanaka, T; Toita, A; Uchiyama, N; Kokubo, H; Morishita, N; Klein, MG; Zou, H; Murakami, M; Kondo, M; Sameshima, T; Araki, S; Endo, S; Kawamoto, T; Morin, GB; Aparicio, SA; Nakanishi, A; Maezaki, H; Imaeda, Y J Med Chem 61: 7710-7728 (2018)
- Saito, S; Itoh, M; Fujisawa, T; Saito, H; Kiyotsuka, Y; Watanabe, H; Matsunaga, H; Kagoshima, Y; Suzuki, T; Ogawara, Y; Kitabayashi, K US Patent US10040791 (2018)
- Shinozuka, T; Ito, S; Kimura, T; Izumi, M; Wakabayashi, K ACS Med Chem Lett 12: 817-821 (2021)
- Lacivita, E; Leopoldo, M; Masotti, AC; Inglese, C; Berardi, F; Perrone, R; Ganguly, S; Jafurulla, M; Chattopadhyay, A J Med Chem 52: 7892-6 (2009)
- Vishnu Nayak, B; Ciftci-Yabanoglu, S; Jadav, SS; Jagrat, M; Sinha, BN; Ucar, G; Jayaprakash, V Eur J Med Chem 69: 762-7 (2013)
- Jadav, P; Bahekar, R; Shah, SR; Patel, D; Joharapurkar, A; Jain, M; Sairam, KV; Singh, PK Bioorg Med Chem Lett 24: 1918-22 (2014)
- Cui, JJ; McTigue, M; Nambu, M; Tran-Dubé, M; Pairish, M; Shen, H; Jia, L; Cheng, H; Hoffman, J; Le, P; Jalaie, M; Goetz, GH; Ryan, K; Grodsky, N; Deng, YL; Parker, M; Timofeevski, S; Murray, BW; Yamazaki, S; Aguirre, S; Li, Q; Zou, H; Christensen, J J Med Chem 55: 8091-109 (2012)
- Zificsak, CA; Gingrich, DE; Breslin, HJ; Dunn, DD; Milkiewicz, KL; Theroff, JP; Thieu, TV; Underiner, TL; Weinberg, LR; Aimone, LD; Albom, MS; Mason, JL; Saville, L; Husten, J; Angeles, TS; Finn, JP; Jan, M; O'Kane, TM; Dobrzanski, P; Dorsey, BD Bioorg Med Chem Lett 22: 133-7 (2011)
- Conway, JG; McDonald, B; Parham, J; Keith, B; Rusnak, DW; Shaw, E; Jansen, M; Lin, P; Payne, A; Crosby, RM; Johnson, JH; Frick, L; Lin, MH; Depee, S; Tadepalli, S; Votta, B; James, I; Fuller, K; Chambers, TJ; Kull, FC; Chamberlain, SD; Hutchins, JT Proc Natl Acad Sci U S A 102: 16078-83 (2005)
- Thede, K; Flamme, I; Oehme, F; Ergüden, J; Stoll, F; Wild, H; Kolkhof, P; Beck, H; Jeske, M US Patent US8609698 (2013)
- Lü, Z; Li, X; Li, K; Wang, C; Du, T; Huang, W; Ji, M; Li, C; Xu, F; Xu, P; Niu, Y ACS Med Chem Lett 12: 696-703 (2021)
- Qiu, Z; Lin, X; Zhou, M; Liu, Y; Zhu, W; Chen, W; Zhang, W; Guo, L; Liu, H; Wu, G; Huang, M; Jiang, M; Xu, Z; Zhou, Z; Qin, N; Ren, S; Qiu, H; Zhong, S; Zhang, Y; Zhang, Y; Wu, X; Shi, L; Shen, F; Mao, Y; Zhou, X; Yang, W; Wu, JZ; Yang, G; Mayweg, AV; Shen, HC; Tang, G J Med Chem 59: 7651-66 (2016)
- Burns, CJ; Harte, MF; Bu, X; Fantino, E; Giarrusso, M; Joffe, M; Kurek, M; Legge, FS; Razzino, P; Su, S; Treutlein, H; Wan, SS; Zeng, J; Wilks, AF Bioorg Med Chem Lett 19: 1206-9 (2009)
- Zapf, CW; Bloom, JD; Li, Z; Dushin, RG; Nittoli, T; Otteng, M; Nikitenko, A; Golas, JM; Liu, H; Lucas, J; Boschelli, F; Vogan, E; Olland, A; Johnson, M; Levin, JI Bioorg Med Chem Lett 21: 4602-7 (2011)
- Jovanovi?, M; Zhukovsky, D; Podolski-Reni?, A; Domra?eva, I; ?alubovskis, R; Sen?anski, M; Gli?i?, S; Sharoyko, V; Tennikova, T; Dar'in, D; Pe?i?, M; Krasavin, M Eur J Med Chem 181: (2019)
- Ojima, I; Deutsch, D; Kaczocha, M; Hu, K; Tong, S; Elmes, M; Yan, S US Patent US10968163 (2021)
- Alnabulsi, S; Santina, E; Russo, I; Hussein, B; Kadirvel, M; Chadwick, A; Bichenkova, EV; Bryce, RA; Nolan, K; Demonacos, C; Stratford, IJ; Freeman, S Eur J Med Chem 111: 33-45 (2016)
- Molette, J; Routier, J; Abla, N; Besson, D; Bombrun, A; Brun, R; Burt, H; Georgi, K; Kaiser, M; Nwaka, S; Muzerelle, M; Scheer, A ACS Med Chem Lett 4: 1037-41 (2013)
- Kasai, S; Kamata, M; Masada, S; Kunitomo, J; Kamaura, M; Okawa, T; Takami, K; Ogino, H; Nakano, Y; Ashina, S; Watanabe, K; Kaisho, T; Imai, YN; Ryu, S; Nakayama, M; Nagisa, Y; Takekawa, S; Kato, K; Murata, T; Suzuki, N; Ishihara, Y J Med Chem 55: 4336-51 (2012)
- Kasai, S; Kamata, M; Masada, S; Kunitomo, J; Kamaura, M; Okawa, T; Takami, K; Ogino, H; Nakano, Y; Ashina, S; Watanabe, K; Kaisho, T; Imai, YN; Ryu, S; Nakayama, M; Nagisa, Y; Takekawa, S; Kato, K; Murata, T; Suzuki, N; Ishihara, Y J Med Chem 55: 4336-51 (2012)
- Hidaka, K; Kimura, T; Sankaranarayanan, R; Wang, J; McDaniel, KF; Kempf, DJ; Kameoka, M; Adachi, M; Kuroki, R; Nguyen, JT; Hayashi, Y; Kiso, Y J Med Chem 61: 5138-5153 (2018)
- Yamazaki, K; Hasegawa, H; Umekawa, K; Ueki, Y; Ohashi, N; Kanaoka, M Bioorg Med Chem Lett 12: 1275-8 (2002)
- Nguyen, P; Doan, P; Rimpilainen, T; Konda Mani, S; Murugesan, A; Yli-Harja, O; Candeias, NR; Kandhavelu, M J Med Chem 64: 10908-10918 (2021)
- Kim, M; Kim, G; Kang, M; Ko, D; Nam, Y; Moon, CS; Kang, HM; Shin, JS; Werz, O; Lee, KT; Lee, JY Bioorg Med Chem Lett 41: (2021)
- Keith, JM; Apodaca, R; Tichenor, M; Xiao, W; Jones, W; Pierce, J; Seierstad, M; Palmer, J; Webb, M; Karbarz, M; Scott, B; Wilson, S; Luo, L; Wennerholm, M; Chang, L; Brown, S; Rizzolio, M; Rynberg, R; Chaplan, S; Breitenbucher, JG ACS Med Chem Lett 3: 823-827 (2012)
- Fushimi, M; Fujimori, I; Wakabayashi, T; Hasui, T; Kawakita, Y; Imamura, K; Kato, T; Murakami, M; Ishii, T; Kikko, Y; Kasahara, M; Nakatani, A; Hiura, Y; Miyamoto, M; Saikatendu, K; Zou, H; Lane, SW; Lawson, JD; Imoto, H J Med Chem 62: 4915-4935 (2019)
- Vercouillie, J; Mavel, S; Galineau, L; Ragusa, T; Innis, R; Kassiou, M; Chalon, S; Dollé, F; Besnard, JC; Guilloteau, D; Emond, P Bioorg Med Chem Lett 16: 1297-300 (2006)
- Zorbaz, T; Malinak, D; Marakovi?, N; Ma?ek Hrvat, N; Zandona, A; Novotny, M; Skarka, A; Andrys, R; Benkova, M; Soukup, O; Katalini?, M; Kuca, K; Kovarik, Z; Musilek, K J Med Chem 61: 10753-10766 (2018)
- Seko, T; Kato, M; Kohno, H; Ono, S; Hashimura, K; Takimizu, H; Nakai, K; Maegawa, H; Katsube, N; Toda, M Bioorg Med Chem Lett 11: 2067-70 (2001)
- Shirai, J; Sugiyama, H; Morimoto, S; Maezaki, H; Yamamoto, Y; Okanishi, S; Kamo, I; Matsumoto, S; Ishigami, K; Inatomi, N; Imanishi, A; Kawamoto, M; Tarui, N; Hashimoto, T; Ikeura, Y Bioorg Med Chem 20: 962-77 (2012)
- Kawai, M; Nakamura, H; Sakurada, I; Shimokawa, H; Tanaka, H; Matsumizu, M; Ando, K; Hattori, K; Ohta, A; Nukui, S; Omura, A; Kawamura, M Bioorg Med Chem Lett 17: 5533-6 (2007)
- Axford, L; Boot, JR; Hotten, TM; Keenan, M; Martin, FM; Milutinovic, S; Moore, NA; O'Neill, MF; Pullar, IA; Tupper, DE; Van Belle, KR; Vivien, V Bioorg Med Chem Lett 13: 3277-80 (2003)
- She, X; Pegoli, A; Gruber, CG; Wifling, D; Carpenter, J; Hübner, H; Chen, M; Wan, J; Bernhardt, G; Gmeiner, P; Holliday, ND; Keller, M J Med Chem 63: 4133-4154 (2020)
- Jones, A; Kemp, M; Stockley, M; Gibson, K; Whitlock, G US Patent US11053198 (2021)
- Bezençon, O; Heidmann, B; Siegrist, R; Stamm, S; Richard, S; Pozzi, D; Corminboeuf, O; Roch, C; Kessler, M; Ertel, EA; Reymond, I; Pfeifer, T; de Kanter, R; Toeroek-Schafroth, M; Moccia, LG; Mawet, J; Moon, R; Rey, M; Capeleto, B; Fournier, E J Med Chem 60: 9769-9789 (2017)
- Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252-9 (2013)
- Iraji, A; Nouri, A; Edraki, N; Pirhadi, S; Khoshneviszadeh, M; Khoshneviszadeh, M Bioorg Med Chem 28: (2020)
- Kobe, A; Caaveiro, JM; Tashiro, S; Kajihara, D; Kikkawa, M; Mitani, T; Tsumoto, K J Med Chem 56: 2155-9 (2013)
- Lee, J; Jo, S; Park, AY; Lee, G; Kim, JE; Kim, M; Jung, G; Lim, SM; Lim, K; Lee, M; Yang, H; Kim, H; Kim, H; Li, W; Fan, M US Patent US10968188 (2021)
- Gilbert, AM; Kirisits, M; Toy, P; Nunn, DS; Failli, A; Dushin, EG; Novikova, E; Petersen, PJ; Joseph-McCarthy, D; McFadyen, I; Fritz, CC Bioorg Med Chem Lett 14: 37-41 (2003)
- Chen, HY; Plummer, CW; Xiao, D; Chobanian, HR; DeMong, D; Miller, M; Trujillo, ME; Kirkland, M; Kosinski, D; Mane, J; Pachanski, M; Cheewatrakoolpong, B; Di Salvo, J; Thomas-Fowlkes, B; Souza, S; Tatosian, DA; Chen, Q; Hafey, MJ; Houle, R; Nolting, AF; Orr, R; Ehrhart, J; Weinglass, AB; Tschirret-Guth, R; Howard, AD; Colletti, SL ACS Med Chem Lett 9: 685-690 (2018)
- Fallacara, AL; Passannanti, R; Mori, M; Iovenitti, G; Musumeci, F; Greco, C; Crespan, E; Kissova, M; Maga, G; Tarantelli, C; Spriano, F; Gaudio, E; Bertoni, F; Botta, M; Schenone, S Eur J Med Chem 181: (2019)
- Lehr, M; Klimt, M; Elfringhoff, AS Bioorg Med Chem Lett 11: 2569-72 (2001)
- Fyfe, MC; Knaggs, M; Meghani, P; Thom, SM US Patent US9796742 (2017)
- Gazvoda, M; Beranic, N; Turk, S; Burja, B; Kocevar, M; Rižner, TL; Gobec, S; Polanc, S Eur J Med Chem 62: 89-97 (2013)
- Ebiike, H; Taka, N; Matsushita, M; Ohmori, M; Takami, K; Hyohdoh, I; Kohchi, M; Hayase, T; Nishii, H; Morikami, K; Nakanishi, Y; Akiyama, N; Shindoh, H; Ishii, N; Isobe, T; Matsuoka, H J Med Chem 59: 10586-10600 (2016)
- Gentry, PR; Kokubo, M; Bridges, TM; Kett, NR; Harp, JM; Cho, HP; Smith, E; Chase, P; Hodder, PS; Niswender, CM; Daniels, JS; Conn, PJ; Wood, MR; Lindsley, CW J Med Chem 56: 9351-5 (2013)
- Coteron, JM; Marco, M; Esquivias, J; Deng, X; White, KL; White, J; Koltun, M; El Mazouni, F; Kokkonda, S; Katneni, K; Bhamidipati, R; Shackleford, DM; Angulo-Barturen, I; Ferrer, SB; Jiménez-Díaz, MB; Gamo, FJ; Goldsmith, EJ; Charman, WN; Bathurst, I; Floyd, D; Matthews, D; Burrows, JN; Rathod, PK; Charman, SA; Phillips, MA J Med Chem 54: 5540-61 (2011)
- Yokota, M; Imamaki, K; Uchibori, S; Kondo, M; Kosakai, K; Tomiyama, T Bioorg Med Chem Lett 3: 1687-1692 (1993)
- Klar, U; Koppitz, M; Kosemund, D; Bohlmann, R; Bader, B; Lienau, P; Siemeister, G; Prechtl, S; Nguyen, D; Scott, W US Patent US9468642 (2016)
- Wichur, T; Pasieka, A; Gody?, J; Panek, D; Góral, I; Latacz, G; Honkisz-Orzechowska, E; Bucki, A; Siwek, A; G?uch-Lutwin, M; Knez, D; Brazzolotto, X; Gobec, S; Ko?aczkowski, M; Sabate, R; Malawska, B; Wi?ckowska, A Eur J Med Chem 225: (2021)
- Jarvis, MF; Honore, P; Shieh, CC; Chapman, M; Joshi, S; Zhang, XF; Kort, M; Carroll, W; Marron, B; Atkinson, R; Thomas, J; Liu, D; Krambis, M; Liu, Y; McGaraughty, S; Chu, K; Roeloffs, R; Zhong, C; Mikusa, JP; Hernandez, G; Gauvin, D; Wade, C; Zhu, C; Pai, M; Scanio, M; Shi, L; Drizin, I; Gregg, R; Matulenko, M; Hakeem, A; Gross, M; Johnson, M; Marsh, K; Wagoner, PK; Sullivan, JP; Faltynek, CR; Krafte, DS Proc Natl Acad Sci U S A 104: 8520-5 (2007)
- Kumaran, D; Adler, M; Levit, M; Krebs, M; Sweeney, R; Swaminathan, S Bioorg Med Chem 23: 7264-73 (2015)
- Pedreira, JGB; Nahidino, P; Kudolo, M; Pantsar, T; Berger, BT; Forster, M; Knapp, S; Laufer, S; Barreiro, EJ J Med Chem 63: 7347-7354 (2020)
- Winter-Holt, JJ; Bardelle, C; Chiarparin, E; Dale, IL; Davey, PRJ; Davies, NL; Denz, C; Fillery, SM; Guérot, CM; Han, F; Hughes, SJ; Kulkarni, M; Liu, Z; Milbradt, A; Moss, TA; Niu, H; Patel, J; Rabow, AA; Schimpl, M; Shi, J; Sun, D; Yang, D; Guichard, S J Med Chem 65: 3306-3331 (2022)
- Tomic, M; Kundakovic, M; Butorovic, B; Janac, B; Andric, D; Roglic, G; Ignjatovic, D; Kostic-Rajacic, S Bioorg Med Chem Lett 14: 4263-6 (2004)
- Burns, CJ; Harte, MF; Bu, X; Fantino, E; Giarrusso, M; Joffe, M; Kurek, M; Legge, FS; Razzino, P; Su, S; Treutlein, H; Wan, SS; Zeng, J; Wilks, AF Bioorg Med Chem Lett 19: 1206-9 (2009)
- Misawa, T; Yorioka, M; Demizu, Y; Noguchi-Yachide, T; Ohoka, N; Kurashima-Kinoshita, M; Motoyoshi, H; Nojiri, H; Kittaka, A; Makishima, M; Naito, M; Kurihara, M Bioorg Med Chem Lett 25: 5362-6 (2015)
- Shimazawa, R; Kuriyama, M; Shirai, R Bioorg Med Chem Lett 18: 3350-3 (2008)
- Yamamoto, S; Kurono, M; Yoshida, A; Hotta, S US Patent US11052091 (2021)
- Syrjänen, L; Kuuslahti, M; Tolvanen, M; Vullo, D; Parkkila, S; Supuran, CT Bioorg Med Chem 23: 2303-9 (2015)
- Borsari, C; Jiménez-Antón, MD; Eick, J; Bifeld, E; Torrado, JJ; Olías-Molero, AI; Corral, MJ; Santarem, N; Baptista, C; Severi, L; Gul, S; Wolf, M; Kuzikov, M; Ellinger, B; Reinshagen, J; Witt, G; Linciano, P; Tait, A; Costantino, L; Luciani, R; Tejera Nevado, P; Zander-Dinse, D; Franco, CH; Ferrari, S; Moraes, CB; Cordeiro-da-Silva, A; Ponterini, G; Clos, J; Alunda, JM; Costi, MP Eur J Med Chem 183: (2019)
- Köse, M; Ritter, K; Thiemke, K; Gillard, M; Kostenis, E; Müller, CE ACS Med Chem Lett 5: 326-30 (2014)
- Fox, BM; Sugimoto, K; Iio, K; Yoshida, A; Zhang, JK; Li, K; Hao, X; Labelle, M; Smith, ML; Rubenstein, SM; Ye, G; McMinn, D; Jackson, S; Choi, R; Shan, B; Ma, J; Miao, S; Matsui, T; Ogawa, N; Suzuki, M; Kobayashi, A; Ozeki, H; Okuma, C; Ishii, Y; Tomimoto, D; Furakawa, N; Tanaka, M; Matsushita, M; Takahashi, M; Inaba, T; Sagawa, S; Kayser, F J Med Chem 57: 3464-83 (2014)
- Parthasarathy, S; Henry, K; Pei, H; Clayton, J; Rempala, M; Johns, D; De Frutos, O; Garcia, P; Mateos, C; Pleite, S; Wang, Y; Stout, S; Condon, B; Ashok, S; Lu, Z; Ehlhardt, W; Raub, T; Lai, M; Geeganage, S; Burkholder, TP Bioorg Med Chem Lett 28: 1887-1891 (2018)
- Lamothe, M; Perrin, D; Blotières, D; Leborgne, M; Gras, S; Bonnet, D; Hill, BT; Halazy, S Bioorg Med Chem Lett 6: 1291-1296 (1996)
- Lu, Q; Chen, Z; Perumattam, J; Wang, DX; Liang, W; Xu, YJ; Do, S; Bonaga, L; Higaki, J; Dong, H; Liclican, A; Sideris, S; Laney, M; Dugar, S; Mavunkel, B; Levy, DE Bioorg Med Chem Lett 18: 2399-403 (2008)
- Cappelli, A; Manini, M; Valenti, S; Castriconi, F; Giuliani, G; Anzini, M; Brogi, S; Butini, S; Gemma, S; Campiani, G; Giorgi, G; Mennuni, L; Lanza, M; Giordani, A; Caselli, G; Letari, O; Makovec, F Eur J Med Chem 63: 85-94 (2013)
- Sweis, RF; Hunt, JA; Sinclair, PJ; Chen, Y; Eveland, SS; Guo, Q; Hyland, SA; Milot, DP; Cumiskey, AM; Latham, M; Rosa, R; Peterson, L; Sparrow, CP; Anderson, MS Bioorg Med Chem Lett 21: 2597-600 (2011)
- Pascard, C; Guilhem, J; Vincent, M; Rémond, G; Portevin, B; Laubie, M J Med Chem 34: 663-9 (1991)
- Furber, M; Alcaraz, L; Bent, JE; Beyerbach, A; Bowers, K; Braddock, M; Caffrey, MV; Cladingboel, D; Collington, J; Donald, DK; Fagura, M; Ince, F; Kinchin, EC; Laurent, C; Lawson, M; Luker, TJ; Mortimore, MM; Pimm, AD; Riley, RJ; Roberts, N; Robertson, M; Theaker, J; Thorne, PV; Weaver, R; Webborn, P; Willis, P J Med Chem 50: 5882-5 (2007)
- Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334-9 (2014)
- Shiryaev, SA; Remacle, AG; Ratnikov, BI; Nelson, NA; Savinov, AY; Wei, G; Bottini, M; Rega, MF; Parent, A; Desjardins, R; Fugere, M; Day, R; Sabet, M; Pellecchia, M; Liddington, RC; Smith, JW; Mustelin, T; Guiney, DG; Lebl, M; Strongin, AY J Biol Chem 282: 20847-53 (2007)
- Beveridge, RE; Wallweber, HA; Ashkenazi, A; Beresini, M; Clark, KR; Gibbons, P; Ghiro, E; Kaufman, S; Larivée, A; Leblanc, M; Leclerc, JP; Lemire, A; Ly, C; Rudolph, J; Schwarz, JB; Srivastava, S; Wang, W; Zhao, L; Braun, MG ACS Med Chem Lett 11: 2389-2396 (2020)
- Lamothe, M; Perrin, D; Blotières, D; Leborgne, M; Gras, S; Bonnet, D; Hill, BT; Halazy, S Bioorg Med Chem Lett 6: 1291-1296 (1996)
- Daniels, MH; Malojcic, G; Clugston, SL; Williams, B; Coeffet-Le Gal, M; Pan-Zhou, XR; Venkatachalan, S; Harmange, JC; Ledeboer, M J Med Chem 65: 3575-3596 (2022)
- Lefrançois, M; Lefebvre, MR; Saint-Onge, G; Boulais, PE; Lamothe, S; Leduc, R; Lavigne, P; Heveker, N; Escher, E ACS Med Chem Lett 2: 597-602 (2011)
- Lehr, M; Klimt, M; Elfringhoff, AS Bioorg Med Chem Lett 11: 2569-72 (2001)
- Li, M; Konteatis, Z; Nagaraja, N; Chen, Y; Zhou, S; Ma, G; Gross, S; Marjon, K; Hyer, ML; Mandley, E; Lein, M; Padyana, AK; Jin, L; Tong, S; Peters, R; Murtie, J; Travins, J; Medeiros, M; Liu, P; Frank, V; Judd, ET; Biller, SA; Marks, KM; Sui, Z; Reznik, SK J Med Chem 65: 4600-4615 (2022)
- Lacivita, E; De Giorgio, P; Lee, IT; Rodeheaver, SI; Weiss, BA; Fracasso, C; Caccia, S; Berardi, F; Perrone, R; Zhang, MR; Maeda, J; Higuchi, M; Suhara, T; Schetz, JA; Leopoldo, M J Med Chem 53: 7344-55 (2010)
- Liégeois, JF; Lespagnard, M; Meneses Salas, E; Mangin, F; Scuvée-Moreau, J; Dilly, S ACS Med Chem Lett 5: 358-62 (2014)
- Gajewski, TF; Spranger, S; Leung, M US Patent US10967060 (2021)
- Benaim, G; Sanders, JM; Garcia-Marchán, Y; Colina, C; Lira, R; Caldera, AR; Payares, G; Sanoja, C; Burgos, JM; Leon-Rossell, A; Concepcion, JL; Schijman, AG; Levin, M; Oldfield, E; Urbina, JA J Med Chem 49: 892-9 (2006)
- Kumaran, D; Adler, M; Levit, M; Krebs, M; Sweeney, R; Swaminathan, S Bioorg Med Chem 23: 7264-73 (2015)
- Lansdell, MI; Hepworth, D; Calabrese, A; Brown, AD; Blagg, J; Burring, DJ; Wilson, P; Fradet, D; Brown, TB; Quinton, F; Mistry, N; Tang, K; Mount, N; Stacey, P; Edmunds, N; Adams, C; Gaboardi, S; Neal-Morgan, S; Wayman, C; Cole, S; Phipps, J; Lewis, M; Verrier, H; Gillon, V; Feeder, N; Heatherington, A; Sultana, S; Haughie, S; Martin, SW; Sudworth, M; Tweedy, S J Med Chem 53: 3183-97 (2010)
- Huang, B; Wang, H; Zheng, Y; Li, M; Kang, G; Barreto-de-Souza, V; Nassehi, N; Knapp, PE; Selley, DE; Hauser, KF; Zhang, Y J Med Chem 64: 7702-7723 (2021)
- Huryn, DM; Wipf, P; LaPorte, MG; Colombo, R; Kovaliov, M; Lim, C; Alverez, CN; Yue, Z; Samankumara, LP; Chatterley, AJ; Yan, Y; Liang, M; Green, NJ; Baldwin, ET; Moore, WJ; Arkin, M; Neitz, RJ; Ang, K; Bryant, C; Bulfer, S US Patent US11247985 (2022)
- Liao M
- Kozlova, A; Thabault, L; Dauguet, N; Deskeuvre, M; Stroobant, V; Pilotte, L; Liberelle, M; Van den Eynde, B; Frédérick, R Eur J Med Chem 227: (2022)
- Burger, MT; Han, W; Lan, J; Nishiguchi, G; Bellamacina, C; Lindval, M; Atallah, G; Ding, Y; Mathur, M; McBride, C; Beans, EL; Muller, K; Tamez, V; Zhang, Y; Huh, K; Feucht, P; Zavorotinskaya, T; Dai, Y; Holash, J; Castillo, J; Langowski, J; Wang, Y; Chen, MY; Garcia, PD ACS Med Chem Lett 4: 1193-7 (2013)
- Lingel, A; Sendzik, M; Huang, Y; Shultz, MD; Cantwell, J; Dillon, MP; Fu, X; Fuller, J; Gabriel, T; Gu, J; Jiang, X; Li, L; Liang, F; McKenna, M; Qi, W; Rao, W; Sheng, X; Shu, W; Sutton, J; Taft, B; Wang, L; Zeng, J; Zhang, H; Zhang, M; Zhao, K; Lindvall, M; Bussiere, DE J Med Chem 60: 415-427 (2017)
- Wang, A; Lv, K; Tao, Z; Gu, J; Fu, L; Liu, M; Wan, B; Franzblau, SG; Ma, C; Ma, X; Han, B; Wang, A; Xu, S; Lu, Y Eur J Med Chem 181: (2019)
- Lizarzaburu, M; Turcotte, S; Du, X; Duquette, J; Fu, A; Houze, J; Li, L; Liu, J; Murakoshi, M; Oda, K; Okuyama, R; Nara, F; Reagan, J; Yu, M; Medina, JC Bioorg Med Chem Lett 22: 5942-7 (2012)
- Camps, P; Formosa, X; Galdeano, C; Gómez, T; Muñoz-Torrero, D; Scarpellini, M; Viayna, E; Badia, A; Clos, MV; Camins, A; Pallàs, M; Bartolini, M; Mancini, F; Andrisano, V; Estelrich, J; Lizondo, M; Bidon-Chanal, A; Luque, FJ J Med Chem 51: 3588-98 (2008)
- Collin, M; Brohm, D; Héroult, M; Lobell, M; Hübsch, W; Lustig, K; Grünewald, S; Bömer, U; Vöhringer, V; Lindner, N US Patent US9598416 (2017)
- Zhu, A; Zhan, W; Liang, Z; Yoon, Y; Yang, H; Grossniklaus, HE; Xu, J; Rojas, M; Lockwood, M; Snyder, JP; Liotta, DC; Shim, H J Med Chem 53: 8556-68 (2010)
- Zhou, C; Garcia-Calvo, M; Pinto, S; Lombardo, M; Feng, Z; Bender, K; Pryor, KD; Bhatt, UR; Chabin, RM; Geissler, WM; Shen, Z; Tong, X; Zhang, Z; Wong, KK; Roy, RS; Chapman, KT; Yang, L; Xiong, Y J Med Chem 53: 7251-63 (2010)
- Singer, M; Lopez, M; Bornaghi, LF; Innocenti, A; Vullo, D; Supuran, CT; Poulsen, SA Bioorg Med Chem Lett 19: 2273-6 (2009)
- Huang, A; Moretto, A; Janz, K; Lowe, M; Bedard, PW; Tam, S; Di, L; Clerin, V; Sushkova, N; Tchernychev, B; Tsao, DH; Keith, JC; Shaw, GD; Schaub, RG; Wang, Q; Kaila, N J Med Chem 53: 6003-17 (2010)
- Tian, C; Yang, C; Wu, T; Lu, M; Chen, Y; Yang, Y; Liu, X; Ling, Y; Deng, M; Jia, Y; Zhou, Y Bioorg Med Chem Lett 48: (2021)
- Butler, KV; Ma, A; Yu, W; Li, F; Tempel, W; Babault, N; Pittella-Silva, F; Shao, J; Wang, J; Luo, M; Vedadi, M; Brown, PJ; Arrowsmith, CH; Jin, J J Med Chem 59: 9881-9889 (2016)
- Stahlecker, J; Klett, T; Schwer, M; Jaag, S; Dammann, M; Ernst, LN; Braun, MB; Zimmermann, MO; Kramer, M; Lämmerhofer, M; Stehle, T; Coles, M; Boeckler, FM RSC Med Chem 13: 1575-1586 (2022)
- A., AK; Irina, CM; M., HD; C., KJ; Jian, L; J., MP; L., RV; T., RM; A., SC; Zhe, W; Dong, X WIPO WO2022094012 (2022)
- J., BM; E., FM; Marie, LH; J., MJ; J., RA; M., SK; J., SS WIPO WO2022115301 (2022)
- Mjalli, AM; Chapman, KT; MacCoss, M Bioorg Med Chem Lett 3: 2693-2698 (1993)
- van der Stelt, M; van Kuik, JA; Bari, M; van Zadelhoff, G; Leeflang, BR; Veldink, GA; Finazzi-Agrò, A; Vliegenthart, JF; Maccarrone, M J Med Chem 45: 3709-20 (2002)
- Sasaki, S; Ehara, T; Alam, MR; Fujino, Y; Harada, N; Kimura, J; Nakamura, H; Maeda, M Bioorg Med Chem Lett 11: 2581-4 (2001)
- Carballa, DM; Seoane, S; Zacconi, F; Pérez, X; Rumbo, A; Alvarez-Díaz, S; Larriba, MJ; Pérez-Fernández, R; Muñoz, A; Maestro, M; Mouriño, A; Torneiro, M J Med Chem 55: 8642-56 (2012)
- Di Fabio, R; Micheli, F; Alvaro, G; Cavanni, P; Donati, D; Gagliardi, T; Fontana, G; Giovannini, R; Maffeis, M; Mingardi, A; Tranquillini, ME; Vitulli, G Bioorg Med Chem Lett 17: 2254-9 (2007)
- Manetti, F; Brullo, C; Magnani, M; Mosci, F; Chelli, B; Crespan, E; Schenone, S; Naldini, A; Bruno, O; Trincavelli, ML; Maga, G; Carraro, F; Martini, C; Bondavalli, F; Botta, M J Med Chem 51: 1252-9 (2008)
- Kotani, H; Tanabe, H; Mizukami, H; Makishima, M; Inoue, M J Nat Prod 73: 1332-6 (2010)
- Reilly, SW; Puentes, LN; Wilson, K; Hsieh, CJ; Weng, CC; Makvandi, M; Mach, RH J Med Chem 61: 5367-5379 (2018)
- Castillo, M; Forns, P; Erra, M; Mir, M; López, M; Maldonado, M; Orellana, A; Carreño, C; Ramis, I; Miralpeix, M; Vidal, B Bioorg Med Chem Lett 22: 5419-23 (2012)
- Rovnyak, GC; Kimball, SD; Beyer, B; Cucinotta, G; DiMarco, JD; Gougoutas, J; Hedberg, A; Malley, M; McCarthy, JP; Zhang, R J Med Chem 38: 119-29 (1995)
- Seifert, T; Malo, M; Lengqvist, J; Sihlbom, C; Jarho, EM; Luthman, K J Med Chem 59: 10794-10799 (2016)
- Cappelli, A; Manini, M; Paolino, M; Gallelli, A; Anzini, M; Mennuni, L; Del Cadia, M; De Rienzo, F; Menziani, MC; Vomero, S ACS Med Chem Lett 2: 571-576 (2011)
- Manning, M; Cheng, LL; Klis, WA; Balaspiri, L; Olma, A; Sawyer, WH; Wo, NC; Chan, WY J Med Chem 38: 1762-9 (1995)
- Manzoni, L; Gornati, D; Manzotti, M; Cairati, S; Bossi, A; Arosio, D; Lecis, D; Seneci, P Bioorg Med Chem Lett 26: 4613-4619 (2016)
- Ahn, JS; Radhakrishnan, ML; Mapelli, M; Choi, S; Tidor, B; Cuny, GD; Musacchio, A; Yeh, LA; Kosik, KS Chem Biol 12: 811-23 (2005)
- Coteron, JM; Marco, M; Esquivias, J; Deng, X; White, KL; White, J; Koltun, M; El Mazouni, F; Kokkonda, S; Katneni, K; Bhamidipati, R; Shackleford, DM; Angulo-Barturen, I; Ferrer, SB; Jiménez-Díaz, MB; Gamo, FJ; Goldsmith, EJ; Charman, WN; Bathurst, I; Floyd, D; Matthews, D; Burrows, JN; Rathod, PK; Charman, SA; Phillips, MA J Med Chem 54: 5540-61 (2011)
- Amori, L; Serpi, M; Marinozzi, M; Costantino, G; Diaz, MG; Hermit, MB; Thomsen, C; Pellicciari, R Bioorg Med Chem Lett 16: 196-9 (2005)
- Palanki, MS; Dneprovskaia, E; Doukas, J; Fine, RM; Hood, J; Kang, X; Lohse, D; Martin, M; Noronha, G; Soll, RM; Wrasidlo, W; Yee, S; Zhu, H J Med Chem 50: 4279-94 (2007)
- Blake, JF; Burkard, M; Chan, J; Chen, H; Chou, KJ; Diaz, D; Dudley, DA; Gaudino, JJ; Gould, SE; Grina, J; Hunsaker, T; Liu, L; Martinson, M; Moreno, D; Mueller, L; Orr, C; Pacheco, P; Qin, A; Rasor, K; Ren, L; Robarge, K; Shahidi-Latham, S; Stults, J; Sullivan, F; Wang, W; Yin, J; Zhou, A; Belvin, M; Merchant, M; Moffat, J; Schwarz, JB J Med Chem 59: 5650-60 (2016)
- Tormählen, NM; Martorelli, M; Kuhn, A; Maier, F; Guezguez, J; Burnet, M; Albrecht, W; Laufer, SA; Koch, P J Med Chem 65: 1225-1242 (2022)
- Shimizu, K; Maruyama, M; Yasui, Y; Minegishi, H; Ban, HS; Nakamura, H Bioorg Med Chem Lett 20: 1453-6 (2010)
- Lavecchia, A; Di Giovanni, C; Pesapane, A; Montuori, N; Ragno, P; Martucci, NM; Masullo, M; De Vendittis, E; Novellino, E J Med Chem 55: 4142-58 (2012)
- Burger, MT; Han, W; Lan, J; Nishiguchi, G; Bellamacina, C; Lindval, M; Atallah, G; Ding, Y; Mathur, M; McBride, C; Beans, EL; Muller, K; Tamez, V; Zhang, Y; Huh, K; Feucht, P; Zavorotinskaya, T; Dai, Y; Holash, J; Castillo, J; Langowski, J; Wang, Y; Chen, MY; Garcia, PD ACS Med Chem Lett 4: 1193-7 (2013)
- Mejdrová, I; Chalupská, D; Placková, P; Müller, C; ?ála, M; Klíma, M; Baumlová, A; Hrebabecký, H; Procházková, E; Dejmek, M; Strunin, D; Weber, J; Lee, G; Matou?ová, M; Mertlíková-Kaiserová, H; Ziebuhr, J; Birkus, G; Boura, E; Nencka, R J Med Chem 60: 100-118 (2017)
- Tamamura, H; Omagari, A; Hiramatsu, K; Gotoh, K; Kanamoto, T; Xu, Y; Kodama, E; Matsuoka, M; Hattori, T; Yamamoto, N; Nakashima, H; Otaka, A; Fujii, N Bioorg Med Chem Lett 11: 1897-902 (2001)
- Ebiike, H; Taka, N; Matsushita, M; Ohmori, M; Takami, K; Hyohdoh, I; Kohchi, M; Hayase, T; Nishii, H; Morikami, K; Nakanishi, Y; Akiyama, N; Shindoh, H; Ishii, N; Isobe, T; Matsuoka, H J Med Chem 59: 10586-10600 (2016)
- Marino, JP; Fisher, PW; Hofmann, GA; Kirkpatrick, RB; Janson, CA; Johnson, RK; Ma, C; Mattern, M; Meek, TD; Ryan, MD; Schulz, C; Smith, WW; Tew, DG; Tomazek, TA; Veber, DF; Xiong, WC; Yamamoto, Y; Yamashita, K; Yang, G; Thompson, SK J Med Chem 50: 3777-85 (2007)
- Jarvis, MF; Honore, P; Shieh, CC; Chapman, M; Joshi, S; Zhang, XF; Kort, M; Carroll, W; Marron, B; Atkinson, R; Thomas, J; Liu, D; Krambis, M; Liu, Y; McGaraughty, S; Chu, K; Roeloffs, R; Zhong, C; Mikusa, JP; Hernandez, G; Gauvin, D; Wade, C; Zhu, C; Pai, M; Scanio, M; Shi, L; Drizin, I; Gregg, R; Matulenko, M; Hakeem, A; Gross, M; Johnson, M; Marsh, K; Wagoner, PK; Sullivan, JP; Faltynek, CR; Krafte, DS Proc Natl Acad Sci U S A 104: 8520-5 (2007)
- Kumar, S; Waldo, J; Jaipuri, F; Mautino, M US Patent US9981973 (2018)
- Qiu, W; Zhou, M; Mazumdar, M; Azzi, A; Ghanmi, D; Luu-The, V; Labrie, F; Lin, SX J Biol Chem 282: 8368-79 (2007)
- Garigipati, RS; Seibel, G; Mayer, RJ; Bolognese, B; McCord, M; Marshall, LA; Adams, JL Bioorg Med Chem Lett 7: 1421-1426 (1997)
- Lingel, A; Sendzik, M; Huang, Y; Shultz, MD; Cantwell, J; Dillon, MP; Fu, X; Fuller, J; Gabriel, T; Gu, J; Jiang, X; Li, L; Liang, F; McKenna, M; Qi, W; Rao, W; Sheng, X; Shu, W; Sutton, J; Taft, B; Wang, L; Zeng, J; Zhang, H; Zhang, M; Zhao, K; Lindvall, M; Bussiere, DE J Med Chem 60: 415-427 (2017)
- Li, M; Konteatis, Z; Nagaraja, N; Chen, Y; Zhou, S; Ma, G; Gross, S; Marjon, K; Hyer, ML; Mandley, E; Lein, M; Padyana, AK; Jin, L; Tong, S; Peters, R; Murtie, J; Travins, J; Medeiros, M; Liu, P; Frank, V; Judd, ET; Biller, SA; Marks, KM; Sui, Z; Reznik, SK J Med Chem 65: 4600-4615 (2022)
- Jia, ZJ; Venkataramani, C; Huang, W; Mehrotra, M; Song, Y; Xu, Q; Bauer, SM; Rose, JW; Kane, B; Pandey, A US Patent US9579320 (2017)
- Vanotti, E; Caldarelli, M; Cirla, A; Forte, B; Ermoli, A; Menichincheri, M; Pillan, A; Scolaro, A US Patent US9670191 (2017)
- Blake, JF; Burkard, M; Chan, J; Chen, H; Chou, KJ; Diaz, D; Dudley, DA; Gaudino, JJ; Gould, SE; Grina, J; Hunsaker, T; Liu, L; Martinson, M; Moreno, D; Mueller, L; Orr, C; Pacheco, P; Qin, A; Rasor, K; Ren, L; Robarge, K; Shahidi-Latham, S; Stults, J; Sullivan, F; Wang, W; Yin, J; Zhou, A; Belvin, M; Merchant, M; Moffat, J; Schwarz, JB J Med Chem 59: 5650-60 (2016)
- Okolotowicz, KJ; Dwyer, M; Ryan, D; Cheng, J; Cashman, EA; Moore, S; Mercola, M; Cashman, JR Bioorg Med Chem 26: 4441-4451 (2018)
- Cutshall, NS; Gage, JL; Gruswitz, FA; Khalaf, J; Little, TL; Metz, M; Nguyen, JH; Nollert von Specht, PK; Tsoung, J; Cicirelli, M; Goldstein, SR; Keshipeddy, SK; Kwon, DY; Lemus, RH; Vaddela, SB US Patent US11584714 (2023)
- Kontopidis, G; McInnes, C; Pandalaneni, SR; McNae, I; Gibson, D; Mezna, M; Thomas, M; Wood, G; Wang, S; Walkinshaw, MD; Fischer, PM Chem Biol 13: 201-11 (2006)
- Brauers, G; Edrada, RA; Ebel, R; Proksch, P; Wray, V; Berg, A; Gräfe, U; Schächtele, C; Totzke, F; Finkenzeller, G; Marme, D; Kraus, J; Münchbach, M; Michel, M; Bringmann, G; Schaumann, K J Nat Prod 63: 739-45 (2000)
- Michels, M; Briem, H; Vakalopoulos, A; Zimmermann, K; Teusch, N US Patent US8604028 (2013)
- Chen, HY; Plummer, CW; Xiao, D; Chobanian, HR; DeMong, D; Miller, M; Trujillo, ME; Kirkland, M; Kosinski, D; Mane, J; Pachanski, M; Cheewatrakoolpong, B; Di Salvo, J; Thomas-Fowlkes, B; Souza, S; Tatosian, DA; Chen, Q; Hafey, MJ; Houle, R; Nolting, AF; Orr, R; Ehrhart, J; Weinglass, AB; Tschirret-Guth, R; Howard, AD; Colletti, SL ACS Med Chem Lett 9: 685-690 (2018)
- Ma, B; Metrick, CM; Gu, C; Hoemberger, M; Bajrami, B; Bame, E; Huang, J; Mingueneau, M; Murugan, P; Santoro, JC; Tang, H; Wang, T; Hopkins, BT Bioorg Med Chem Lett 60: (2022)
- Castillo, M; Forns, P; Erra, M; Mir, M; López, M; Maldonado, M; Orellana, A; Carreño, C; Ramis, I; Miralpeix, M; Vidal, B Bioorg Med Chem Lett 22: 5419-23 (2012)
- Fardis, M; Jin, H; Jabri, S; Cai, RZ; Mish, M; Tsiang, M; Kim, CU Bioorg Med Chem Lett 16: 4031-5 (2006)
- Fushimi, M; Fujimori, I; Wakabayashi, T; Hasui, T; Kawakita, Y; Imamura, K; Kato, T; Murakami, M; Ishii, T; Kikko, Y; Kasahara, M; Nakatani, A; Hiura, Y; Miyamoto, M; Saikatendu, K; Zou, H; Lane, SW; Lawson, JD; Imoto, H J Med Chem 62: 4915-4935 (2019)
- Kashima, Y; Miyazawa, M Bioorg Med Chem Lett 23: 6580-4 (2013)
- Zhang, X; Rueter, JK; Chen, Y; Moorjani, M; Lanier, MC; Lin, E; Gross, RS; Tellew, JE; Williams, JP; Lechner, SM; Markison, S; Joswig, T; Malany, S; Santos, M; Castro-Palomino, JC; Crespo, MI; Prat, M; Gual, S; Díaz, JL; Saunders, J; Slee, DH Bioorg Med Chem Lett 18: 1778-83 (2008)
- Castelli, R; Taranto, S; Furiassi, L; Bozza, N; Marseglia, G; Ferlenghi, F; Rivara, S; Retini, M; Bedini, A; Spadoni, G; Matarazzo, S; Ronca, R; Presta, M; Mor, M; Giacomini, A Eur J Med Chem 221: (2021)
- Carr&aagrovr;, G; Rizzi, A; Guerrini, R; Barnes, TA; McDonald, J; Hebbes, CP; Mela, F; Kenigs, VA; Marzola, G; Rizzi, D; Gavioli, E; Zucchini, S; Regoli, D; Morari, M; Salvadori, S; Rowbotham, DJ; Lambert, DG; Kapusta, DR; Calo', G J Pharmacol Exp Ther 312: 1114-23 (2005)
- Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334-9 (2014)
- Fallacara, AL; Passannanti, R; Mori, M; Iovenitti, G; Musumeci, F; Greco, C; Crespan, E; Kissova, M; Maga, G; Tarantelli, C; Spriano, F; Gaudio, E; Bertoni, F; Botta, M; Schenone, S Eur J Med Chem 181: (2019)
- Cirillo, PF; Hickey, ER; Moss, N; Breitfelder, S; Betageri, R; Fadra, T; Gaenzler, F; Gilmore, T; Goldberg, DR; Kamhi, V; Kirrane, T; Kroe, RR; Madwed, J; Moriak, M; Netherton, M; Pargellis, CA; Patel, UR; Qian, KC; Sharma, R; Sun, S; Swinamer, A; Torcellini, C; Takahashi, H; Tsang, M; Xiong, Z Bioorg Med Chem Lett 19: 2386-91 (2009)
- Desjardins, M; Desgagnes, J; Lacoste, L; Yang, F; Morin, M; Lapointe, J; Chenevert, R Bioorg Med Chem Lett 7: 2363-2366 (1997)
- Inoue, T; Morita, M; Tojo, T; Nagashima, A; Moritomo, A; Miyake, H Bioorg Med Chem 21: 3873-81 (2013)
- Ito, M; Sakamoto, T; Suzuki, T; Egashira, S; Moriya, M; Ishihara, A; Iwaasa, H; Matsushita, H; Nakase, K; Wallace, MA; Dean, D; Sato, N; Tokita, S; Kanatani, A Bioorg Med Chem Lett 19: 2835-9 (2009)
- Johnson, DS; Stiff, C; Lazerwith, SE; Kesten, SR; Fay, LK; Morris, M; Beidler, D; Liimatta, MB; Smith, SE; Dudley, DT; Sadagopan, N; Bhattachar, SN; Kesten, SJ; Nomanbhoy, TK; Cravatt, BF; Ahn, K ACS Med Chem Lett 2: 91-96 (2011)
- Cee, VJ; Albrecht, BK; Geuns-Meyer, S; Hughes, P; Bellon, S; Bready, J; Caenepeel, S; Chaffee, SC; Coxon, A; Emery, M; Fretland, J; Gallant, P; Gu, Y; Hodous, BL; Hoffman, D; Johnson, RE; Kendall, R; Kim, JL; Long, AM; McGowan, D; Morrison, M; Olivieri, PR; Patel, VF; Polverino, A; Powers, D; Rose, P; Wang, L; Zhao, H J Med Chem 50: 627-40 (2007)
- Ali, SM; Ashwell, MA; Kelleher, E; Koerner, S; Lapierre, J; Link, JS; Liu, Y; Moussa, M; Palma, R; Tandon, M; Vensel, D; Westlund, N; Wu, H; Yang, R US Patent US8541407 (2013)
- Wu, S; Vossius, S; Rahmouni, S; Miletic, AV; Vang, T; Vazquez-Rodriguez, J; Cerignoli, F; Arimura, Y; Williams, S; Hayes, T; Moutschen, M; Vasile, S; Pellecchia, M; Mustelin, T; Tautz, L J Med Chem 52: 6716-23 (2009)
- Meegalla, SK; Plössl, K; Kung, MP; Stevenson, DA; Mu, M; Kushner, S; Liable-Sands, LM; Rheingold, AL; Kung, HF J Med Chem 41: 428-36 (1998)
- D'Agostino, LA; Sjin, RT; Niu, D; McDonald, JJ; Zhu, Z; Liu, H; Mazdiyasni, H; Petter, RC; Singh, J; Barrague, M; Gross, A; Munson, M US Patent US9695132 (2017)
- Ito, M; Tanaka, T; Toita, A; Uchiyama, N; Kokubo, H; Morishita, N; Klein, MG; Zou, H; Murakami, M; Kondo, M; Sameshima, T; Araki, S; Endo, S; Kawamoto, T; Morin, GB; Aparicio, SA; Nakanishi, A; Maezaki, H; Imaeda, Y J Med Chem 61: 7710-7728 (2018)
- Toda, N; Hao, X; Ogawa, Y; Oda, K; Yu, M; Fu, Z; Chen, Y; Kim, Y; Lizarzaburu, M; Lively, S; Lawlis, S; Murakoshi, M; Nara, F; Watanabe, N; Reagan, JD; Tian, H; Fu, A; Motani, A; Liu, Q; Lin, YJ; Zhuang, R; Xiong, Y; Fan, P; Medina, J; Li, L; Izumi, M; Okuyama, R; Shibuya, S ACS Med Chem Lett 4: 790-4 (2013)
- Ban, H; Muraoka, M; Ioriya, K; Ohashi, N Bioorg Med Chem Lett 16: 44-8 (2005)
- Misawa, T; Yorioka, M; Demizu, Y; Noguchi-Yachide, T; Ohoka, N; Kurashima-Kinoshita, M; Motoyoshi, H; Nojiri, H; Kittaka, A; Makishima, M; Naito, M; Kurihara, M Bioorg Med Chem Lett 25: 5362-6 (2015)
- Yoshimoto, N; Sakamaki, Y; Haeta, M; Kato, A; Inaba, Y; Itoh, T; Nakabayashi, M; Ito, N; Yamamoto, K J Med Chem 55: 4373-81 (2012)
- Aoyama, Y; Uenaka, M; Konoike, T; Hayasaki-Kajiwara, Y; Naya, N; Nakajima, M Bioorg Med Chem Lett 11: 1691-4 (2001)
- Yoshikawa, M; Saitoh, M; Katoh, T; Seki, T; Bigi, SV; Shimizu, Y; Ishii, T; Okai, T; Kuno, M; Hattori, H; Watanabe, E; Saikatendu, KS; Zou, H; Nakakariya, M; Tatamiya, T; Nakada, Y; Yogo, T J Med Chem 61: 2384-2409 (2018)
- Altenbach, RJ; Khilevich, A; Meyer, MD; Buckner, SA; Milicic, I; Daza, AV; Brune, ME; O'Neill, AB; Gauvin, DM; Cain, JC; Nakane, M; Holladay, MW; Williams, M; Brioni, JD; Sullivan, JP J Med Chem 45: 4395-7 (2002)
- Koike, T; Takai, T; Hoashi, Y; Nakayama, M; Kosugi, Y; Nakashima, M; Yoshikubo, S; Hirai, K; Uchikawa, O J Med Chem 54: 4207-18 (2011)
- Ono, M; Yoshida, N; Ishibashi, K; Haratake, M; Arano, Y; Mori, H; Nakayama, M J Med Chem 48: 7253-60 (2005)
- Nakazono, M; Hasegawa, S; Yamamoto, T; Zaitsu, K Bioorg Med Chem Lett 14: 5619-21 (2004)
- Morera, E; Di Marzo, V; Monti, L; Allarŕ, M; Schiano Moriello, A; Nalli, M; Ortar, G; De Petrocellis, L Bioorg Med Chem Lett 26: 1401-5 (2016)
- Maarisit, W; Yamazaki, H; Kanno, SI; Tomizawa, A; Rotinsulu, H; Wewengkang, DS; Sumilat, DA; Ukai, K; Kapojos, MM; Namikoshi, M Bioorg Med Chem Lett 27: 999-1002 (2017)
- Bressi, JC; Jennings, AJ; Skene, R; Wu, Y; Melkus, R; De Jong, R; O'Connell, S; Grimshaw, CE; Navre, M; Gangloff, AR Bioorg Med Chem Lett 20: 3142-5 (2010)
- Fernández-Bachiller, MI; Hwang, S; Schembri, ME; Lindemann, P; Guberman, M; Herziger, S; Specker, E; Matter, H; Will, DW; Czech, J; Wagner, M; Bauer, A; Schreuder, H; Ritter, K; Urmann, M; Wehner, V; Sun, H; Nazaré, M J Med Chem 65: 13013-13028 (2022)
- Verdugo, DE; Cancilla, MT; Ge, X; Gray, NS; Chang, YT; Schultz, PG; Negishi, M; Leary, JA; Bertozzi, CR J Med Chem 44: 2683-6 (2001)
- Micheli, F; Cavanni, P; Andreotti, D; Arban, R; Benedetti, R; Bertani, B; Bettati, M; Bettelini, L; Bonanomi, G; Braggio, S; Carletti, R; Checchia, A; Corsi, M; Fazzolari, E; Fontana, S; Marchioro, C; Merlo-Pich, E; Negri, M; Oliosi, B; Ratti, E; Read, KD; Roscic, M; Sartori, I; Spada, S; Tedesco, G; Tarsi, L; Terreni, S; Visentini, F; Zocchi, A; Zonzini, L; Di Fabio, R J Med Chem 53: 4989-5001 (2010)
- Brasca, MG; Gnocchi, P; Nesi, M; Amboldi, N; Avanzi, N; Bertrand, J; Bindi, S; Canevari, G; Casero, D; Ciomei, M; Colombo, N; Cribioli, S; Fachin, G; Felder, ER; Galvani, A; Isacchi, A; Motto, I; Panzeri, A; Donati, D Bioorg Med Chem 23: 2387-407 (2015)
- Cirillo, PF; Hickey, ER; Moss, N; Breitfelder, S; Betageri, R; Fadra, T; Gaenzler, F; Gilmore, T; Goldberg, DR; Kamhi, V; Kirrane, T; Kroe, RR; Madwed, J; Moriak, M; Netherton, M; Pargellis, CA; Patel, UR; Qian, KC; Sharma, R; Sun, S; Swinamer, A; Torcellini, C; Takahashi, H; Tsang, M; Xiong, Z Bioorg Med Chem Lett 19: 2386-91 (2009)
- Guba, W; Nettekoven, M; Püllmann, B; Riemer, C; Schmitt, S Bioorg Med Chem Lett 14: 3307-12 (2004)
- Hopkins, BT; Ma, B; Prince, R; Marx, I; Schulz, J; Nevalainen, M; Dechantsreiter, M US Patent US10899753 (2021)
- Taguchi, M; Sugimoto, K; Goda, K; Akama, T; Yamamoto, K; Suzuki, T; Tomishima, Y; Nishiguchi, M; Arai, K; Takahashi, K; Kobori, T Bioorg Med Chem Lett 13: 1963-6 (2003)
- Le Manach, C; Paquet, T; Brunschwig, C; Njoroge, M; Han, Z; Gonzŕlez Cabrera, D; Bashyam, S; Dhinakaran, R; Taylor, D; Reader, J; Botha, M; Churchyard, A; Lauterbach, S; Coetzer, TL; Birkholtz, LM; Meister, S; Winzeler, EA; Waterson, D; Witty, MJ; Wittlin, S; Jiménez-Díaz, MB; Santos Martínez, M; Ferrer, S; Angulo-Barturen, I; Street, LJ; Chibale, K J Med Chem 58: 8713-22 (2015)
- Kotoku, M; Maeba, T; Fujioka, S; Yokota, M; Seki, N; Ito, K; Suwa, Y; Ikenogami, T; Hirata, K; Hase, Y; Katsuda, Y; Miyagawa, N; Arita, K; Asahina, K; Noguchi, M; Nomura, A; Doi, S; Adachi, T; Crowe, P; Tao, H; Thacher, S; Hashimoto, H; Suzuki, T; Shiozaki, M J Med Chem 62: 2837-2842 (2019)
- Heightman, TD; Berdini, V; Braithwaite, H; Buck, IM; Cassidy, M; Castro, J; Courtin, A; Day, JEH; East, C; Fazal, L; Graham, B; Griffiths-Jones, CM; Lyons, JF; Martins, V; Muench, S; Munck, JM; Norton, D; O'Reilly, M; Palmer, N; Pathuri, P; Reader, M; Rees, DC; Rich, SJ; Richardson, C; Saini, H; Thompson, NT; Wallis, NG; Walton, H; Wilsher, NE; Woolford, AJ; Cooke, M; Cousin, D; Onions, S; Shannon, J; Watts, J; Murray, CW J Med Chem 61: 4978-4992 (2018)
- Kiyama, R; Honma, T; Hayashi, K; Ogawa, M; Hara, M; Fujimoto, M; Fujishita, T J Med Chem 38: 2728-41 (1995)
- Oh, M; Im, I; Lee, YJ; Kim, YH; Yoon, JH; Park, HG; Higashiyama, S; Kim, YC; Park, WJ Bioorg Med Chem Lett 14: 6071-4 (2004)
- Ohashi, M; Oyama, T; Nakagome, I; Satoh, M; Nishio, Y; Nobusada, H; Hirono, S; Morikawa, K; Hashimoto, Y; Miyachi, H J Med Chem 54: 331-41 (2011)
- Ishida, J; Yamamoto, H; Kido, Y; Kamijo, K; Murano, K; Miyake, H; Ohkubo, M; Kinoshita, T; Warizaya, M; Iwashita, A; Mihara, K; Matsuoka, N; Hattori, K Bioorg Med Chem 14: 1378-90 (2006)
- Ebiike, H; Taka, N; Matsushita, M; Ohmori, M; Takami, K; Hyohdoh, I; Kohchi, M; Hayase, T; Nishii, H; Morikami, K; Nakanishi, Y; Akiyama, N; Shindoh, H; Ishii, N; Isobe, T; Matsuoka, H J Med Chem 59: 10586-10600 (2016)
- Jacobson, KA; Ohno, M; Duong, HT; Kim, SK; Tchilibon, S; Cesnek, M; Holý, A; Gao, ZG Chem Biol 12: 237-47 (2005)
- Hayakawa, M; Kawaguchi, K; Kaizawa, H; Koizumi, T; Ohishi, T; Yamano, M; Okada, M; Ohta, M; Tsukamoto, S; Raynaud, FI; Parker, P; Workman, P; Waterfield, MD Bioorg Med Chem 15: 5837-44 (2007)
- Tsuri, T; Honma, T; Hiramatsu, Y; Okada, T; Hashizume, H; Mitsumori, S; Inagaki, M; Arimura, A; Yasui, K; Asanuma, F; Kishino, J; Ohtani, M J Med Chem 40: 3504-7 (1997)
- Ichikawa, M; Ohtsuka, M; Ohki, H; Haginoya, N; Itoh, M; Sugita, K; Usui, H; Suzuki, M; Terayama, K; Kanda, A Bioorg Med Chem 20: 3072-93 (2012)
- Hayakawa, M; Kaizawa, H; Kawaguchi, K; Ishikawa, N; Koizumi, T; Ohishi, T; Yamano, M; Okada, M; Ohta, M; Tsukamoto, S; Raynaud, FI; Waterfield, MD; Parker, P; Workman, P Bioorg Med Chem 15: 403-12 (2007)
- Okamoto, M; Takayama, K; Shimizu, T; Ishida, K; Takahashi, O; Furuya, T J Med Chem 52: 7323-7 (2009)
- Moreau, P; Anizon, F; Sancelme, M; Prudhomme, M; Bailly, C; Carrasco, C; Ollier, M; Sevčre, D; Riou, JF; Fabbro, D; Meyer, T; Aubertin, AM J Med Chem 41: 1631-40 (1998)
- Pierre, F; Chua, PC; O'Brien, SE; Siddiqui-Jain, A; Bourbon, P; Haddach, M; Michaux, J; Nagasawa, J; Schwaebe, MK; Stefan, E; Vialettes, A; Whitten, JP; Chen, TK; Darjania, L; Stansfield, R; Anderes, K; Bliesath, J; Drygin, D; Ho, C; Omori, M; Proffitt, C; Streiner, N; Trent, K; Rice, WG; Ryckman, DM J Med Chem 54: 635-54 (2011)
- Kubota, K; Kurebayashi, H; Miyachi, H; Tobe, M; Onishi, M; Isobe, Y Bioorg Med Chem Lett 19: 2766-71 (2009)
- Nagata, T; Inoue, M; Ashida, Y; Noguchi, K; Ono, M US Patent US8609710 (2013)
- Manetti, F; Santucci, A; Locatelli, GA; Maga, G; Spreafico, A; Serchi, T; Orlandini, M; Bernardini, G; Caradonna, NP; Spallarossa, A; Brullo, C; Schenone, S; Bruno, O; Ranise, A; Bondavalli, F; Hoffmann, O; Bologna, M; Angelucci, A; Botta, M J Med Chem 50: 5579-88 (2007)
- Tsou, HR; Otteng, M; Tran, T; Floyd, MB; Reich, M; Birnberg, G; Kutterer, K; Ayral-Kaloustian, S; Ravi, M; Nilakantan, R; Grillo, M; McGinnis, JP; Rabindran, SK J Med Chem 51: 3507-25 (2008)
- Gauthier, JY; Black, WC; Courchesne, I; Cromlish, W; Desmarais, S; Houle, R; Lamontagne, S; Li, CS; Massé, F; McKay, DJ; Ouellet, M; Robichaud, J; Truchon, JF; Truong, VL; Wang, Q; Percival, MD Bioorg Med Chem Lett 17: 4929-33 (2007)
- Sanchez-Martinez, C; Shih, C; Faul, MM; Zhu, G; Paal, M; Somoza, C; Li, T; Kumrich, CA; Winneroski, LL; Xun, Z; Brooks, HB; Patel, BK; Schultz, RM; DeHahn, TB; Spencer, CD; Watkins, SA; Considine, E; Dempsey, JA; Ogg, CA; Campbell, RM; Anderson, BA; Wagner, J Bioorg Med Chem Lett 13: 3835-9 (2003)
- Liessi, N; Cichero, E; Pesce, E; Arkel, M; Salis, A; Tomati, V; Paccagnella, M; Damonte, G; Tasso, B; Galietta, LJV; Pedemonte, N; Fossa, P; Millo, E Eur J Med Chem 144: 179-200 (2018)
- Jarvis, MF; Honore, P; Shieh, CC; Chapman, M; Joshi, S; Zhang, XF; Kort, M; Carroll, W; Marron, B; Atkinson, R; Thomas, J; Liu, D; Krambis, M; Liu, Y; McGaraughty, S; Chu, K; Roeloffs, R; Zhong, C; Mikusa, JP; Hernandez, G; Gauvin, D; Wade, C; Zhu, C; Pai, M; Scanio, M; Shi, L; Drizin, I; Gregg, R; Matulenko, M; Hakeem, A; Gross, M; Johnson, M; Marsh, K; Wagoner, PK; Sullivan, JP; Faltynek, CR; Krafte, DS Proc Natl Acad Sci U S A 104: 8520-5 (2007)
- Liu, Y; Richardson, J; Tran, T; Al-Muhtasib, N; Xie, T; Yenugonda, VM; Sexton, HG; Rezvani, AH; Levin, ED; Sahibzada, N; Kellar, KJ; Brown, ML; Xiao, Y; Paige, M J Med Chem 56: 3000-11 (2013)
- Li, YL; Shi, E; Burns, D; Li, Y; Covington, MB; Pan, M; Scherle, P; Friedman, S; Metcalf, B; Yao, W Bioorg Med Chem Lett 19: 5037-42 (2009)
- Razavi, H; Riether, D; Harcken, C; Bentzien, J; Dinallo, RM; Souza, D; Nelson, RM; Kukulka, A; Fadra-Khan, TN; Pack, EJ; Zuvela-Jelaska, L; Pelletier, J; Panzenbeck, M; Torcellini, CA; Proudfoot, JR; Nabozny, GH; Thomson, DS Bioorg Med Chem Lett 24: 1934-40 (2014)
- Cappelli, A; Manini, M; Paolino, M; Gallelli, A; Anzini, M; Mennuni, L; Del Cadia, M; De Rienzo, F; Menziani, MC; Vomero, S ACS Med Chem Lett 2: 571-576 (2011)
- Piemontese, L; Fracchiolla, G; Carrieri, A; Parente, M; Laghezza, A; Carbonara, G; Sblano, S; Tauro, M; Gilardi, F; Tortorella, P; Lavecchia, A; Crestani, M; Desvergne, B; Loiodice, F Eur J Med Chem 90: 583-94 (2015)
- Cui, JJ; McTigue, M; Nambu, M; Tran-Dubé, M; Pairish, M; Shen, H; Jia, L; Cheng, H; Hoffman, J; Le, P; Jalaie, M; Goetz, GH; Ryan, K; Grodsky, N; Deng, YL; Parker, M; Timofeevski, S; Murray, BW; Yamazaki, S; Aguirre, S; Li, Q; Zou, H; Christensen, J J Med Chem 55: 8091-109 (2012)
- Rossi, C; Porcelloni, M; D'Andrea, P; Fincham, CI; Ettorre, A; Mauro, S; Squarcia, A; Bigioni, M; Parlani, M; Nardelli, F; Binaschi, M; Maggi, CA; Fattori, D Bioorg Med Chem Lett 21: 2305-8 (2011)
- Kellenberger, E; Springael, JY; Parmentier, M; Hachet-Haas, M; Galzi, JL; Rognan, D J Med Chem 50: 1294-303 (2007)
- Vidadala, RS; Rivas, KL; Ojo, KK; Hulverson, MA; Zambriski, JA; Bruzual, I; Schultz, TL; Huang, W; Zhang, Z; Scheele, S; DeRocher, AE; Choi, R; Barrett, LK; Siddaramaiah, LK; Hol, WG; Fan, E; Merritt, EA; Parsons, M; Freiberg, G; Marsh, K; Kempf, DJ; Carruthers, VB; Isoherranen, N; Doggett, JS; Van Voorhis, WC; Maly, DJ J Med Chem 59: 6531-46 (2016)
- Chu, M; Mierzwa, R; He, L; King, A; Patel, M; Pichardo, J; Hart, A; Butkiewicz, N; Puar, MS Bioorg Med Chem Lett 9: 1949-52 (1999)
- Canale, V; Guzik, P; Kurczab, R; Verdie, P; Satala, G; Kubica, B; Pawlowski, M; Martinez, J; Subra, G; Bojarski, AJ; Zajdel, P Eur J Med Chem 78: 10-22 (2014)
- Cee, VJ; Schenkel, LB; Hodous, BL; Deak, HL; Nguyen, HN; Olivieri, PR; Romero, K; Bak, A; Be, X; Bellon, S; Bush, TL; Cheng, AC; Chung, G; Coats, S; Eden, PM; Hanestad, K; Gallant, PL; Gu, Y; Huang, X; Kendall, RL; Lin, MH; Morrison, MJ; Patel, VF; Radinsky, R; Rose, PE; Ross, S; Sun, JR; Tang, J; Zhao, H; Payton, M; Geuns-Meyer, SD J Med Chem 53: 6368-77 (2010)
- Shiryaev, SA; Remacle, AG; Ratnikov, BI; Nelson, NA; Savinov, AY; Wei, G; Bottini, M; Rega, MF; Parent, A; Desjardins, R; Fugere, M; Day, R; Sabet, M; Pellecchia, M; Liddington, RC; Smith, JW; Mustelin, T; Guiney, DG; Lebl, M; Strongin, AY J Biol Chem 282: 20847-53 (2007)
- Flohr, A; Hutter, R; Mueller, B; Bohnert, C; Pellisson, M; Schaffhauser, H Bioorg Med Chem Lett 27: 5415-5419 (2017)
- Jones, LH; Allan, G; Barba, O; Burt, C; Corbau, R; Dupont, T; Knöchel, T; Irving, S; Middleton, DS; Mowbray, CE; Perros, M; Ringrose, H; Swain, NA; Webster, R; Westby, M; Phillips, C J Med Chem 52: 1219-23 (2009)
- Helmboldt, A; Petitou, M; Mallet, J; Herault, J; Lormeau, J; Driguez, PA; Herbert, J; Sinay, P Bioorg Med Chem Lett 7: 1507-1510 (1997)
- Malosh, C; Turlington, M; Bridges, TM; Rook, JM; Noetzel, MJ; Vinson, PN; Steckler, T; Lavreysen, H; Mackie, C; Bartolomé-Nebreda, JM; Conde-Ceide, S; Martínez-Viturro, CM; Piedrafita, M; Sánchez-Casado, MR; Macdonald, GJ; Daniels, JS; Jones, CK; Niswender, CM; Conn, PJ; Lindsley, CW; Stauffer, SR Bioorg Med Chem Lett 25: 5115-20 (2015)
- Haile, PA; Votta, BJ; Marquis, RW; Bury, MJ; Mehlmann, JF; Singhaus, R; Charnley, AK; Lakdawala, AS; Convery, MA; Lipshutz, DB; Desai, BM; Swift, B; Capriotti, CA; Berger, SB; Mahajan, MK; Reilly, MA; Rivera, EJ; Sun, HH; Nagilla, R; Beal, AM; Finger, JN; Cook, MN; King, BW; Ouellette, MT; Totoritis, RD; Pierdomenico, M; Negroni, A; Stronati, L; Cucchiara, S; Ziólkowski, B; Vossenkämper, A; MacDonald, TT; Gough, PJ; Bertin, J; Casillas, LN J Med Chem 59: 4867-80 (2016)
- Angeli, A; Pinteala, M; Maier, SS; Toti, A; Di Cesare Mannelli, L; Ghelardini, C; Selleri, S; Carta, F; Supuran, CT Bioorg Med Chem Lett 45: (2021)
- Prezzavento, O; Campisi, A; Parenti, C; Ronsisvalle, S; Aricò, G; Arena, E; Pistolozzi, M; Scoto, GM; Bertucci, C; Vanella, A; Ronsisvalle, G J Med Chem 53: 5881-5 (2010)
- Proudfoot, JR; Betageri, R; Cardozo, M; Gilmore, TA; Glynn, S; Hickey, ER; Jakes, S; Kabcenell, A; Kirrane, TM; Tibolla, AK; Lukas, S; Patel, UR; Sharma, R; Yazdanian, M; Moss, N; Beaulieu, PL; Cameron, DR; Ferland, JM; Gauthier, J; Gillard, J; Gorys, V; Poirier, M; Rancourt, J; Wernic, D; Llinas-Brunet, M J Med Chem 44: 2421-31 (2001)
- Pace, P; Di Francesco, ME; Gardelli, C; Harper, S; Muraglia, E; Nizi, E; Orvieto, F; Petrocchi, A; Poma, M; Rowley, M; Scarpelli, R; Laufer, R; Gonzalez Paz, O; Monteagudo, E; Bonelli, F; Hazuda, D; Stillmock, KA; Summa, V J Med Chem 50: 2225-39 (2007)
- Gilbert, J; Fuentes, M; Ojasoo, T; Doré, JC; Pons, M J Med Chem 40: 1104-11 (1997)
- Rossi, C; Porcelloni, M; D'Andrea, P; Fincham, CI; Ettorre, A; Mauro, S; Squarcia, A; Bigioni, M; Parlani, M; Nardelli, F; Binaschi, M; Maggi, CA; Fattori, D Bioorg Med Chem Lett 21: 2305-8 (2011)
- Buchler, I; Akuma, D; Au, V; Carr, G; de León, P; DePasquale, M; Ernst, G; Huang, Y; Kimos, M; Kolobova, A; Poslusney, M; Wei, H; Swinnen, D; Montel, F; Moureau, F; Jigorel, E; Schulze, MED; Wood, M; Barrow, JC J Med Chem 61: 9647-9665 (2018)
- He, L; Seitz, SP; Trainor, GL; Tortolani, D; Vaccaro, W; Poss, M; Tarby, CM; Tokarski, JS; Penhallow, B; Hung, CY; Attar, R; Lin, TA Bioorg Med Chem Lett 22: 5995-8 (2012)
- Hansen, JD; Correa, M; Alexander, M; Nagy, M; Huang, D; Sapienza, J; Lu, G; LeBrun, LA; Cathers, BE; Zhang, W; Tang, Y; Ammirante, M; Narla, RK; Piccotti, JR; Pourdehnad, M; Lopez-Girona, A J Med Chem 64: 1835-1843 (2021)
- Moorjani, M; Zhang, X; Chen, Y; Lin, E; Rueter, JK; Gross, RS; Lanier, MC; Tellew, JE; Williams, JP; Lechner, SM; Malany, S; Santos, M; Ekhlassi, P; Castro-Palomino, JC; Crespo, MI; Prat, M; Gual, S; Díaz, JL; Saunders, J; Slee, DH Bioorg Med Chem Lett 18: 1269-73 (2008)
- Pearlstein, RA; Vaz, RJ; Kang, J; Chen, XL; Preobrazhenskaya, M; Shchekotikhin, AE; Korolev, AM; Lysenkova, LN; Miroshnikova, OV; Hendrix, J; Rampe, D Bioorg Med Chem Lett 13: 1829-35 (2003)
- Castelli, R; Taranto, S; Furiassi, L; Bozza, N; Marseglia, G; Ferlenghi, F; Rivara, S; Retini, M; Bedini, A; Spadoni, G; Matarazzo, S; Ronca, R; Presta, M; Mor, M; Giacomini, A Eur J Med Chem 221: (2021)
- Pretze, M; Pallavi, P; Roscher, M; Klotz, S; Caballero, J; Binzen, U; Greffrath, W; Treede, RD; Harmsen, MC; Hafner, M; Yard, B; Wängler, C; Wängler, B J Med Chem 59: 9855-9865 (2016)
- Whittaker, M; Thompson, TM; Spavold, ZM; Price, M; Miller, A; Galloway, W; Fraser, F; Floyd, CD; Drummond, AH; Davidson, AH; Bowles, SA; Bebbington, DS Bioorg Med Chem Lett 3: 1493-1498 (1993)
- Hill, D; Horwell, D; Hunter, J; Kneen, C; Pritchard, M; Suman-Chauhan, N Bioorg Med Chem Lett 3: 885-888 (1993)
- Tummalapalli, SR; Bhat, R; Chojnowski, A; Prorok, M; Kreiss, T; Goldberg, R; Canan, S; Hawryluk, N; Mortensen, D; Khetani, V; Zeldis, J; Siekierka, JJ; Rotella, DP ACS Med Chem Lett 9: 210-214 (2018)
- Reddy, TJ; Chan, L; Turcotte, N; Proulx, M; Pereira, OZ; Das, SK; Siddiqui, A; Wang, W; Poisson, C; Yannopoulos, CG; Bilimoria, D; L'Heureux, L; Alaoui, HM; Nguyen-Ba, N Bioorg Med Chem Lett 13: 3341-4 (2003)
- Moreau, P; Anizon, F; Sancelme, M; Prudhomme, M; Bailly, C; Carrasco, C; Ollier, M; Sevčre, D; Riou, JF; Fabbro, D; Meyer, T; Aubertin, AM J Med Chem 41: 1631-40 (1998)
- Chen, XT; Ghavimi, B; Corbett, RL; Xue, CB; Liu, RQ; Covington, MB; Qian, M; Vaddi, KG; Christ, DD; Hartman, KD; Ribadeneira, MD; Trzaskos, JM; Newton, RC; Decicco, CP; Duan, JJ Bioorg Med Chem Lett 17: 1865-70 (2007)
- Li, Y; Ye, T; Xu, L; Dong, Y; Luo, Y; Wang, C; Han, Y; Chen, K; Qin, M; Liu, Y; Zhao, Y Eur J Med Chem 181: (2019)
- Quibell, M; Watts, JP; Flinn, NS US Patent US8552202 (2013)
- Piticchio, SG; Martínez-Cartró, M; Scaffidi, S; Rachman, M; Rodriguez-Arevalo, S; Sanchez-Arfelis, A; Escolano, C; Picaud, S; Krojer, T; Filippakopoulos, P; von Delft, F; Galdeano, C; Barril, X J Med Chem 64: 17887-17900 (2021)
- Crespan, E; Radi, M; Zanoli, S; Schenone, S; Botta, M; Maga, G Bioorg Med Chem 18: 3999-4008 (2010)
- Rockwell, AL; Rafalski, M; Pitts, WJ; Batt, DG; Petraitis, JJ; DeGrado, WF; Mousa, S; Jadhav, PK Bioorg Med Chem Lett 9: 937-42 (1999)
- Belayet, JB; Beamish, S; Rahaman, M; Alanani, S; Virdi, RS; Frick, DN; Rahman, AFMT; Ulicki, JS; Biswas, S; Arnold, LA; Roni, MSR; Cheng, EY; Steeber, DA; Frick, KM; Hossain, MM J Med Chem 65: 3388-3403 (2022)
- Korhonen, LE; Rahnasto, M; Mähönen, NJ; Wittekindt, C; Poso, A; Juvonen, RO; Raunio, H J Med Chem 48: 3808-15 (2005)
- Rueda, DC; Schöffmann, A; De Mieri, M; Raith, M; Jähne, EA; Hering, S; Hamburger, M Bioorg Med Chem 22: 1276-84 (2014)
- Rajabi, M; Mansell, D; Freeman, S; Bryce, RA Eur J Med Chem 46: 1165-71 (2011)
- Marsault, E; Hoveyda, HR; Peterson, ML; Saint-Louis, C; Landry, A; Vézina, M; Ouellet, L; Wang, Z; Ramaseshan, M; Beaubien, S; Benakli, K; Beauchemin, S; Déziel, R; Peeters, T; Fraser, GL J Med Chem 49: 7190-7 (2006)
- Long, DD; Armstrong, SR; Beattie, DT; Campbell, CB; Church, TJ; Colson, PJ; Dalziel, SM; Jacobsen, JR; Jiang, L; Obedencio, GP; Rapta, M; Saito, D; Stergiades, I; Tsuruda, PR; Van Dyke, PM; Vickery, RG ACS Med Chem Lett 10: 1641-1647 (2019)
- Tsou, HR; Otteng, M; Tran, T; Floyd, MB; Reich, M; Birnberg, G; Kutterer, K; Ayral-Kaloustian, S; Ravi, M; Nilakantan, R; Grillo, M; McGinnis, JP; Rabindran, SK J Med Chem 51: 3507-25 (2008)
- Heightman, TD; Berdini, V; Braithwaite, H; Buck, IM; Cassidy, M; Castro, J; Courtin, A; Day, JEH; East, C; Fazal, L; Graham, B; Griffiths-Jones, CM; Lyons, JF; Martins, V; Muench, S; Munck, JM; Norton, D; O'Reilly, M; Palmer, N; Pathuri, P; Reader, M; Rees, DC; Rich, SJ; Richardson, C; Saini, H; Thompson, NT; Wallis, NG; Walton, H; Wilsher, NE; Woolford, AJ; Cooke, M; Cousin, D; Onions, S; Shannon, J; Watts, J; Murray, CW J Med Chem 61: 4978-4992 (2018)
- Tsou, HR; Otteng, M; Tran, T; Floyd, MB; Reich, M; Birnberg, G; Kutterer, K; Ayral-Kaloustian, S; Ravi, M; Nilakantan, R; Grillo, M; McGinnis, JP; Rabindran, SK J Med Chem 51: 3507-25 (2008)
- Shen, L; Zhang, Y; Wang, A; Sieber-McMaster, E; Chen, X; Pelton, P; Xu, JZ; Yang, M; Zhu, P; Zhou, L; Reuman, M; Hu, Z; Russell, R; Gibbs, AC; Ross, H; Demarest, K; Murray, WV; Kuo, GH Bioorg Med Chem 16: 3321-41 (2008)
- Tosstorff, A; Rudolph, MG; Cole, JC; Reutlinger, M; Kramer, C; Schaffhauser, H; Nilly, A; Flohr, A; Kuhn, B J Comput Aided Mol Des 36: 753-765 (2022)
- Bharathan, IT; Blackburn, C; Ciavarri, JP; Chouitar, J; Cullis, CA; D Amore, N; Fleming, PE; Gigstad, KM; Gipson, KE; Girard, M; Hu, Y; Lee, J; Li, G; Rezaei, M; Sintchak, MD; Soucy, F; Stroud, SG; Vos, TJ; Xu, H; Ye, Y US Patent US10202373 (2019)
- Taha, M; Ismail, NH; Imran, S; Wadood, A; Rahim, F; Riaz, M Bioorg Med Chem 23: 7211-8 (2015)
- Fantini, M; Rivara, M; Zuliani, V; Kalmar, CL; Vacondio, F; Silva, C; Baheti, AR; Singh, N; Merrick, EC; Katari, RS; Cocconcelli, G; Ghiron, C; Patel, MK Bioorg Med Chem 17: 3642-8 (2009)
- Keith, JM; Apodaca, R; Tichenor, M; Xiao, W; Jones, W; Pierce, J; Seierstad, M; Palmer, J; Webb, M; Karbarz, M; Scott, B; Wilson, S; Luo, L; Wennerholm, M; Chang, L; Brown, S; Rizzolio, M; Rynberg, R; Chaplan, S; Breitenbucher, JG ACS Med Chem Lett 3: 823-827 (2012)
- Kozikowski, AP; Simoni, D; Roberti, M; Rondanin, R; Wang, S; Du, P; Johnson, KM Bioorg Med Chem Lett 9: 1831-6 (1999)
- Baxter, A; Bent, J; Bowers, K; Braddock, M; Brough, S; Fagura, M; Lawson, M; McInally, T; Mortimore, M; Robertson, M; Weaver, R; Webborn, P Bioorg Med Chem Lett 13: 4047-50 (2003)
- Zhu, A; Zhan, W; Liang, Z; Yoon, Y; Yang, H; Grossniklaus, HE; Xu, J; Rojas, M; Lockwood, M; Snyder, JP; Liotta, DC; Shim, H J Med Chem 53: 8556-68 (2010)
- Pretze, M; Pallavi, P; Roscher, M; Klotz, S; Caballero, J; Binzen, U; Greffrath, W; Treede, RD; Harmsen, MC; Hafner, M; Yard, B; Wängler, C; Wängler, B J Med Chem 59: 9855-9865 (2016)
- Micheli, F; Cavanni, P; Andreotti, D; Arban, R; Benedetti, R; Bertani, B; Bettati, M; Bettelini, L; Bonanomi, G; Braggio, S; Carletti, R; Checchia, A; Corsi, M; Fazzolari, E; Fontana, S; Marchioro, C; Merlo-Pich, E; Negri, M; Oliosi, B; Ratti, E; Read, KD; Roscic, M; Sartori, I; Spada, S; Tedesco, G; Tarsi, L; Terreni, S; Visentini, F; Zocchi, A; Zonzini, L; Di Fabio, R J Med Chem 53: 4989-5001 (2010)
- Hale, JJ; Neway, W; Mills, SG; Hajdu, R; Ann Keohane, C; Rosenbach, M; Milligan, J; Shei, GJ; Chrebet, G; Bergstrom, J; Card, D; Koo, GC; Koprak, SL; Jackson, JJ; Rosen, H; Mandala, S Bioorg Med Chem Lett 14: 3351-5 (2004)
- Wu, T; Nagle, A; Kuhen, K; Gagaring, K; Borboa, R; Francek, C; Chen, Z; Plouffe, D; Goh, A; Lakshminarayana, SB; Wu, J; Ang, HQ; Zeng, P; Kang, ML; Tan, W; Tan, M; Ye, N; Lin, X; Caldwell, C; Ek, J; Skolnik, S; Liu, F; Wang, J; Chang, J; Li, C; Hollenbeck, T; Tuntland, T; Isbell, J; Fischli, C; Brun, R; Rottmann, M; Dartois, V; Keller, T; Diagana, T; Winzeler, E; Glynne, R; Tully, DC; Chatterjee, AK J Med Chem 54: 5116-30 (2011)
- Beneker, CM; Rovoli, M; Kontopidis, G; Röring, M; Galda, S; Braun, S; Brummer, T; McInnes, C J Med Chem 62: 3886-3897 (2019)
- Scarpelli, R; Di Marco, A; Ferrigno, F; Laufer, R; Marcucci, I; Muraglia, E; Ontoria, JM; Rowley, M; Serafini, S; Steinkühler, C; Jones, P Bioorg Med Chem Lett 18: 6078-82 (2008)
- Guerlet, G; Spangenberg, T; Mann, A; Faure, H; Ruat, M Bioorg Med Chem Lett 21: 3608-12 (2011)
- Liu, J; He, S; Jian, T; Dobbelaar, PH; Sebhat, IK; Lin, LS; Goodman, A; Guo, C; Guzzo, PR; Hadden, M; Henderson, AJ; Pattamana, K; Ruenz, M; Sargent, BJ; Swenson, B; Yet, L; Tamvakopoulos, C; Peng, Q; Pan, J; Kan, Y; Palyha, O; Kelly, TM; Guan, XM; Howard, AD; Marsh, DJ; Metzger, JM; Reitman, ML; Wyvratt, MJ; Nargund, RP Bioorg Med Chem Lett 20: 2074-7 (2010)
- Chiellini, G; Nesi, G; Sestito, S; Chiarugi, S; Runfola, M; Espinoza, S; Sabatini, M; Bellusci, L; Laurino, A; Cichero, E; Gainetdinov, RR; Fossa, P; Raimondi, L; Zucchi, R; Rapposelli, S J Med Chem 59: 9825-9836 (2016)
- Parodi, A; Righetti, G; Pesce, E; Salis, A; Tasso, B; Urbinati, C; Tomati, V; Damonte, G; Rusnati, M; Pedemonte, N; Cichero, E; Millo, E Eur J Med Chem 208: (2020)
- Beneker, CM; Rovoli, M; Kontopidis, G; Röring, M; Galda, S; Braun, S; Brummer, T; McInnes, C J Med Chem 62: 3886-3897 (2019)
- Kong, Y; Grembecka, J; Edler, MC; Hamel, E; Mooberry, SL; Sabat, M; Rieger, J; Brown, ML Chem Biol 12: 1007-14 (2005)
- Chiellini, G; Nesi, G; Sestito, S; Chiarugi, S; Runfola, M; Espinoza, S; Sabatini, M; Bellusci, L; Laurino, A; Cichero, E; Gainetdinov, RR; Fossa, P; Raimondi, L; Zucchi, R; Rapposelli, S J Med Chem 59: 9825-9836 (2016)
- Shiryaev, SA; Remacle, AG; Ratnikov, BI; Nelson, NA; Savinov, AY; Wei, G; Bottini, M; Rega, MF; Parent, A; Desjardins, R; Fugere, M; Day, R; Sabet, M; Pellecchia, M; Liddington, RC; Smith, JW; Mustelin, T; Guiney, DG; Lebl, M; Strongin, AY J Biol Chem 282: 20847-53 (2007)
- Peukert, S; Sun, Y; Zhang, R; Hurley, B; Sabio, M; Shen, X; Gray, C; Dzink-Fox, J; Tao, J; Cebula, R; Wattanasin, S Bioorg Med Chem Lett 18: 1840-4 (2008)
- Sadeghzadeh, M; Sheibani, S; Ghandi, M; Daha, FJ; Amanlou, M; Arjmand, M; Hasani Bozcheloie, A Eur J Med Chem 64: 488-97 (2013)
- Yoshikawa, M; Saitoh, M; Kato, T; Nakayama, Y; Seki, T; Nakagawa, Y; Tominari, Y; Seto, M; Sasaki, Y; Okaniwa, M; Oda, T; Shibuya, A; Hidaka, K; Shiokawa, Z; Murata, S; Okabe, A; Nakada, Y; Mochizuki, M; Freeze, BS; Tawaraishi, T; Wada, Y; Greenspan, PD US Patent US11666594 (2023)
- Aoki, T; Hyohdoh, I; Furuichi, N; Ozawa, S; Watanabe, F; Matsushita, M; Sakaitani, M; Morikami, K; Takanashi, K; Harada, N; Tomii, Y; Shiraki, K; Furumoto, K; Tabo, M; Yoshinari, K; Ori, K; Aoki, Y; Shimma, N; Iikura, H ACS Med Chem Lett 5: 309-14 (2014)
- Braun, F; Bertoletti, N; Möller, G; Adamski, J; Steinmetzer, T; Salah, M; Abdelsamie, AS; van Koppen, CJ; Heine, A; Klebe, G; Marchais-Oberwinkler, S J Med Chem 59: 10719-10737 (2016)
- Filipuzzi, I; Thomas, JR; Pries, V; Estoppey, D; Salcius, M; Studer, C; Schirle, M; Hoepfner, D ACS Chem Biol 12: 2264-2269 (2017)
- Garner, AL; Gloeckner, C; Tricoche, N; Zakhari, JS; Samje, M; Cho-Ngwa, F; Lustigman, S; Janda, KD J Med Chem 54: 3963-72 (2011)
- Moreau, P; Anizon, F; Sancelme, M; Prudhomme, M; Bailly, C; Carrasco, C; Ollier, M; Sevčre, D; Riou, JF; Fabbro, D; Meyer, T; Aubertin, AM J Med Chem 41: 1631-40 (1998)
- Manca, I; Mastinu, A; Olimpieri, F; Falzoi, M; Sani, M; Ruiu, S; Loriga, G; Volonterio, A; Tambaro, S; Bottazzi, ME; Zanda, M; Pinna, GA; Lazzari, P Eur J Med Chem 62: 256-69 (2013)
- Moorjani, M; Zhang, X; Chen, Y; Lin, E; Rueter, JK; Gross, RS; Lanier, MC; Tellew, JE; Williams, JP; Lechner, SM; Malany, S; Santos, M; Ekhlassi, P; Castro-Palomino, JC; Crespo, MI; Prat, M; Gual, S; Díaz, JL; Saunders, J; Slee, DH Bioorg Med Chem Lett 18: 1269-73 (2008)
- Saquib, M; Ansari, MI; Johnson, CR; Khatoon, S; Kamil Hussain, M; Coop, A Eur J Med Chem 182: (2019)
- Skerlj, R; Bridger, G; Zhou, Y; Bourque, E; McEachern, E; Langille, J; Harwig, C; Veale, D; Yang, W; Li, T; Zhu, Y; Bey, M; Baird, I; Sartori, M; Metz, M; Mosi, R; Nelson, K; Bodart, V; Wong, R; Fricker, S; Mac Farland, R; Huskens, D; Schols, D Bioorg Med Chem Lett 21: 6950-4 (2011)
- Harada, K; Mizukami, J; Watanabe, T; Mori, G; Ubukata, M; Suwa, K; Fukuda, S; Negoro, T; Sato, M; Inaba, T Bioorg Med Chem Lett 29: 2100-2106 (2019)
- Ohashi, M; Oyama, T; Nakagome, I; Satoh, M; Nishio, Y; Nobusada, H; Hirono, S; Morikawa, K; Hashimoto, Y; Miyachi, H J Med Chem 54: 331-41 (2011)
- Asami, T; Kawahata, W; Sawa, M Bioorg Med Chem Lett 25: 2033-6 (2015)
- Jarvis, MF; Honore, P; Shieh, CC; Chapman, M; Joshi, S; Zhang, XF; Kort, M; Carroll, W; Marron, B; Atkinson, R; Thomas, J; Liu, D; Krambis, M; Liu, Y; McGaraughty, S; Chu, K; Roeloffs, R; Zhong, C; Mikusa, JP; Hernandez, G; Gauvin, D; Wade, C; Zhu, C; Pai, M; Scanio, M; Shi, L; Drizin, I; Gregg, R; Matulenko, M; Hakeem, A; Gross, M; Johnson, M; Marsh, K; Wagoner, PK; Sullivan, JP; Faltynek, CR; Krafte, DS Proc Natl Acad Sci U S A 104: 8520-5 (2007)
- Shen, Y; Li, F; Szewczyk, MM; Halabelian, L; Chau, I; Eram, MS; Dela Seńa, C; Park, KS; Meng, F; Chen, H; Zeng, H; Dong, A; Wu, H; Trush, VV; McLeod, D; Zepeda-Velázquez, CA; Campbell, RM; Mader, MM; Watson, BM; Schapira, M; Arrowsmith, CH; Al-Awar, R; Barsyte-Lovejoy, D; Kaniskan, HÜ; Brown, PJ; Vedadi, M; Jin, J J Med Chem 64: 3697-3706 (2021)
- Klein, T; Abgottspon, D; Wittwer, M; Rabbani, S; Herold, J; Jiang, X; Kleeb, S; Lüthi, C; Scharenberg, M; Bezençon, J; Gubler, E; Pang, L; Smiesko, M; Cutting, B; Schwardt, O; Ernst, B J Med Chem 53: 8627-41 (2010)
- Sundén, H; Schäfer, A; Scheepstra, M; Leysen, S; Malo, M; Ma, JN; Burstein, ES; Ottmann, C; Brunsveld, L; Olsson, R J Med Chem 59: 1232-8 (2016)
- Vucicevic, J; Srdic-Rajic, T; Pieroni, M; Laurila, JM; Perovic, V; Tassini, S; Azzali, E; Costantino, G; Glisic, S; Agbaba, D; Scheinin, M; Nikolic, K; Radi, M; Veljkovic, N Bioorg Med Chem 24: 3174-83 (2016)
- Bolli, MH; Abele, S; Binkert, C; Bravo, R; Buchmann, S; Bur, D; Gatfield, J; Hess, P; Kohl, C; Mangold, C; Mathys, B; Menyhart, K; Müller, C; Nayler, O; Scherz, M; Schmidt, G; Sippel, V; Steiner, B; Strasser, D; Treiber, A; Weller, T J Med Chem 53: 4198-211 (2010)
- Winter-Holt, JJ; Bardelle, C; Chiarparin, E; Dale, IL; Davey, PRJ; Davies, NL; Denz, C; Fillery, SM; Guérot, CM; Han, F; Hughes, SJ; Kulkarni, M; Liu, Z; Milbradt, A; Moss, TA; Niu, H; Patel, J; Rabow, AA; Schimpl, M; Shi, J; Sun, D; Yang, D; Guichard, S J Med Chem 65: 3306-3331 (2022)
- Filipuzzi, I; Thomas, JR; Pries, V; Estoppey, D; Salcius, M; Studer, C; Schirle, M; Hoepfner, D ACS Chem Biol 12: 2264-2269 (2017)
- von Rauch, M; Schlenk, M; Gust, R J Med Chem 47: 915-27 (2004)
- Quillet, R; Schneider, S; Utard, V; Drieu la Rochelle, A; Elhabazi, K; Henningsen, JB; Gizzi, P; Schmitt, M; Kugler, V; Simonneaux, V; Ilien, B; Simonin, F; Bihel, F J Med Chem 64: 7555-7564 (2021)
- Swahn, BM; Sandell, J; Pyring, D; Bergh, M; Jeppsson, F; Juréus, A; Neelissen, J; Johnström, P; Schou, M; Svensson, S Bioorg Med Chem Lett 22: 4332-7 (2012)
- Chaikuad, A; Diharce, J; Schröder, M; Foucourt, A; Leblond, B; Casagrande, AS; Désiré, L; Bonnet, P; Knapp, S; Besson, T J Med Chem 59: 10315-10321 (2016)
- Schuster, M; Blechert, S Bioorg Med Chem Lett 11: 1809-11 (2001)
- Sechi, M; Innocenti, A; Pala, N; Rogolino, D; Carcelli, M; Scozzafava, A; Supuran, CT Bioorg Med Chem Lett 22: 5801-6 (2012)
- Michaelis, S; Marais, A; Schrey, AK; Graebner, OY; Schaudt, C; Sefkow, M; Kroll, F; Dreger, M; Glinski, M; Koester, H; Metternich, R; Fischer, JJ J Med Chem 55: 3934-44 (2012)
- Apodaca, R; Breitenbucher, JG; Pattabiraman, K; Seierstad, M; Xiao, W US Patent US9169224 (2015)
- Kuntz, KW; Campbell, JE; Seki, M US Patent US10098888 (2018)
- Hosoguchi, K; Maeda, T; Furukawa, J; Shinohara, Y; Hinou, H; Sekiguchi, M; Togame, H; Takemoto, H; Kondo, H; Nishimura, S J Med Chem 53: 5607-19 (2010)
- Taha, M; Ismail, NH; Imran, S; Selvaraj, M; Rahim, A; Ali, M; Siddiqui, S; Rahim, F; Khan, KM Bioorg Med Chem 23: 7394-404 (2015)
- Fidan, I; Salmas, RE; Arslan, M; Sentürk, M; Durdagi, S; Ekinci, D; Sentürk, E; Cosgun, S; Supuran, CT Bioorg Med Chem 23: 7353-8 (2015)
- Jovanovi?, M; Zhukovsky, D; Podolski-Reni?, A; Domra?eva, I; ?alubovskis, R; Sen?anski, M; Gli?i?, S; Sharoyko, V; Tennikova, T; Dar'in, D; Pe?i?, M; Krasavin, M Eur J Med Chem 181: (2019)
- Amori, L; Serpi, M; Marinozzi, M; Costantino, G; Diaz, MG; Hermit, MB; Thomsen, C; Pellicciari, R Bioorg Med Chem Lett 16: 196-9 (2005)
- Yoshikawa, M; Saitoh, M; Kato, T; Nakayama, Y; Seki, T; Nakagawa, Y; Tominari, Y; Seto, M; Sasaki, Y; Okaniwa, M; Oda, T; Shibuya, A; Hidaka, K; Shiokawa, Z; Murata, S; Okabe, A; Nakada, Y; Mochizuki, M; Freeze, BS; Tawaraishi, T; Wada, Y; Greenspan, PD US Patent US11666594 (2023)
- Olivier, A; Sevrin, M; Durant, F; George, P Bioorg Med Chem Lett 7: 2277-2282 (1997)
- Saeed, A; Mahesar, PA; Zaib, S; Khan, MS; Matin, A; Shahid, M; Iqbal, J Eur J Med Chem 78: 43-53 (2014)
- O' Donovan, DH; Gregson, C; Packer, MJ; Greenwood, R; Pike, KG; Kawatkar, S; Bloecher, A; Robinson, J; Read, J; Code, E; Hsu, JH; Shen, M; Woods, H; Barton, P; Fillery, S; Williamson, B; Rawlins, PB; Bagal, SK Bioorg Med Chem Lett 39: (2021)
- Gopalsamy, A; Chopra, R; Lim, K; Ciszewski, G; Shi, M; Curran, KJ; Sukits, SF; Svenson, K; Bard, J; Ellingboe, JW; Agarwal, A; Krishnamurthy, G; Howe, AY; Orlowski, M; Feld, B; O'Connell, J; Mansour, TS J Med Chem 49: 3052-5 (2006)
- Kiyokawa, S; Hirata, Y; Nagaoka, Y; Shibano, M; Taniguchi, M; Yasuda, M; Baba, K; Uesato, S Bioorg Med Chem 18: 3925-33 (2010)
- Nam, SJ; Ko, H; Shin, M; Ham, J; Chin, J; Kim, Y; Kim, H; Shin, K; Choi, H; Kang, H Bioorg Med Chem Lett 16: 5398-402 (2006)
- Wu, MY; Esteban, G; Brogi, S; Shionoya, M; Wang, L; Campiani, G; Unzeta, M; Inokuchi, T; Butini, S; Marco-Contelles, J Eur J Med Chem 121: 864-879 (2016)
- Noji, S; Seki, N; Maeba, T; Sakai, T; Watanabe, E; Maeda, K; Fukushima, K; Noguchi, T; Ogawa, K; Toyonaga, Y; Negoro, T; Kawasaki, H; Shiozaki, M ACS Med Chem Lett 7: 919-923 (2016)
- Choi, K; Siegel, M; Piper, JL; Yuan, L; Cho, E; Strnad, P; Omary, B; Rich, KM; Khosla, C Chem Biol 12: 469-75 (2005)
- Allan, AC; Billinton, A; Brown, SH; Chowdhury, A; Eatherton, AJ; Fieldhouse, C; Giblin, GM; Goldsmith, P; Hall, A; Hurst, DN; Naylor, A; Rawlings, DA; Sime, M; Scoccitti, T; Theobald, PJ Bioorg Med Chem Lett 21: 4343-8 (2011)
- Singer, M; Lopez, M; Bornaghi, LF; Innocenti, A; Vullo, D; Supuran, CT; Poulsen, SA Bioorg Med Chem Lett 19: 2273-6 (2009)
- Zahid, H; Buchholz, CR; Singh, M; Ciccone, MF; Chan, A; Nithianantham, S; Shi, K; Aihara, H; Fischer, M; Schönbrunn, E; Dos Santos, CO; Landry, JW; Pomerantz, WCK J Med Chem 64: 13902-13917 (2021)
- Hu, LY; Ryder, TR; Rafferty, MF; Feng, MR; Lotarski, SM; Rock, DM; Sinz, M; Stoehr, SJ; Taylor, CP; Weber, ML; Bowersox, SS; Miljanich, GP; Millerman, E; Wang, YX; Szoke, BG J Med Chem 42: 4239-49 (1999)
- Weber, C; Sipos, M; Paczal, A; Balint, B; Kun, V; Foloppe, N; Dokurno, P; Massey, AJ; Walmsley, DL; Hubbard, RE; Murray, J; Benwell, K; Edmonds, T; Demarles, D; Bruno, A; Burbridge, M; Cruzalegui, F; Kotschy, A J Med Chem 64: 6745-6764 (2021)
- Juli, C; Sippel, M; Jäger, J; Thiele, A; Weiwad, M; Schweimer, K; Rösch, P; Steinert, M; Sotriffer, CA; Holzgrabe, U J Med Chem 54: 277-83 (2011)
- Skiles, JW; Miao, C; Sorcek, R; Jacober, S; Mui, PW; Chow, G; Weldon, SM; Possanza, G; Skoog, M; Keirns, J J Med Chem 35: 4795-808 (1993)
- Kees, KL; Musser, JH; Chang, J; Skowronek, M; Lewis, AJ J Med Chem 29: 2329-34 (1986)
- Castanedo, GM; Blaquiere, N; Beresini, M; Bravo, B; Brightbill, H; Chen, J; Cui, HF; Eigenbrot, C; Everett, C; Feng, J; Godemann, R; Gogol, E; Hymowitz, S; Johnson, A; Kayagaki, N; Kohli, PB; Knüppel, K; Kraemer, J; Krüger, S; Loke, P; McEwan, P; Montalbetti, C; Roberts, DA; Smith, M; Steinbacher, S; Sujatha-Bhaskar, S; Takahashi, R; Wang, X; Wu, LC; Zhang, Y; Staben, ST J Med Chem 60: 627-640 (2017)
- Witten, MR; Wissler, L; Snow, M; Geschwindner, S; Read, JA; Brandon, NJ; Nairn, AC; Lombroso, PJ; Käck, H; Ellman, JA J Med Chem 60: 9299-9319 (2017)
- El-Kabbani, O; Dhagat, U; Soda, M; Endo, S; Matsunaga, T; Hara, A Bioorg Med Chem Lett 21: 2564-7 (2011)
- Pinheiro, F; Pallarčs, I; Peccati, F; Sánchez-Morales, A; Varejăo, N; Bezerra, F; Ortega-Alarcon, D; Gonzalez, D; Osorio, M; Navarro, S; Velázquez-Campoy, A; Almeida, MR; Reverter, D; Busqué, F; Alibés, R; Sodupe, M; Ventura, S J Med Chem 65: 14673-14691 (2022)
- Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334-9 (2014)
- Andrés, JI; Alonso, JM; Díaz, A; Fernández, J; Iturrino, L; Martínez, P; Matesanz, E; Freyne, EJ; Deroose, F; Boeckx, G; Petit, D; Diels, G; Megens, A; Somers, M; Van Wauwe, J; Stoppie, P; Cools, M; De Clerck, F; Peeters, D; de Chaffoy, D Bioorg Med Chem Lett 12: 653-8 (2002)
- Sorge M
- Focken, T; Burford, K; Grimwood, ME; Zenova, A; Andrez, JC; Gong, W; Wilson, M; Taron, M; Decker, S; Lofstrand, V; Chowdhury, S; Shuart, N; Lin, S; Goodchild, SJ; Young, C; Soriano, M; Tari, PK; Waldbrook, M; Nelkenbrecher, K; Kwan, R; Lindgren, A; de Boer, G; Lee, S; Sojo, L; DeVita, RJ; Cohen, CJ; Wesolowski, SS; Johnson, JP; Dehnhardt, CM; Empfield, JR J Med Chem 62: 9618-9641 (2019)
- Haßfeld, J; Kinzel, T; Köbberling, J; Cancho-Grande, Y; Beyer, K; Röhrig, S; Köllnberger, M; Sperzel, M; Burkhardt, N; Schlemmer, K; Stegmann, C; Schuhmacher, J; Werner, M; Ellermann, M US Patent US10098883 (2018)
- Spyvee, M; Satoh, T; Carlson, JE US Patent US8686018 (2014)
- Raghavan, S; Yang, Z; Mosley, RT; Schleif, WA; Gabryelski, L; Olsen, DB; Stahlhut, M; Kuo, LC; Emini, EA; Chapman, KT; Tata, JR Bioorg Med Chem Lett 12: 2855-8 (2002)
- Pelish, HE; Peterson, JR; Salvarezza, SB; Rodriguez-Boulan, E; Chen, JL; Stamnes, M; Macia, E; Feng, Y; Shair, MD; Kirchhausen, T Nat Chem Biol 2: 39-46 (2006)
- Mincione, F; Starnotti, M; Menabuoni, L; Scozzafava, A; Casini, A; Supuran, CT Bioorg Med Chem Lett 11: 1787-91 (2001)
- Guryn, R; Staszewski, M; Walczy?ski, K Med Chem Res 22: 3640-3652 (2013)
- Juli, C; Sippel, M; Jäger, J; Thiele, A; Weiwad, M; Schweimer, K; Rösch, P; Steinert, M; Sotriffer, CA; Holzgrabe, U J Med Chem 54: 277-83 (2011)
- Kunkle, T; Abdeen, S; Salim, N; Ray, AM; Stevens, M; Ambrose, AJ; Victorino, J; Park, Y; Hoang, QQ; Chapman, E; Johnson, SM J Med Chem 61: 10651-10664 (2018)
- Sisay, MT; Steinmetzer, T; Stirnberg, M; Maurer, E; Hammami, M; Bajorath, J; Gütschow, M J Med Chem 53: 5523-35 (2010)
- Jones, A; Kemp, M; Stockley, M; Gibson, K; Whitlock, G US Patent US11053198 (2021)
- Moravec, J; Krystof, V; Hanus, J; Havlícek, L; Moravcová, D; Fuksová, K; Kuzma, M; Lenobel, R; Otyepka, M; Strnad, M Bioorg Med Chem Lett 13: 2993-6 (2003)
- Stucchi, M; Gmeiner, P; Huebner, H; Rainoldi, G; Sacchetti, A; Silvani, A; Lesma, G ACS Med Chem Lett 6: 882-7 (2015)
- Ioannidis, S; Lamb, ML; Wang, T; Almeida, L; Block, MH; Davies, AM; Peng, B; Su, M; Zhang, HJ; Hoffmann, E; Rivard, C; Green, I; Howard, T; Pollard, H; Read, J; Alimzhanov, M; Bebernitz, G; Bell, K; Ye, M; Huszar, D; Zinda, M J Med Chem 54: 262-76 (2011)
- Lansdell, MI; Hepworth, D; Calabrese, A; Brown, AD; Blagg, J; Burring, DJ; Wilson, P; Fradet, D; Brown, TB; Quinton, F; Mistry, N; Tang, K; Mount, N; Stacey, P; Edmunds, N; Adams, C; Gaboardi, S; Neal-Morgan, S; Wayman, C; Cole, S; Phipps, J; Lewis, M; Verrier, H; Gillon, V; Feeder, N; Heatherington, A; Sultana, S; Haughie, S; Martin, SW; Sudworth, M; Tweedy, S J Med Chem 53: 3183-97 (2010)
- Goi, T; Nakajima, T; Komatsu, Y; Kawata, A; Yamakoshi, S; Okada, O; Sugahara, M; Umeda, A; Takada, Y; Murakami, J; Ohashi, R; Watanabe, T; Fukase, K ACS Med Chem Lett 11: 1416-1420 (2020)
- Quinn, RJ; Taylor, C; Suganuma, M; Fujiki, H Bioorg Med Chem Lett 3: 1029-1034 (1993)
- Ichikawa, M; Ohtsuka, M; Ohki, H; Haginoya, N; Itoh, M; Sugita, K; Usui, H; Suzuki, M; Terayama, K; Kanda, A Bioorg Med Chem 20: 3072-93 (2012)
- Bouaboula, M; Brollo, M; Certal, V; El-Ahmad, Y; Filoche-Romme, B; Halley, F; McCort, G; Schio, L; Tabart, M; Terrier, C; Thompson, F US Patent US9714221 (2017)
- Taguchi, M; Sugimoto, K; Goda, K; Akama, T; Yamamoto, K; Suzuki, T; Tomishima, Y; Nishiguchi, M; Arai, K; Takahashi, K; Kobori, T Bioorg Med Chem Lett 13: 1963-6 (2003)
- Taha, M; Ismail, NH; Imran, S; Selvaraj, M; Rahim, A; Ali, M; Siddiqui, S; Rahim, F; Khan, KM Bioorg Med Chem 23: 7394-404 (2015)
- Sato, H; Kitagawa, O; Aida, Y; Chikazawa, J; Kurimoto, T; Takei, M; Fukuta, Y; Yoshida, K Bioorg Med Chem Lett 9: 1553-8 (1999)
- Yoshikawa, K; Yoshino, T; Yokomizo, Y; Uoto, K; Naito, H; Kawakami, K; Mochizuki, A; Nagata, T; Suzuki, M; Kanno, H; Takemura, M; Ohta, T Bioorg Med Chem Lett 21: 2133-40 (2011)
- Wan, ZK; Follows, B; Kirincich, S; Wilson, D; Binnun, E; Xu, W; Joseph-McCarthy, D; Wu, J; Smith, M; Zhang, YL; Tam, M; Erbe, D; Tam, S; Saiah, E; Lee, J Bioorg Med Chem Lett 17: 2913-20 (2007)
- Tami, M; Dale, R; Brock, S; Jocelyn, W WIPO WO2022109580 (2022)
- Zwaagstra, ME; Timmerman, H; Tamura, M; Tohma, T; Wada, Y; Onogi, K; Zhang, MQ J Med Chem 40: 1075-89 (1997)
- Wu, T; Nagle, A; Kuhen, K; Gagaring, K; Borboa, R; Francek, C; Chen, Z; Plouffe, D; Goh, A; Lakshminarayana, SB; Wu, J; Ang, HQ; Zeng, P; Kang, ML; Tan, W; Tan, M; Ye, N; Lin, X; Caldwell, C; Ek, J; Skolnik, S; Liu, F; Wang, J; Chang, J; Li, C; Hollenbeck, T; Tuntland, T; Isbell, J; Fischli, C; Brun, R; Rottmann, M; Dartois, V; Keller, T; Diagana, T; Winzeler, E; Glynne, R; Tully, DC; Chatterjee, AK J Med Chem 54: 5116-30 (2011)
- Bradner, JE; Qi, J; Tanaka, M US Patent US11406645 (2022)
- Kiyokawa, S; Hirata, Y; Nagaoka, Y; Shibano, M; Taniguchi, M; Yasuda, M; Baba, K; Uesato, S Bioorg Med Chem 18: 3925-33 (2010)
- Chatterjee, S; Dunn, D; Tao, M; Wells, G; Gu, ZQ; Bihovsky, R; Ator, MA; Siman, R; Mallamo, JP Bioorg Med Chem Lett 9: 2371-4 (1999)
- Piemontese, L; Fracchiolla, G; Carrieri, A; Parente, M; Laghezza, A; Carbonara, G; Sblano, S; Tauro, M; Gilardi, F; Tortorella, P; Lavecchia, A; Crestani, M; Desvergne, B; Loiodice, F Eur J Med Chem 90: 583-94 (2015)
- Ananthan, S; Saini, SK; Zhou, G; Hobrath, JV; Padmalayam, I; Zhai, L; Bostwick, JR; Antonio, T; Reith, ME; McDowell, S; Cho, E; McAleer, L; Taylor, M; Luedtke, RR J Med Chem 57: 7042-60 (2014)
- Carroll, C; Goldby, A; Teall, M US Patent US9475795 (2016)
- Teng, M; Nammalwar, B; Li, X; Perez, C; Yule, I; Faulkner, A; Atton, H; Parkes, A; Convers-Reignier, S; Southey, M; Puerta, DT US Patent US11407740 (2022)
- Kontopidis, G; McInnes, C; Pandalaneni, SR; McNae, I; Gibson, D; Mezna, M; Thomas, M; Wood, G; Wang, S; Walkinshaw, MD; Fischer, PM Chem Biol 13: 201-11 (2006)
- Chan, WN; Evans, JM; Hadley, MS; Herdon, HJ; Jerman, JC; Parsons, AA; Read, SJ; Stean, TO; Thompson, M; Upton, N Bioorg Med Chem Lett 9: 285-90 (1999)
- Ledneczki, I; Horváth, A; Tapolcsányi, P; Éles, J; Molnár, KD; Vágó, I; Visegrády, A; Kiss, L; Szigetvári, Á; Kóti, J; Krámos, B; Mahó, S; Holm, P; Kolok, S; Fodor, L; Thán, M; Kostyalik, D; Balázs, O; Vastag, M; Greiner, I; Lévay, G; Lendvai, B; Némethy, Z Eur J Med Chem 222: (2021)
- Schmidt, B; Lindman, S; Tong, W; Lindeberg, G; Gogoll, A; Lai, Z; Thörnwall, M; Synnergren, B; Nilsson, A; Welch, CJ; Sohtell, M; Westerlund, C; Nyberg, F; Karlén, A; Hallberg, A J Med Chem 40: 903-19 (1997)
- Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296-315 (2010)
- Kubota, K; Kurebayashi, H; Miyachi, H; Tobe, M; Onishi, M; Isobe, Y Bioorg Med Chem Lett 19: 2766-71 (2009)
- Todorov M
- Konishi, A; Tokumasu, M; Suzuki, T; Koshiba, T; Ohsumi, K; Ikehara, O; Kodama, Y US Patent US8609715 (2013)
- Syrjänen, L; Kuuslahti, M; Tolvanen, M; Vullo, D; Parkkila, S; Supuran, CT Bioorg Med Chem 23: 2303-9 (2015)
- Tomic, M; Kundakovic, M; Butorovic, B; Janac, B; Andric, D; Roglic, G; Ignjatovic, D; Kostic-Rajacic, S Bioorg Med Chem Lett 14: 4263-6 (2004)
- Carballa, DM; Seoane, S; Zacconi, F; Pérez, X; Rumbo, A; Alvarez-Díaz, S; Larriba, MJ; Pérez-Fernández, R; Muñoz, A; Maestro, M; Mouriño, A; Torneiro, M J Med Chem 55: 8642-56 (2012)
- Cirillo, PF; Hickey, ER; Moss, N; Breitfelder, S; Betageri, R; Fadra, T; Gaenzler, F; Gilmore, T; Goldberg, DR; Kamhi, V; Kirrane, T; Kroe, RR; Madwed, J; Moriak, M; Netherton, M; Pargellis, CA; Patel, UR; Qian, KC; Sharma, R; Sun, S; Swinamer, A; Torcellini, C; Takahashi, H; Tsang, M; Xiong, Z Bioorg Med Chem Lett 19: 2386-91 (2009)
- Fardis, M; Jin, H; Jabri, S; Cai, RZ; Mish, M; Tsiang, M; Kim, CU Bioorg Med Chem Lett 16: 4031-5 (2006)
- Anzai, H; Terai, T; Wakabayashi-Nakao, K; Noguchi, T; Kumachi, S; Tsuchiya, M; Nemoto, N ACS Med Chem Lett 12: 1427-1434 (2021)
- Uchida, T; Koshino, H; Takahashi, S; Shimizu, E; Takahashi, H; Yoshida, J; Shinden, H; Tsujimura, M; Kofujita, H; Uesugi, S; Kimura, KI J Nat Prod 81: 1070-1074 (2018)
- Parcella, K; Eastman, K; Yeung, KS; Grant-Young, KA; Zhu, J; Wang, T; Zhang, Z; Yin, Z; Parker, D; Mosure, K; Fang, H; Wang, YK; Lemm, J; Zhuo, X; Hanumegowda, U; Liu, M; Rigat, K; Donoso, M; Tuttle, M; Zvyaga, T; Haarhoff, Z; Meanwell, NA; Soars, MG; Roberts, SB; Kadow, JF ACS Med Chem Lett 8: 771-774 (2017)
- Harada, K; Mizukami, J; Watanabe, T; Mori, G; Ubukata, M; Suwa, K; Fukuda, S; Negoro, T; Sato, M; Inaba, T Bioorg Med Chem Lett 29: 2100-2106 (2019)
- Aoyama, Y; Uenaka, M; Konoike, T; Hayasaki-Kajiwara, Y; Naya, N; Nakajima, M Bioorg Med Chem Lett 11: 1691-4 (2001)
- Labadie, S; Dragovich, PS; Chen, J; Fauber, BP; Boggs, J; Corson, LB; Ding, CZ; Eigenbrot, C; Ge, H; Ho, Q; Lai, KW; Ma, S; Malek, S; Peterson, D; Purkey, HE; Robarge, K; Salphati, L; Sideris, S; Ultsch, M; VanderPorten, E; Wei, B; Xu, Q; Yen, I; Yue, Q; Zhang, H; Zhang, X; Zhou, A Bioorg Med Chem Lett 25: 75-82 (2015)
- Teno, N; Yamashita, Y; Masuda, A; Iguchi, Y; Oda, K; Fujimori, K; Hiramoto, T; Nishimaki-Mogami, T; Une, M; Gohda, K Bioorg Med Chem 27: 2220-2227 (2019)
- Wu, MY; Esteban, G; Brogi, S; Shionoya, M; Wang, L; Campiani, G; Unzeta, M; Inokuchi, T; Butini, S; Marco-Contelles, J Eur J Med Chem 121: 864-879 (2016)
- Guerrero, M; Urbano, M; Schaeffer, MT; Brown, S; Rosen, H; Roberts, E Bioorg Med Chem Lett 23: 614-9 (2013)
- Fernández-Bachiller, MI; Hwang, S; Schembri, ME; Lindemann, P; Guberman, M; Herziger, S; Specker, E; Matter, H; Will, DW; Czech, J; Wagner, M; Bauer, A; Schreuder, H; Ritter, K; Urmann, M; Wehner, V; Sun, H; Nazaré, M J Med Chem 65: 13013-13028 (2022)
- Mallinger, A; Schiemann, K; Rink, C; Stieber, F; Calderini, M; Crumpler, S; Stubbs, M; Adeniji-Popoola, O; Poeschke, O; Busch, M; Czodrowski, P; Musil, D; Schwarz, D; Ortiz-Ruiz, MJ; Schneider, R; Thai, C; Valenti, M; de Haven Brandon, A; Burke, R; Workman, P; Dale, T; Wienke, D; Clarke, PA; Esdar, C; Raynaud, FI; Eccles, SA; Rohdich, F; Blagg, J J Med Chem 59: 1078-101 (2016)
- Colabufo, NA; Berardi, F; Perrone, R; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A J Med Chem 51: 1415-22 (2008)
- Thaler, F; Varasi, M; Abate, A; Carenzi, G; Colombo, A; Bigogno, C; Boggio, R; Zuffo, RD; Rapetti, D; Resconi, A; Regalia, N; Vultaggio, S; Dondio, G; Gagliardi, S; Minucci, S; Mercurio, C Eur J Med Chem 64: 273-84 (2013)
- Gualtieri, MJ; Malafronte, N; Vassallo, A; Braca, A; Cotugno, R; Vasaturo, M; De Tommasi, N; Dal Piaz, F J Nat Prod 77: 596-602 (2014)
- Ledneczki, I; Horváth, A; Tapolcsányi, P; Éles, J; Molnár, KD; Vágó, I; Visegrády, A; Kiss, L; Szigetvári, Á; Kóti, J; Krámos, B; Mahó, S; Holm, P; Kolok, S; Fodor, L; Thán, M; Kostyalik, D; Balázs, O; Vastag, M; Greiner, I; Lévay, G; Lendvai, B; Némethy, Z Eur J Med Chem 222: (2021)
- de Lera Ruiz, M; Favuzza, P; Guo, Z; Zhao, L; Hu, B; Lei, Z; Zhan, D; Murgolo, N; Boyce, CW; Vavrek, M; Thompson, J; Ngo, A; Jarman, KE; Robbins, J; Boddey, J; Sleebs, BE; Lowes, KN; Cowman, AF; Olsen, DB; McCauley, JA ACS Med Chem Lett 13: 1745-1754 (2022)
- Hammitzsch, A; Tallant, C; Fedorov, O; O'Mahony, A; Brennan, PE; Hay, DA; Martinez, FO; Al-Mossawi, MH; de Wit, J; Vecellio, M; Wells, C; Wordsworth, P; Müller, S; Knapp, S; Bowness, P Proc Natl Acad Sci U S A 112: 10768-73 (2015)
- Shen, Y; Li, F; Szewczyk, MM; Halabelian, L; Chau, I; Eram, MS; Dela Seńa, C; Park, KS; Meng, F; Chen, H; Zeng, H; Dong, A; Wu, H; Trush, VV; McLeod, D; Zepeda-Velázquez, CA; Campbell, RM; Mader, MM; Watson, BM; Schapira, M; Arrowsmith, CH; Al-Awar, R; Barsyte-Lovejoy, D; Kaniskan, HÜ; Brown, PJ; Vedadi, M; Jin, J J Med Chem 64: 3697-3706 (2021)
- Vettorazzi M
- Preuss, J; Maloney, P; Peddibhotla, S; Hedrick, MP; Hershberger, P; Gosalia, P; Milewski, M; Li, YL; Sugarman, E; Hood, B; Suyama, E; Nguyen, K; Vasile, S; Sergienko, E; Mangravita-Novo, A; Vicchiarelli, M; McAnally, D; Smith, LH; Roth, GP; Diwan, J; Chung, TD; Jortzik, E; Rahlfs, S; Becker, K; Pinkerton, AB; Bode, L J Med Chem 55: 7262-72 (2012)
- Dossetter, AG; Beeley, H; Bowyer, J; Cook, CR; Crawford, JJ; Finlayson, JE; Heron, NM; Heyes, C; Highton, AJ; Hudson, JA; Jestel, A; Kenny, PW; Krapp, S; Martin, S; MacFaul, PA; McGuire, TM; Gutierrez, PM; Morley, AD; Morris, JJ; Page, KM; Ribeiro, LR; Sawney, H; Steinbacher, S; Smith, C; Vickers, M J Med Chem 55: 6363-74 (2012)
- Courme, C; Gresh, N; Vidal, M; Lenoir, C; Garbay, C; Florent, JC; Bertounesque, E Eur J Med Chem 45: 244-55 (2010)
- Wang, Y; Liu, JJ; Dransfield, PJ; Zhu, L; Wang, Z; Du, X; Jiao, X; Su, Y; Li, AR; Brown, SP; Kasparian, A; Vimolratana, M; Yu, M; Pattaropong, V; Houze, JB; Swaminath, G; Tran, T; Nguyen, K; Guo, Q; Zhang, J; Zhuang, R; Li, F; Miao, L; Bartberger, MD; Correll, TL; Chow, D; Wong, S; Luo, J; Lin, DC; Medina, JC ACS Med Chem Lett 4: 551-5 (2013)
- Shawn, C; Paul, CD; Lee, DR; Andrew, F; Magdalena, K; Yvette, LS; Timothy, LA; Vincent, M; Walter, PD; Andre, S; Mike, TM; Tao, W; Maria, WH WIPO WO2022112919 (2022)
- Lanni, TB; Greene, KL; Kolz, CN; Para, KS; Visnick, M; Mobley, JL; Dudley, DT; Baginski, TJ; Liimatta, MB Bioorg Med Chem Lett 17: 756-60 (2007)
- Papillon, JPN; Nakajima, K; Adair, CD; Hempel, J; Jouk, AO; Karki, RG; Mathieu, S; Möbitz, H; Ntaganda, R; Smith, T; Visser, M; Hill, SE; Hurtado, FK; Chenail, G; Bhang, HC; Bric, A; Xiang, K; Bushold, G; Gilbert, T; Vattay, A; Dooley, J; Costa, EA; Park, I; Li, A; Farley, D; Lounkine, E; Yue, QK; Xie, X; Zhu, X; Kulathila, R; King, D; Hu, T; Vulic, K; Cantwell, J; Luu, C; Jagani, Z J Med Chem 61: 10155-10172 (2018)
- Volgraf, M; Chan, L; Huestis, MP; Purkey, HE; Burkard, M; Geck Do, M; Harris, J; Hunt, KW; Liu, X; Lyssikatos, JP; Rana, S; Thomas, AA; Vigers, GP; Siu, M Bioorg Med Chem Lett 24: 2477-80 (2014)
- Fernández-Bachiller, MI; Hwang, S; Schembri, ME; Lindemann, P; Guberman, M; Herziger, S; Specker, E; Matter, H; Will, DW; Czech, J; Wagner, M; Bauer, A; Schreuder, H; Ritter, K; Urmann, M; Wehner, V; Sun, H; Nazaré, M J Med Chem 65: 13013-13028 (2022)
- Fukuda, M; Sasaki, T; Hashimoto, T; Miyachi, H; Waki, M; Asai, A; Takikawa, O; Ohno, O; Matsuno, K Bioorg Med Chem Lett 28: 2846-2849 (2018)
- Inoue, A; Kawai, T; Wakita, M; Iimura, Y; Sugimoto, H; Kawakami, Y J Med Chem 39: 4460-70 (1996)
- Focken, T; Burford, K; Grimwood, ME; Zenova, A; Andrez, JC; Gong, W; Wilson, M; Taron, M; Decker, S; Lofstrand, V; Chowdhury, S; Shuart, N; Lin, S; Goodchild, SJ; Young, C; Soriano, M; Tari, PK; Waldbrook, M; Nelkenbrecher, K; Kwan, R; Lindgren, A; de Boer, G; Lee, S; Sojo, L; DeVita, RJ; Cohen, CJ; Wesolowski, SS; Johnson, JP; Dehnhardt, CM; Empfield, JR J Med Chem 62: 9618-9641 (2019)
- Wang, M; Lu, J; Wang, M; Yang, CY; Wang, S J Med Chem 63: 7510-7528 (2020)
- Ishida, J; Yamamoto, H; Kido, Y; Kamijo, K; Murano, K; Miyake, H; Ohkubo, M; Kinoshita, T; Warizaya, M; Iwashita, A; Mihara, K; Matsuoka, N; Hattori, K Bioorg Med Chem 14: 1378-90 (2006)
- Tber, Z; Wartenberg, M; Jacques, JE; Roy, V; Lecaille, F; Warszycki, D; Bojarski, AJ; Lalmanach, G; Agrofoglio, LA Bioorg Med Chem 26: 4310-4319 (2018)
- Yan, VC; Yang, KL; Ballato, ES; Khadka, S; Shrestha, P; Arthur, K; Georgiou, DK; Washington, M; Tran, T; Poral, AH; Pham, CD; Yan, MJ; Muller, FL ACS Med Chem Lett 11: 1484-1489 (2020)
- Keith, JM; Jones, WM; Pierce, JM; Seierstad, M; Palmer, JA; Webb, M; Karbarz, MJ; Scott, BP; Wilson, SJ; Luo, L; Wennerholm, ML; Chang, L; Brown, SM; Rizzolio, M; Rynberg, R; Chaplan, SR; Breitenbucher, JG Bioorg Med Chem Lett 24: 737-41 (2014)
- Zhang, N; Zhang, X; Zhu, J; Turpoff, A; Chen, G; Morrill, C; Huang, S; Lennox, W; Kakarla, R; Liu, R; Li, C; Ren, H; Almstead, N; Venkatraman, S; Njoroge, FG; Gu, Z; Clausen, V; Graci, J; Jung, SP; Zheng, Y; Colacino, JM; Lahser, F; Sheedy, J; Mollin, A; Weetall, M; Nomeir, A; Karp, GM J Med Chem 57: 2121-35 (2014)
- Meena, CL; Singh, D; Weinmüller, M; Reichart, F; Dangi, A; Marelli, UK; Zahler, S; Sanjayan, GJ Bioorg Med Chem Lett 30: (2020)
- Juli, C; Sippel, M; Jäger, J; Thiele, A; Weiwad, M; Schweimer, K; Rösch, P; Steinert, M; Sotriffer, CA; Holzgrabe, U J Med Chem 54: 277-83 (2011)
- Keith, JM; Apodaca, R; Tichenor, M; Xiao, W; Jones, W; Pierce, J; Seierstad, M; Palmer, J; Webb, M; Karbarz, M; Scott, B; Wilson, S; Luo, L; Wennerholm, M; Chang, L; Brown, S; Rizzolio, M; Rynberg, R; Chaplan, S; Breitenbucher, JG ACS Med Chem Lett 3: 823-827 (2012)
- Jones, LH; Allan, G; Barba, O; Burt, C; Corbau, R; Dupont, T; Knöchel, T; Irving, S; Middleton, DS; Mowbray, CE; Perros, M; Ringrose, H; Swain, NA; Webster, R; Westby, M; Phillips, C J Med Chem 52: 1219-23 (2009)
- Moss, N; Choi, Y; Cogan, D; Flegg, A; Kahrs, A; Loke, P; Meyn, O; Nagaraja, R; Napier, S; Parker, A; Thomas Peterson, J; Ramsden, P; Sarko, C; Skow, D; Tomlinson, J; Tye, H; Whitaker, M Bioorg Med Chem Lett 19: 2206-10 (2009)
- Kochanny, MJ; Adler, M; Ewing, J; Griedel, BD; Ho, E; Karanjawala, R; Lee, W; Lentz, D; Liang, AM; Morrissey, MM; Phillips, GB; Post, J; Sacchi, KL; Sakata, ST; Subramanyam, B; Vergona, R; Walters, J; White, KA; Whitlow, M; Ye, B; Zhao, Z; Shaw, KJ Bioorg Med Chem 15: 2127-46 (2007)
- Pratt, LM; Beckett, RP; Davies, SJ; Launchbury, SB; Miller, A; Spavold, ZM; Todd, RS; Whittaker, M Bioorg Med Chem Lett 11: 2585-8 (2001)
- Kalaba, P; Aher, NY; Ili?, M; Draga?evi?, V; Wieder, M; Miklosi, AG; Zehl, M; Wackerlig, J; Roller, A; Beryozkina, T; Radoman, B; Saroja, SR; Lindner, W; Gonzalez, EP; Bakulev, V; Leban, JJ; Sitte, HH; Urban, E; Langer, T; Lubec, G J Med Chem 60: 9330-9348 (2017)
- Mollica, L; Theret, I; Antoine, M; Perron-Sierra, F; Charton, Y; Fourquez, JM; Wierzbicki, M; Boutin, JA; Ferry, G; Decherchi, S; Bottegoni, G; Ducrot, P; Cavalli, A J Med Chem 59: 7167-76 (2016)
- Krapf, MK; Gallus, J; Namasivayam, V; Wiese, M J Med Chem 61: 7952-7976 (2018)
- Burgess, A; Wigan, M; Giles, N; Depinto, W; Gillespie, P; Stevens, F; Gabrielli, B J Biol Chem 281: 9987-95 (2006)
- Wijtmans, M; Verzijl, D; Bergmans, S; Lai, M; Bosch, L; Smit, MJ; de Esch, IJ; Leurs, R Bioorg Med Chem 19: 3384-93 (2011)
- Hancock, AA; Buckner, SA; Brune, ME; Esbenshade, TA; Ireland, LM; Katwala, S; Milicic, I; Meyer, MD; Kerwin, JF; Williams, M J Pharmacol Exp Ther 300: 478-86 (2002)
- Kuduk, SD; Chang, RK; Greshock, TJ; Ray, WJ; Ma, L; Wittmann, M; Seager, MA; Koeplinger, KA; Thompson, CD; Hartman, GD; Bilodeau, MT ACS Med Chem Lett 3: 1070-1074 (2012)
- Klein, T; Abgottspon, D; Wittwer, M; Rabbani, S; Herold, J; Jiang, X; Kleeb, S; Lüthi, C; Scharenberg, M; Bezençon, J; Gubler, E; Pang, L; Smiesko, M; Cutting, B; Schwardt, O; Ernst, B J Med Chem 53: 8627-41 (2010)
- Maga, G; Falchi, F; Garbelli, A; Belfiore, A; Witvrouw, M; Manetti, F; Botta, M J Med Chem 51: 6635-8 (2008)
- Borsari, C; Jiménez-Antón, MD; Eick, J; Bifeld, E; Torrado, JJ; Olías-Molero, AI; Corral, MJ; Santarem, N; Baptista, C; Severi, L; Gul, S; Wolf, M; Kuzikov, M; Ellinger, B; Reinshagen, J; Witt, G; Linciano, P; Tait, A; Costantino, L; Luciani, R; Tejera Nevado, P; Zander-Dinse, D; Franco, CH; Ferrari, S; Moraes, CB; Cordeiro-da-Silva, A; Ponterini, G; Clos, J; Alunda, JM; Costi, MP Eur J Med Chem 183: (2019)
- Colley, HE; Muthana, M; Danson, SJ; Jackson, LV; Brett, ML; Harrison, J; Coole, SF; Mason, DP; Jennings, LR; Wong, M; Tulasi, V; Norman, D; Lockey, PM; Williams, L; Dossetter, AG; Griffen, EJ; Thompson, MJ J Med Chem 58: 9309-33 (2015)
- Buchler, I; Akuma, D; Au, V; Carr, G; de León, P; DePasquale, M; Ernst, G; Huang, Y; Kimos, M; Kolobova, A; Poslusney, M; Wei, H; Swinnen, D; Montel, F; Moureau, F; Jigorel, E; Schulze, MED; Wood, M; Barrow, JC J Med Chem 61: 9647-9665 (2018)
- Metobo, S; Mish, M; Jin, H; Jabri, S; Lansdown, R; Chen, X; Tsiang, M; Wright, M; Kim, CU Bioorg Med Chem Lett 19: 1187-90 (2009)
- Debenham, SD; Chan, A; Lau, FW; Liu, W; Wood, HB; Lemme, K; Colwell, L; Habulihaz, B; Akiyama, TE; Einstein, M; Doebber, TW; Sharma, N; Wang, CF; Wu, M; Berger, JP; Meinke, PT Bioorg Med Chem Lett 18: 4798-801 (2008)
- Flesch, D; Cheung, SY; Schmidt, J; Gabler, M; Heitel, P; Kramer, J; Kaiser, A; Hartmann, M; Lindner, M; Lüddens-Dämgen, K; Heering, J; Lamers, C; Lüddens, H; Wurglics, M; Proschak, E; Schubert-Zsilavecz, M; Merk, D J Med Chem 60: 7199-7205 (2017)
- Zehnder, L; Bennett, M; Meng, J; Huang, B; Ninkovic, S; Wang, F; Braganza, J; Tatlock, J; Jewell, T; Zhou, JZ; Burke, B; Wang, J; Maegley, K; Mehta, PP; Yin, MJ; Gajiwala, KS; Hickey, MJ; Yamazaki, S; Smith, E; Kang, P; Sistla, A; Dovalsantos, E; Gehring, MR; Kania, R; Wythes, M; Kung, PP J Med Chem 54: 3368-85 (2011)
- Xia, M; Hou, C; DeMong, DE; Pollack, SR; Pan, M; Brackley, JA; Jain, N; Gerchak, C; Singer, M; Malaviya, R; Matheis, M; Olini, G; Cavender, D; Wachter, M J Med Chem 50: 5561-3 (2007)
- Xu, P; Xu, M; Jiang, L; Yang, Q; Luo, Z; Dauter, Z; Huang, M; Andreasen, PA J Med Chem 58: 8868-76 (2015)
- Kaller, MR; Harried, SS; Albrecht, B; Amarante, P; Babu-Khan, S; Bartberger, MD; Brown, J; Brown, R; Chen, K; Cheng, Y; Citron, M; Croghan, MD; Graceffa, R; Hickman, D; Judd, T; Kriemen, C; La, D; Li, V; Lopez, P; Luo, Y; Masse, C; Monenschein, H; Nguyen, T; Pennington, LD; Miguel, TS; Sickmier, EA; Wahl, RC; Weiss, MM; Wen, PH; Williamson, T; Wood, S; Xue, M; Yang, B; Zhang, J; Patel, V; Zhong, W; Hitchcock, S ACS Med Chem Lett 3: 886-891 (2012)
- Yamada, M; Okagaki, C; Higashijima, T; Tanaka, S; Ohnuki, T; Sugita, T Bioorg Med Chem Lett 8: 1537-40 (1999)
- Yamaguchi, M; Kamei, K; Koga, T; Akima, M; Maruyama, A; Kuroki, T; Ohi, N J Med Chem 36: 4061-8 (1994)
- Hayakawa, M; Kawaguchi, K; Kaizawa, H; Koizumi, T; Ohishi, T; Yamano, M; Okada, M; Ohta, M; Tsukamoto, S; Raynaud, FI; Parker, P; Workman, P; Waterfield, MD Bioorg Med Chem 15: 5837-44 (2007)
- Ishikawa, M; Furuuchi, T; Yamauchi, M; Yokoyama, F; Kakui, N; Sato, Y Bioorg Med Chem 18: 5441-8 (2010)
- Buchanan, JL; Vu, CB; Merry, TJ; Corpuz, EG; Pradeepan, SG; Mani, UN; Yang, M; Plake, HR; Varkhedkar, VM; Lynch, BA; MacNeil, IA; Loiacono, KA; Tiong, CL; Holt, DA Bioorg Med Chem Lett 9: 2359-64 (1999)
- Kiyokawa, S; Hirata, Y; Nagaoka, Y; Shibano, M; Taniguchi, M; Yasuda, M; Baba, K; Uesato, S Bioorg Med Chem 18: 3925-33 (2010)
- Proudfoot, JR; Betageri, R; Cardozo, M; Gilmore, TA; Glynn, S; Hickey, ER; Jakes, S; Kabcenell, A; Kirrane, TM; Tibolla, AK; Lukas, S; Patel, UR; Sharma, R; Yazdanian, M; Moss, N; Beaulieu, PL; Cameron, DR; Ferland, JM; Gauthier, J; Gillard, J; Gorys, V; Poirier, M; Rancourt, J; Wernic, D; Llinas-Brunet, M J Med Chem 44: 2421-31 (2001)
- Dawson, MI; Xia, Z; Jiang, T; Ye, M; Fontana, JA; Farhana, L; Patel, B; Xue, LP; Bhuiyan, M; Pellicciari, R; Macchiarulo, A; Nuti, R; Zhang, XK; Han, YH; Tautz, L; Hobbs, PD; Jong, L; Waleh, N; Chao, WR; Feng, GS; Pang, Y; Su, Y J Med Chem 51: 5650-62 (2008)
- Hodgson, ST; Wates, PJ; Blackwell, GJ; Craig, C; Yeadon, M; Boughton-Smith, N Bioorg Med Chem Lett 3: 2565-2570 (1993)
- Kwag, R; Lee, J; Kim, D; Lee, H; Yeom, M; Woo, J; Cho, Y; Kim, HJ; Kim, J; Keum, G; Jeon, B; Choo, H J Med Chem 64: 13766-13779 (2021)
- Cheung, AW; Danho, W; Swistok, J; Qi, L; Kurylko, G; Rowan, K; Yeon, M; Franco, L; Chu, XJ; Chen, L; Yagaloff, K Bioorg Med Chem Lett 13: 133-7 (2002)
- Miwa, S; Yokota, M; Ueyama, Y; Maeda, K; Ogoshi, Y; Seki, N; Ogawa, N; Nishihata, J; Nomura, A; Adachi, T; Kitao, Y; Nozawa, K; Ishikawa, T; Ukaji, Y; Shiozaki, M ACS Med Chem Lett 12: 745-751 (2021)
- Wang, A; Prouty, CP; Pelton, PD; Yong, M; Demarest, KT; Murray, WV; Kuo, GH Bioorg Med Chem Lett 20: 1432-5 (2010)
- Yoshikawa, M; Saitoh, M; Kato, T; Nakayama, Y; Seki, T; Nakagawa, Y; Tominari, Y; Seto, M; Sasaki, Y; Okaniwa, M; Oda, T; Shibuya, A; Hidaka, K; Shiokawa, Z; Murata, S; Okabe, A; Nakada, Y; Mochizuki, M; Freeze, BS; Tawaraishi, T; Wada, Y; Greenspan, PD US Patent US11666594 (2023)
- Imbriglio, JE; Shen, DM; Liang, R; Marby, K; You, M; Youm, HW; Feng, Z; London, C; Xiong, Y; Tata, J; Verras, A; Garcia-Calvo, M; Song, X; Addona, GH; McLaren, DG; He, T; Murphy, B; Metzger, DE; Salituro, G; Deckman, D; Chen, Q; Jin, X; Stout, SJ; Wang, SP; Wilsie, L; Palyha, O; Han, S; Hubbard, BK; Previs, SF; Pinto, S; Taggart, A J Med Chem 58: 9345-53 (2015)
- Asghar, A; Yousuf, M; Mubeen, H; Nazir, R; Haruna, K; Onawole, AT; Rasheed, L Bioorg Med Chem 27: 2397-2404 (2019)
- Wang, Y; Liu, JJ; Dransfield, PJ; Zhu, L; Wang, Z; Du, X; Jiao, X; Su, Y; Li, AR; Brown, SP; Kasparian, A; Vimolratana, M; Yu, M; Pattaropong, V; Houze, JB; Swaminath, G; Tran, T; Nguyen, K; Guo, Q; Zhang, J; Zhuang, R; Li, F; Miao, L; Bartberger, MD; Correll, TL; Chow, D; Wong, S; Luo, J; Lin, DC; Medina, JC ACS Med Chem Lett 4: 551-5 (2013)
- Le Manach, C; Nchinda, AT; Paquet, T; Gonzŕlez Cabrera, D; Younis, Y; Han, Z; Bashyam, S; Zabiulla, M; Taylor, D; Lawrence, N; White, KL; Charman, SA; Waterson, D; Witty, MJ; Wittlin, S; Botha, ME; Nondaba, SH; Reader, J; Birkholtz, LM; Jiménez-Díaz, MB; Martínez, MS; Ferrer, S; Angulo-Barturen, I; Meister, S; Antonova-Koch, Y; Winzeler, EA; Street, LJ; Chibale, K J Med Chem 59: 9890-9905 (2016)
- Stefanowicz, J; S?owi?ski, T; Wróbel, MZ; Herold, F; Gomó?ka, AE; Weso?owska, A; Jastrz?bska-Wi?sek, M; Partyka, A; Andres-Mach, M; Czuczwar, SJ; ?uszczki, JJ; Zagaja, M; Siwek, A; Nowak, G; ?o?nierek, M; B?czek, T; Ulenberg, S; Belka, M; Tur?o, J Bioorg Med Chem 24: 3994-4007 (2016)
- Starck, JP; Talaga, P; Quéré, L; Collart, P; Christophe, B; Lo Brutto, P; Jadot, S; Chimmanamada, D; Zanda, M; Wagner, A; Mioskowski, C; Massingham, R; Guyaux, M Bioorg Med Chem Lett 16: 373-7 (2005)
- Kalaba, P; Aher, NY; Ili?, M; Draga?evi?, V; Wieder, M; Miklosi, AG; Zehl, M; Wackerlig, J; Roller, A; Beryozkina, T; Radoman, B; Saroja, SR; Lindner, W; Gonzalez, EP; Bakulev, V; Leban, JJ; Sitte, HH; Urban, E; Langer, T; Lubec, G J Med Chem 60: 9330-9348 (2017)
- Zhang, M; Jiang, L; Tao, J; Pan, Z; He, M; Su, D; He, G; Jiang, Q Bioorg Med Chem 27: 2268-2279 (2019)
- Zheng, M; Zheng, Y; Xue, Y; Liu, Y; An, L; Zhang, L; Ji, M; Xue, B; Wu, X; Gong, X; Gu, N; Zhan, X Chem Biol Drug Des 81: 399-407 (2013)
- Qiu, W; Zhou, M; Mazumdar, M; Azzi, A; Ghanmi, D; Luu-The, V; Labrie, F; Lin, SX J Biol Chem 282: 8368-79 (2007)
- Zhu, M; Dong, B; Zhang, GN; Wang, JX; Cen, S; Wang, YC Bioorg Med Chem Lett 29: 1541-1545 (2019)
- Smethurst, CA; Bevan, N; Brooks, C; Emmons, A; Gough, PJ; Mookherjee, C; Moores, K; Peace, S; Philp, J; Piercy, V; Watson, SP; Zippoli, M Bioorg Med Chem Lett 22: 7252-5 (2012)
- Beaufils, F; Cmiljanovic, N; Cmiljanovic, V; Bohnacker, T; Melone, A; Marone, R; Jackson, E; Zhang, X; Sele, A; Borsari, C; Mestan, J; Hebeisen, P; Hillmann, P; Giese, B; Zvelebil, M; Fabbro, D; Williams, RL; Rageot, D; Wymann, MP J Med Chem 60: 7524-7538 (2017)
- Hauck, S; Hiesinger, K; Khageh Hosseini, S; Achenbach, J; Biondi, RM; Proschak, E; Zörnig, M; Odadzic, D Bioorg Med Chem 24: 5717-5729 (2016)
- Stefanowicz, J; S?owi?ski, T; Wróbel, MZ; Herold, F; Gomó?ka, AE; Weso?owska, A; Jastrz?bska-Wi?sek, M; Partyka, A; Andres-Mach, M; Czuczwar, SJ; ?uszczki, JJ; Zagaja, M; Siwek, A; Nowak, G; ?o?nierek, M; B?czek, T; Ulenberg, S; Belka, M; Tur?o, J Bioorg Med Chem 24: 3994-4007 (2016)